Found 3 Enz. Inhib. hit(s) with Target = 'Serine/threonine-protein kinase N1' and Ligand = 'BDBM50545100'
Affinity DataKi: 540nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+5nMAssay Description:Inhibition of His/GST-tagged PKN1 (unknown origin) using biotinylated peptide as substrate measured after 1 hr in presence of [gamma-33P]-ATP by fluo...More data for this Ligand-Target Pair
Affinity DataIC50: 1.10E+3nMAssay Description:Displacement of tracer from PKN1 (unknown origin) by TR-FRET assayMore data for this Ligand-Target Pair