Compile Data Set for Download or QSAR
Report error Found 3171 Enz. Inhib. hit(s) with Target = 'Corticotropin-releasing factor receptor 1'
TargetCorticotropin-releasing factor receptor 1(Human)
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50276840(CHEMBL4160471)
Affinity DataEC50:  1.10nMAssay Description:Antagonist activity at human CRFR1 expressed in HEK293 cells assessed as inhibition of sauvagine-induced cAMP accumulation by measuring sauvagine EC5...More data for this Ligand-Target Pair
In Depth
Date in BDB:
5/26/2020
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50144193(Dicyclopropylmethyl-propyl-[4-(2,4,6-trimethoxy-ph...)
Affinity DataEC50:  990nMAssay Description:Effective dose against CRF stimulated cAMP production in CHO cells expressing human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50144193(Dicyclopropylmethyl-propyl-[4-(2,4,6-trimethoxy-ph...)
Affinity DataEC50:  970nMAssay Description:Effective dose against human Corticotropin releasing factor receptor 1 stimulated ACTH release from primary rat anterior pituitary cell culturesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50144204([4-(2-Chloro-4,6-dimethoxy-phenyl)-pyrimidin-2-yl]...)
Affinity DataEC50:  1.60E+3nMAssay Description:Effective dose against CRF stimulated cAMP production in CHO cells expressing human Corticotropin releasing factor receptor 1More data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Human)
South Dakota State University

Curated by ChEMBL
LigandPNGBDBM50144204([4-(2-Chloro-4,6-dimethoxy-phenyl)-pyrimidin-2-yl]...)
Affinity DataEC50:  1.10E+3nMAssay Description:Effective dose against human Corticotropin releasing factor receptor 1 stimulated ACTH release from primary rat anterior pituitary cell culturesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158951(Sauvagine derivative | CHEMBL429069)
Affinity DataEC50: >1.00E+3nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158954(Sauvagine derivative | CHEMBL442112)
Affinity DataEC50:  103nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158952(Sauvagine derivative | CHEMBL438948)
Affinity DataEC50:  64nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158958(Sauvagine derivative | CHEMBL439102)
Affinity DataEC50:  756nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158959(Sauvagine derivative | CHEMBL429719)
Affinity DataEC50:  606nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158960(Sauvagine derivative | CHEMBL428296)
Affinity DataEC50:  408nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158961(Sauvagine derivative | CHEMBL263862)
Affinity DataEC50:  103nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158963(Sauvagine derivative | CHEMBL438220)
Affinity DataEC50:  188nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158965(Sauvagine derivative | CHEMBL437089)
Affinity DataEC50:  112nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158967(Sauvagine derivative | CHEMBL414130)
Affinity DataEC50:  163nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158969(Sauvagine derivative | CHEMBL428975)
Affinity DataEC50: >1.00E+3nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158970(Sauvagine derivative | CHEMBL441564)
Affinity DataEC50: >1.00E+3nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158972(Sauvagine derivative | CHEMBL268549)
Affinity DataEC50:  404nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158971(Sauvagine derivative | CHEMBL427923)
Affinity DataEC50:  106nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158975(Sauvagine derivative | CHEMBL410814)
Affinity DataEC50:  582nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158953(Sauvagine derivative | CHEMBL438928)
Affinity DataEC50:  65nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158978(Sauvagine derivative | CHEMBL428824)
Affinity DataEC50:  78nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158977(Sauvagine derivative | CHEMBL438939)
Affinity DataEC50:  76nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158957(Sauvagine derivative | CHEMBL411961)
Affinity DataEC50: >1.00E+3nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158980(Sauvagine derivative | CHEMBL410347)
Affinity DataEC50:  98nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158968(Sauvagine derivative | CHEMBL427611)
Affinity DataEC50:  367nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158986(Sauvagine derivative | CHEMBL410568)
Affinity DataEC50:  189nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158956(Sauvagine derivative | CHEMBL409748)
Affinity DataEC50:  423nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158982(Sauvagine derivative | CHEMBL413414)
Affinity DataEC50:  48nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158989(Sauvagine derivative | CHEMBL440427)
Affinity DataEC50: >1.00E+3nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158988(Sauvagine derivative | CHEMBL412296)
Affinity DataEC50:  312nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158987(Sauvagine derivative | CHEMBL439887)
Affinity DataEC50: >1.00E+3nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158979(Sauvagine derivative | CHEMBL427811)
Affinity DataEC50:  108nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158981(Sauvagine derivative | CHEMBL429547)
Affinity DataEC50:  562nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158991(Sauvagine derivative | CHEMBL438210)
Affinity DataEC50:  608nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158973(Sauvagine derivative | CHEMBL438391)
Affinity DataEC50:  116nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158993(Sauvagine derivative | CHEMBL437289)
Affinity DataEC50:  707nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158994(Sauvagine derivative | CHEMBL436912)
Affinity DataEC50:  81nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158964(Sauvagine derivative | CHEMBL428127)
Affinity DataEC50:  221nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158983(CHEMBL439883 | E G P P I S I D L S L E L L R K M I...)
Affinity DataEC50:  18nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158990(Sauvagine derivative | CHEMBL438601)
Affinity DataEC50:  266nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158992(Sauvagine derivative | CHEMBL415130)
Affinity DataEC50:  237nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50119607(E G P P I S I D L S L E L L R K M I E I E K Q E K ...)
Affinity DataEC50:  20nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158955(Sauvagine derivative | CHEMBL414568)
Affinity DataEC50: >1.00E+3nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158962(Sauvagine derivative | CHEMBL411474)
Affinity DataEC50: >1.00E+3nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158976(Sauvagine derivative | CHEMBL429243)
Affinity DataEC50: >1.00E+3nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158974(Sauvagine derivative | CHEMBL428809)
Affinity DataEC50:  385nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158997(Sauvagine derivative | CHEMBL267635)
Affinity DataEC50:  52nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158995(Sauvagine derivative | CHEMBL264275)
Affinity DataEC50:  100nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetCorticotropin-releasing factor receptor 1(Mouse)
Procter & Gamble Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50158966(Sauvagine derivative | CHEMBL429403)
Affinity DataEC50:  325nMAssay Description:In vitro effective concentration for mouse corticotropin releasing factor 1 receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
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