BDBM50487259 CHEBI:64219::[3H]NEMONAPRIDE
SMILES CNc1cc(OC)c(cc1Cl)C(=O)N[C@@H]1CCN(Cc2ccccc2)[C@@H]1C
InChI Key InChIKey=KRVOJOCLBAAKSJ-RDTXWAMCSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 10 hits for monomerid = 50487259
Affinity DataKi: 0.75nMAssay Description:Displacement of [3H]-methylspiperone from dopamine D4 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Displacement of [3H]-methylspiperone from dopamine D3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 0.860nMAssay Description:Displacement of [3H]-N-Methylspiperone from human dopamine D4 receptor expressed in stable HEK cells incubated for 90 mins by microbeta counting meth...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Displacement of [3H]-N-Methylspiperone from dopamine D3 receptor (unknown origin) incubated for 90 mins by microbeta counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Displacement of [3H]N-methylspiperone from dopamine D2 receptor (unknown origin)More data for this Ligand-Target Pair
TargetSigma intracellular receptor 2(Homo sapiens (Human))
City University Of New York
Curated by ChEMBL
City University Of New York
Curated by ChEMBL
Affinity DataKi: 7.20nMAssay Description:Displacement of [3H]DTG from sigma2 receptor(unknown origin)More data for this Ligand-Target Pair
Affinity DataKd: 0.0160nMAssay Description:Binding affinity to Rattus norvegicus (rat) chimeric dopamine D2 trunk/D2 tail receptor transfected in african green monkey COS7 cells after 1 hr by ...More data for this Ligand-Target Pair
Affinity DataKd: 0.0640nMAssay Description:Binding affinity to Rattus norvegicus (rat) wild type dopamine D3 receptor transfected in african green monkey COS7 cells after 1 hr by beta scintill...More data for this Ligand-Target Pair
Affinity DataKd: 0.0140nMAssay Description:Binding affinity to Rattus norvegicus (rat) wild type dopamine D2 receptor transfected in african green monkey COS7 cells after 1 hr by beta scintill...More data for this Ligand-Target Pair
Affinity DataKd: 0.0600nMAssay Description:Binding affinity to Rattus norvegicus (rat) chimeric dopamine D3 trunk/D3 tail receptor transfected in african green monkey COS7 cells after 1 hr by ...More data for this Ligand-Target Pair