BDBM50221985 CHEMBL241010::H-Dmt-Tic-NH-CH2-CH2-NH2

SMILES Cc1cc(O)cc(C)c1C[C@H](N)C(=O)N1Cc2ccccc2CC1C(=O)NCCN

InChI Key InChIKey=VIPTXSCSZKOVSA-BGERDNNASA-N

Data  2 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50221985   

TargetDelta-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50221985(CHEMBL241010 | H-Dmt-Tic-NH-CH2-CH2-NH2)
Affinity DataKi:  1.81nMAssay Description:Displacement of [3H]deltorphin 2 from delta-opioid receptor in Sprague-Dawley rat brain P2 synaptosome membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50221985(CHEMBL241010 | H-Dmt-Tic-NH-CH2-CH2-NH2)
Affinity DataKi:  2.72nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Sprague-Dawley rat brain P2 synaptosome membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50221985(CHEMBL241010 | H-Dmt-Tic-NH-CH2-CH2-NH2)
Affinity DataIC50:  286nMAssay Description:Agonist activity at mu-opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed