Report error Found 2693 Enz. Inhib. hit(s) with Target = 'Fatty-acid amide hydrolase 1 [30-579]'
Affinity DataKi: 0.100nMAssay Description:Irreversible inhibition of recombinant rat FAAH preincubated for 3 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.100nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain homogenate using arachidonoyl-ethanolamide and anandamide [ethanolamine-1-3H] as substrate pre-incubat...More data for this Ligand-Target Pair
Affinity DataKi: 0.140nMAssay Description:Inhibitory constant determined against recombinant Fatty-acid amide hydrolase from rat expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibition of recombinant rat FAAH preincubated for 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Irreversible inhibition of recombinant rat FAAH preincubated for 3 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.170nMAssay Description:Apparent inhibition of rat FAAH using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.190nMAssay Description:Inhibition of recombinant rat FAAH preincubated for 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Time-dependent inhibition of recombinant rat FAAH expressed in Escherichia coli assessed as breakdown of [14C]-oleamide preincubated for 3 hrs by Dix...More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of rat FAAH assessed as reduction in [14C]oleamide conversion to oleic acid by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of rat FAAHMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Time-dependent inhibition of recombinant rat FAAH expressed in Escherichia coli assessed as breakdown of [14C]-oleamide preincubated for 6 hrs by Dix...More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Time-dependent inhibition of recombinant rat FAAH expressed in Escherichia coli assessed as breakdown of [14C]-oleamide preincubated for 1 hr by Dixo...More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of rat FAAHMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity for rat fatty acid amide hydrolaseMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibition of rat recombinant FAAH expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Time-dependent inhibition of recombinant rat FAAH expressed in Escherichia coli assessed as breakdown of [14C]-oleamide preincubated for 6 hrs by Dix...More data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Inhibitory constant determined against recombinant Fatty-acid amide hydrolase from rat expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataIC50: 0.230nMAssay Description:Rat FAAH was prepared from male Sprague Dawley rat brains, homogenized in a potter in 20 mM of Tris HCl pH 7.4, 0.32 M sucrose.The radiometric assay ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.230nMAssay Description:Rat FAAH was prepared from male Sprague Dawley rat brains, homogenized in a potter in 20 mM of Tris HCl pH 7.4, 0.32 M sucrose.The radiometric assay ...More data for this Ligand-Target Pair
Affinity DataIC50: 0.240nMAssay Description:Inhibition of FAAH in Wistar rat cerebral membrane by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.280nMAssay Description:Apparent inhibition of rat FAAH using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Inhibition of rat FAAH assessed as reduction in [14C]oleamide conversion to oleic acid by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.280nMAssay Description:Inhibitory constant determined against recombinant Fatty-acid amide hydrolase from rat expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMpH: 9.0Assay Description:Inhibition of rat FAAH expressed in Escherichia coli at pH 9.0More data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Inhibition of rat FAAH expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Irreversible inhibition of recombinant rat FAAH preincubated for 3 hrsMore data for this Ligand-Target Pair
Affinity DataKi: 0.290nMAssay Description:Inhibition of rat FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of FAAH in Sprague-Dawley rat brain homogenate using arachidonoyl-ethanolamide and anandamide [ethanolamine-1-3H] as substrate pre-incubat...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of rat FAAH expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Time-dependent inhibition of recombinant rat FAAH expressed in Escherichia coli assessed as breakdown of [14C]-oleamide preincubated for 3 hrs by Dix...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Time-dependent inhibition of recombinant rat FAAH expressed in Escherichia coli assessed as breakdown of [14C]-oleamide preincubated for 6 hrs by Dix...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Time-dependent inhibition of recombinant rat FAAH expressed in Escherichia coli assessed as breakdown of [14C]-oleamide preincubated for 3 hrs by Dix...More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of Wistar rat brain FAAH using [3H]-ethanolamine as substrate preincubated for 20 mins followed by substrate addition by liquid scintillat...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibition of rat FAAH assessed as reduction in [14C]oleamide conversion to oleic acid by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Time-dependent inhibition of recombinant rat FAAH expressed in Escherichia coli assessed as breakdown of [14C]-oleamide preincubated for 1 hr by Dixo...More data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Inhibition of rat FAAH using [3H]-AEA as substrate by liquid chromatography-mass spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 0.316nMpH: 9.0 T: 2°CAssay Description:The effect of the test compounds on the enzymatic hydrolysis of [3H]anandamide was evaluated by using rat brain homogenate preparations. [3H]Ethanola...More data for this Ligand-Target Pair
Affinity DataIC50: 0.331nMAssay Description:Displacement of [3H]-anandamide from rat brain FAAH after 30 mins by scintillation countingMore data for this Ligand-Target Pair
Affinity DataIC50: 0.340nMAssay Description:Apparent inhibition of rat FAAH using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.340nMpH: 9.0Assay Description:Inhibition of rat FAAH expressed in Escherichia coli at pH 9.0More data for this Ligand-Target Pair
Affinity DataKi: 0.360nMAssay Description:Irreversible inhibition of recombinant rat FAAH preincubated for 3 hrsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.360nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Inhibition of rat FAAH expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 0.390nMAssay Description:Inhibition of rat FAAH assessed as reduction in [14C]oleamide conversion to oleic acid by Lineweaver-Burk plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibition of rat FAAH expressed in CHO cell lysates assessed as arachidonyl-7-amino-4-methylcoumarin amide hydrolysis to 7-amino 4-methyl coumarin p...More data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of rat FAAHMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of rat recombinant FAAH expressed in Escherichia coliMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibition of rat FAAHMore data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Inhibition of FAAH1 in Wistar rat brain homogenates using [3H]anandamide as substrate incubated for 30 mins by liquid scintillation counting methodMore data for this Ligand-Target Pair
Affinity DataIC50: 0.430nMAssay Description:Apparent inhibition of rat FAAH using AMCAA as substrate after 30 mins by fluorescence assayMore data for this Ligand-Target Pair

































