BDBM50323006 1'-(5-(4-chlorophenyl)-4-(2,4-dichlorophenyl)-1-(3-(methylsulfonamido)propyl)-1H-pyrrole-2-carbonyl)-4,4-difluoro-1,4'-bipiperidine-4'-carboxamide::CHEMBL1210782
SMILES CS(=O)(=O)NCCCn1c(cc(c1-c1ccc(Cl)cc1)-c1ccc(Cl)cc1Cl)C(=O)N1CCC(CC1)(N1CCC(F)(F)CC1)C(N)=O
InChI Key InChIKey=YHONTRPKANXJPY-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50323006
Affinity DataIC50: 1nMAssay Description:Binding affinity to CB1 receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Antagonist activity at CB1 receptor in forskolin-stimulated human U373-MG cells assessed as inhibition of CP-55940-induced cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataIC50: 1.40nMAssay Description:Inhibition of human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair