Report error Found 136 Enz. Inhib. hit(s) with Target = 'Lutropin-choriogonadotropic hormone receptor'
Affinity DataKi: 0.0182nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 0.0245nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0427nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0776nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.0933nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.155nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.186nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.209nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.282nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 0.311nMAssay Description:Displacement of [125I]hCG from LH receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.380nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 0.457nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 0.525nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataEC50: 1nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 1.90nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 4.60nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataEC50: 5nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 9.30nMAssay Description:Negative logarithm of equilibrium dissociation constant in the rat pituitary luteinizing releasing hormone receptor binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataEC50: 10nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataKi: 17nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataEC50: 20nMAssay Description:Agonist activity at human LH receptor expressed in CHO cells assessed as production of cAMP after 60 mins by SPAMore data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Antagonist activity at rat luteinizing hormone receptor expressed in rat ovary granulosa GLHR15 cell suspension assessed as reduction in agonist-indu...More data for this Ligand-Target Pair
Affinity DataEC50: 24nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataKi: 25nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataEC50: 27nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataKi: 36nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataKi: 37nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataEC50: 39nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataKi: 42nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataEC50: 43nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Antagonist activity at rat luteinizing hormone receptor expressed in rat ovary granulosa GLHR15 cell suspension assessed as reduction in agonist-indu...More data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:In vitro binding affinity for Luteinizing hormone releasing hormone receptor from rat pituitary cells, expressed as negative logarithm of the equilib...More data for this Ligand-Target Pair
Affinity DataEC50: 55nMAssay Description:Agonist activity at human LH receptor expressed in CHO-K1 cells assessed as stimulation of luciferase activity by CRE-driven luciferase reporter gene...More data for this Ligand-Target Pair
















































