BDBM50536439 CHEMBL4581001
SMILES C[C@H](NC(=O)[C@H](Cc1ccccc1)NC(=O)[C@H](C[C@H]1CC[C@@H](CC1)C1CCCCC1)NC(=O)[C@H](Cc1ccccc1)N=[N+]=[N-])C(=O)[C@@]1(C)CO1
InChI Key InChIKey=PLWFGVRFZQSLKE-NKXOHJQVSA-N
Data 6 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50536439
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Leiden Institute Of Chemistry
Curated by ChEMBL
Leiden Institute Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 1.32E+4nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta5 in human Raji cells incubated for 1 hr by BODIPY(TMR)-NC-005-VS probe based co...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Leiden Institute Of Chemistry
Curated by ChEMBL
Leiden Institute Of Chemistry
Curated by ChEMBL
Affinity DataIC50: 4.90nMAssay Description:Inhibition of catalytic activity of constitutive proteasome 20s subunit beta5 in human Raji cells incubated for 1 hr by BODIPY(TMR)-NC-005-VS probe b...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Leiden Institute Of Chemistry
Curated by ChEMBL
Leiden Institute Of Chemistry
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of catalytic activity of constitutive proteasome 20s subunit beta1 in human Raji cells incubated for 1 hr by Cy5-NC-001 probe based compet...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry
Curated by ChEMBL
Leiden Institute Of Chemistry
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based compet...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Leiden Institute Of Chemistry
Curated by ChEMBL
Leiden Institute Of Chemistry
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of catalytic activity of immunoproteasome 20s subunit beta1 in human Raji cells incubated for 1 hr by Cy5-NC-001 probe based competitive a...More data for this Ligand-Target Pair
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Leiden Institute Of Chemistry
Curated by ChEMBL
Leiden Institute Of Chemistry
Curated by ChEMBL
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of catalytic activity of constitutive proteasome 20s subunit beta2 in human Raji cells incubated for 1 hr by BODIPY(FL)-LU-112 probe based...More data for this Ligand-Target Pair