BDBM50273370 CHEMBL503473::GWTLNSAGYLLGPPPGFSPFR-CONH2::Galanin (1-13)-bradikinin(2-9)::Galanin-(1-13)-bradykinin-(2-9)-amide::M35
SMILES CC(C)C[C@H](NC(=O)[C@H](CC(C)C)NC(=O)[C@H](Cc1ccc(O)cc1)NC(=O)CNC(=O)[C@H](C)NC(=O)[C@H](CO)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CC(C)C)NC(=O)[C@@H](NC(=O)[C@H](Cc1c[nH]c2ccccc12)NC(=O)CN)[C@@H](C)O)C(=O)NCC(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)N1CCC[C@H]1C(=O)NCC(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CO)C(=O)N1CCC[C@H]1C(=O)N[C@@H](Cc1ccccc1)C(=O)N[C@@H](CCCN=C(N)N)C(N)=O
InChI Key InChIKey=JWMXJVFGTXYBFM-AEXVMZOXSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 20 hits for monomerid = 50273370
Affinity DataKi: 0.0100nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Displacement of Eu-labeled galanin from human GalR2 by DELFIA competitive assayMore data for this Ligand-Target Pair
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical
Curated by PDSP Ki Database
Synaptic Pharmaceutical
Curated by PDSP Ki Database
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical
Curated by PDSP Ki Database
Synaptic Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKd: 0.100nMAssay Description:Binding affinity to human GalR1More data for this Ligand-Target Pair
TargetGalanin receptor type 3(Homo sapiens (Human))
Synaptic Pharmaceutical
Curated by PDSP Ki Database
Synaptic Pharmaceutical
Curated by PDSP Ki Database
Affinity DataKd: 15nMAssay Description:Binding affinity to human GalR3More data for this Ligand-Target Pair
Affinity DataKd: 2nMAssay Description:Displacement of europium-labeled galanin from human GalR2 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair