BDBM50232675 CHEMBL4100295
SMILES C[C@@]1(CO1)C(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](CO)NC(=O)c1cccc(=O)[nH]1
InChI Key InChIKey=QYDASSGXBXGRBS-CKJXQJPGSA-N
Data 10 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 50232675
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of proteasome beta2 in human MOLT4 cell lysate after 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: >2.50E+5nMAssay Description:Inhibition of MECL1 in human MOLT4 cell lysate after 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 6.89E+3nMAssay Description:Inhibition of proteasome beta5 in human MOLT4 cell lysate after 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 4.27E+3nMAssay Description:Inhibition of LMP7 in human MOLT4 cell lysate after 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of Beta5 in human 20S immunoproteasome usingAc-WLA-AMC as substrate after 1 hr by fluorescence based microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 51nMAssay Description:Inhibition of LMP2 in human MOLT4 cell lysate after 1 hr by ELISAMore data for this Ligand-Target Pair
Affinity DataIC50: 158nMAssay Description:Inhibition of LMP2 in human 20S immunoproteasome using Ac-PAL-AMC as substrate after 1 hr by fluorescence based microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4.76E+3nMAssay Description:Inhibition of Beta1 subunit in human 20S proteasome using Ac-nLPnLD-AMC as substrate after 1 hr by fluorescence based microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of LMP7 in human 20S immunoproteasome using Ac-ANW-AMC as substrate after 1 hr by fluorescence based microplate reader analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 4.64E+4nMAssay Description:Inhibition of proteasome beta1 in human MOLT4 cell lysate after 1 hr by ELISAMore data for this Ligand-Target Pair