Compile Data Set for Download or QSAR
Report error Found 96 Enz. Inhib. hit(s) with Target = 'Kallikrein-5 [D153N]'
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50124906(CHEMBL3623776)
Affinity DataKi:  2.10nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris X33 using Ac-YRSR-pNA by spectrophotometry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2016
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50125021(CHEMBL3623779)
Affinity DataKi:  5.20nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris X33 using Ac-YRSR-pNA by spectrophotometry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2016
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50154254(CHEMBL3775705)
Affinity DataIC50: 112nMAssay Description:Inhibition of human KLK5 using Abz-KLRSSKQ-EDDnp as substrate preincubated for 5 mins followed by substrate addition by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2017
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50154253(CHEMBL3775377)
Affinity DataIC50: 115nMAssay Description:Inhibition of human KLK5 using Abz-KLRSSKQ-EDDnp as substrate preincubated for 5 mins followed by substrate addition by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2017
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50154254(CHEMBL3775705)
Affinity DataKi:  120nMAssay Description:Competitive inhibition of human KLK5 using Abz-KLRSSKQ-EDDnp as substrate preincubated for 5 mins followed by substrate addition by Lineweaver-Burk p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2017
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50154252(CHEMBL3774934)
Affinity DataIC50: 122nMAssay Description:Inhibition of human KLK5 using Abz-KLRSSKQ-EDDnp as substrate preincubated for 5 mins followed by substrate addition by spectrofluorimetric analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2017
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50154253(CHEMBL3775377)
Affinity DataKi:  130nMAssay Description:Competitive inhibition of human KLK5 using Abz-KLRSSKQ-EDDnp as substrate preincubated for 5 mins followed by substrate addition by Lineweaver-Burk p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2017
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50154252(CHEMBL3774934)
Affinity DataKi:  130nMAssay Description:Competitive inhibition of human KLK5 using Abz-KLRSSKQ-EDDnp as substrate preincubated for 5 mins followed by substrate addition by Lineweaver-Burk p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/6/2017
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM51911(3-(2-methoxyphenyl)-3-(4-methoxyphenyl)-N-[(4-prop...)
Affinity DataIC50: 140nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113060(US9695194, 1)
Affinity DataKi:  200nM ΔG°:  -39.8kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM32709(1-(4-methylbenzoyl)-3-(3-pyridinyl)-1H-1,2,4-triaz...)
Affinity DataIC50: 270nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446220(CHEMBL3109164)
Affinity DataKi:  300nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50125044(CHEMBL3623790)
Affinity DataKi:  362nMAssay Description:Inhibition of KLK5 (unknown origin) expressed in Pichia pastoris X33 using Ac-YRSR-pNA by spectrophotometry methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/11/2016
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446221(CHEMBL3109163)
Affinity DataKi:  400nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113299(US9695194, 15)
Affinity DataKi:  500nM ΔG°:  -37.4kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113069(US9695194, 5)
Affinity DataKi:  500nM ΔG°:  -37.4kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113065(US9695194, 2)
Affinity DataKi:  500nM ΔG°:  -37.4kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113067(US9695194, 3)
Affinity DataKi:  600nM ΔG°:  -36.9kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446218(CHEMBL3109166)
Affinity DataKi:  600nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113297(US9695194, 14)
Affinity DataKi:  600nM ΔG°:  -36.9kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113296(US9695194, 13)
Affinity DataKi:  600nM ΔG°:  -36.9kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446219(CHEMBL3109165)
Affinity DataKi:  700nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM33453((3-Amino-[1,2,4]triazol-4-yl)-(4-methoxy-phenyl)-m...)
Affinity DataIC50: 990nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113119(US9695194, 6)
Affinity DataKi:  1.00E+3nM ΔG°:  -35.6kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113283(US9695194, 8)
Affinity DataKi:  1.00E+3nM ΔG°:  -35.6kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113301(US9695194, 17)
Affinity DataKi:  1.00E+3nM ΔG°:  -35.6kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113295(US9695194, 12)
Affinity DataKi:  1.00E+3nM ΔG°:  -35.6kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113300(US9695194, 16)
Affinity DataKi:  1.00E+3nM ΔG°:  -35.6kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113068(US9695194, 4)
Affinity DataKi:  1.00E+3nM ΔG°:  -35.6kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM33882(SMR000306508 | (5-azanyl-3-pyridin-3-yl-1,2,4-tria...)
Affinity DataIC50: 1.14E+3nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113292(US9695194, 9)
Affinity DataKi:  1.30E+3nM ΔG°:  -34.9kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM33437(MLS000099650 | SMR000074479 | 1-(3,4-dimethoxybenz...)
Affinity DataIC50: 1.30E+3nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446228(CHEMBL3109061)
Affinity DataKi:  1.70E+3nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113293(US9695194, 10)
Affinity DataKi:  1.90E+3nM ΔG°:  -34.0kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113248(US9695194, 7)
Affinity DataKi:  2.20E+3nM ΔG°:  -33.6kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446211(CHEMBL3109058)
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446224(CHEMBL3109160)
Affinity DataKi:  2.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446229(CHEMBL3109060)
Affinity DataKi:  3.40E+3nMAssay Description:Competitive inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446220(CHEMBL3109164)
Affinity DataIC50: 3.70E+3nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446221(CHEMBL3109163)
Affinity DataIC50: 3.90E+3nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM32709(1-(4-methylbenzoyl)-3-(3-pyridinyl)-1H-1,2,4-triaz...)
Affinity DataKi:  4.40E+3nMAssay Description:Inhibition of human kallikrein 5 measured after 15 mins at pH 8 by double-reciprocal plot analysisMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50289001(2-(2-Iodo-phenyl)-6,7-dimethoxy-benzo[d][1,3]oxazi...)
Affinity DataKi:  4.50E+3nM ΔG°:  -31.7kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446218(CHEMBL3109166)
Affinity DataIC50: 4.70E+3nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446219(CHEMBL3109165)
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50302107(Grassystatin A | CHEMBL567893)
Affinity DataIC50: 1.00E+4nMAssay Description:Inhibition of kallikrein 5 after 10 to 15 mins by fluorescence assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/26/2012
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM113294(US9695194, 11)
Affinity DataKi: >1.00E+4nM ΔG°: >-29.7kJ/molepH: 8.0 T: 2°CAssay Description:Materials: Recombinant human KLK5, Substrate S-2288 (Chromogenics, cat. no. 820852) KLK5 activity was determined at 37° C. in 0.1 M Tris, pH 8.0,...More data for this Ligand-Target Pair
In Depth
Date in BDB:
1/26/2018
Entry Details
US Patent

TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446228(CHEMBL3109061)
Affinity DataIC50: 1.18E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50292533(Fukugetin | CHEMBL446790)
Affinity DataIC50: 1.25E+4nMAssay Description:Inhibition of human tissue kallikrein-5 expressed in baculovirus infected insect cells using Abz-KLRSSQ-EDDnp as substrate preincubated for 10 mins f...More data for this Ligand-Target Pair
In Depth
Date in BDB:
6/26/2017
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446211(CHEMBL3109058)
Affinity DataIC50: 1.33E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
TargetKallikrein-5 [D153N](Human)
Queensland University of Technology

Curated by ChEMBL
LigandPNGBDBM50446224(CHEMBL3109160)
Affinity DataIC50: 1.55E+4nMAssay Description:Inhibition of human recombinant KLK5 expressed in baculovirus-infected insect cell system using Abz-KLRSSKQ-Eddnp as substrate incubated for 5 mins p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
7/25/2014
Entry Details Article
PubMed
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