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Found 2 Enz. Inhib. hit(s) with Target = 'Mu-type opioid receptor' and Ligand = 'BDBM50221985'
TargetMu-type opioid receptor(Rattus norvegicus (rat))
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50221985(CHEMBL241010 | H-Dmt-Tic-NH-CH2-CH2-NH2)
Affinity DataKi:  2.72nMAssay Description:Displacement of [3H]DAMGO from mu-opioid receptor in Sprague-Dawley rat brain P2 synaptosome membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
University Of Ferrara

Curated by ChEMBL
LigandPNGBDBM50221985(CHEMBL241010 | H-Dmt-Tic-NH-CH2-CH2-NH2)
Affinity DataIC50:  286nMAssay Description:Agonist activity at mu-opioid receptor in Hartley guinea pig ileum assessed as inhibition of electrically-stimulated muscle contractionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed