BDBM8958 10-(2-diethylaminopropyl)phenothiazine::CHEMBL1200970::CHEMBL1206::Ethopropazine::diethyl[1-(10H-phenothiazin-10-yl)propan-2-yl]amine
SMILES CCN(CC)C(C)CN1c2ccccc2Sc2ccccc12
InChI Key InChIKey=CDOZDBSBBXSXLB-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 15 hits for monomerid = 8958
Affinity DataKi: 2.47E+4nMAssay Description:Dissociation constant for enzyme-inhibitor complex of human recombinant AChE by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 2.47E+4nMAssay Description:Inhibition of human recombinant AChE assessed as dissociation constant for enzyme-inhibitor complex by Lineweaver-Burk plotMore data for this Ligand-Target Pair
Affinity DataKi: 2.50E+4nMAssay Description:Inhibition of human erythrocytes recombinant AChE assessed as dissociation constant for enzyme-inhibitor complexMore data for this Ligand-Target Pair
Affinity DataKi: 1.73E+5nM ΔG°: -5.13kcal/molepH: 8.0 T: 2°CAssay Description:Inhibition of enzyme activity was measured over a substrate concentration range of 0.01-30 mM and at least six inhibitor concentrations to determine ...More data for this Ligand-Target Pair
Affinity DataKi: 1.73E+5nMAssay Description:Inhibition of fetal Bovine serum AChEMore data for this Ligand-Target Pair
Affinity DataKi: 1.21E+7nMAssay Description:Inhibition of human erythrocytes recombinant AChE assessed as dissociation constant for enzyme-inhibitor-substrate complexMore data for this Ligand-Target Pair
Affinity DataKi: 1.21E+7nMAssay Description:Dissociation constant for enzyme-inhibitor-substrate complex of human recombinant AChE by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+6nMAssay Description:Inhibition of human recombinant AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human plasma BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 300nMAssay Description:Inhibition of human erythrocytes BChEMore data for this Ligand-Target Pair
Affinity DataIC50: 2.60E+5nMAssay Description:Inhibition of human plasma AChEMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+6nMAssay Description:Inhibition of human recombinant AChE by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 1.02E+6nMAssay Description:Inhibition of human erythrocyte recombinant AChE by modified Ellman's methodMore data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of AChE (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 260nMAssay Description:Inhibition of human erythrocytes AChEMore data for this Ligand-Target Pair