BDBM50518026 CHEMBL4449152
SMILES CC(Cc1ccsc1)NC(=O)NCC(Cc1ccccc1)N(C)C
InChI Key InChIKey=LGUNAZMQJSOQTG-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50518026
Affinity DataKi: 42nMAssay Description:Displacement of [3H]-Diprenorphine from mu opioid receptor (unknown origin) expressed in sf9 insect cell membranes after 1 hr by liquid scintillation...More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:Inhibition of mu opioid receptor (unknown origin) assessed as reduction in intracellular cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Inhibition of mu opioid receptor (unknown origin) assessed as reduction in intracellular cAMP accumulationMore data for this Ligand-Target Pair
Affinity DataEC50: 940nMAssay Description:Inhibition of mu opioid receptor (unknown origin) assessed as increase in beta arrestin 2 recruitmentMore data for this Ligand-Target Pair
Affinity DataEC50: 940nMAssay Description:Agonist activity at human mu opioid receptor expressed in HEK293T cells co-transfected with venus-tagged N-terminal beta-arrestin-2 assessed as incre...More data for this Ligand-Target Pair
Affinity DataEC50: 180nMAssay Description:Agonist activity at Gi/o coupled human mu opioid receptor expressed in HEK293T cells co-expressing luciferase based cAMP biosensor and GRK2 assessed ...More data for this Ligand-Target Pair