Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Cannabinoid receptor 1' and Ligand = 'BDBM50323006'
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50323006(1'-(5-(4-chlorophenyl)-4-(2,4-dichlorophenyl)-1-(3...)
Affinity DataIC50:  1nMAssay Description:Binding affinity to CB1 receptor in rat brain synaptosomal membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50323006(1'-(5-(4-chlorophenyl)-4-(2,4-dichlorophenyl)-1-(3...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition of human recombinant CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Sanofi-Aventis R&D

Curated by ChEMBL
LigandPNGBDBM50323006(1'-(5-(4-chlorophenyl)-4-(2,4-dichlorophenyl)-1-(3...)
Affinity DataEC50:  15nMAssay Description:Antagonist activity at CB1 receptor in forskolin-stimulated human U373-MG cells assessed as inhibition of CP-55940-induced cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed