BDBM50214264 1-{[(5R,8R,11S)-6,9,12-trioxo-8-(propan-2-yl)-5-{[3-(trifluoromethyl)phenyl]methyl}-3,4,5,6,7,8,9,10,11,12,13,14,15,16-tetradecahydro-2H-1,4,7,10,13-benzoxatetrazacyclooctadecin-11-yl]methyl}guanidine::CHEMBL396413
SMILES [#6]-[#6](-[#6])-[#6@H]-1-[#7]-[#6](=O)-[#6@@H](-[#6]-c2cccc(c2)C(F)(F)F)-[#7]-[#6]-[#6]-[#8]-c2ccccc2-[#6]-[#6]-[#6]-[#7]-[#6](=O)-[#6@H](-[#6]\[#7]=[#6](\[#7])-[#7])-[#7]-[#6]-1=O
InChI Key InChIKey=FOPMEOGNSDLKOM-GIFXNVAJSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50214264
Affinity DataKi: 6nMAssay Description:Displacement of [125I]-motilin from human motilin receptor expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 28nMAssay Description:Antagonist activity against human motilin receptor in aequoscreen cells assessed as inhibition of motilin induced calcium release by aequorin assayMore data for this Ligand-Target Pair