Found 2 Enz. Inhib. hit(s) with Target = 'Corticotropin-releasing factor receptor 1' and Ligand = 'BDBM50276840' TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University
Curated by ChEMBL
South Dakota State University
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Displacement of [125I]-Tyr0-sauvagine from human CRFR1 expressed in HEK293 cell membrane homogenates after 120 mins by gamma counting methodMore data for this Ligand-Target Pair
TargetCorticotropin-releasing factor receptor 1(Homo sapiens (Human))
South Dakota State University
Curated by ChEMBL
South Dakota State University
Curated by ChEMBL
Affinity DataEC50: 1.10nMAssay Description:Antagonist activity at human CRFR1 expressed in HEK293 cells assessed as inhibition of sauvagine-induced cAMP accumulation by measuring sauvagine EC5...More data for this Ligand-Target Pair
