BDBM50276840 CHEMBL4160471
SMILES CCCCN(CC)c1nc(C)nc2n(-c3c(C)cc(C)cc3C)c(=N)sc12
InChI Key InChIKey=WOWDTPMKMJMTLC-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50276840
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University
Curated by ChEMBL
South Dakota State University
Curated by ChEMBL
Affinity DataEC50: 1.10nMAssay Description:Antagonist activity at human CRFR1 expressed in HEK293 cells assessed as inhibition of sauvagine-induced cAMP accumulation by measuring sauvagine EC5...More data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University
Curated by ChEMBL
South Dakota State University
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRFR1 expressed in HEK293 cell membrane homogenates after 120 mins by gamma counting methodMore data for this Ligand-Target Pair