BDBM50545100 CHEMBL1990482

SMILES NC(=O)c1cccc2[nH]c(nc12)-c1ccncc1

InChI Key InChIKey=CZIGMBNEFWBEMD-UHFFFAOYSA-N

Data  5 KI  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 7 hits for monomerid = 50545100   

TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataKi:  30nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataKi:  40nMAssay Description:Inhibition of His/GST-tagged PKN2 (unknown origin) using biotinylated peptide as substrate measured after 1 hr in presence of [gamma-33P]-ATP by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataKi:  540nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDual specificity protein kinase CLK4(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataKi: <1.00E+5nMAssay Description:Inhibition of His/GST-tagged CLK4 (unknown origin) using biotinylated peptide as substrate measured after 1 hr in presence of [gamma-33P]-ATP by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataKi: <1.00E+5nMAssay Description:Inhibition of His/GST-tagged PKN1 (unknown origin) using biotinylated peptide as substrate measured after 1 hr in presence of [gamma-33P]-ATP by fluo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N2(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataIC50:  64nMAssay Description:Displacement of tracer from PKN2 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase N1(Homo sapiens (Human))
University Of Sussex

Curated by ChEMBL
LigandPNGBDBM50545100(CHEMBL1990482)
Affinity DataIC50:  1.10E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed