Compile Data Set for Download or QSAR
Report error Found 170 Enz. Inhib. hit(s) with Target = 'Nuclear receptor subfamily 1 group D member 1'
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630585(CHEMBL5434615)
Affinity DataEC50:  6nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630586(CHEMBL5408866)
Affinity DataEC50:  7nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630556(CHEMBL5419854)
Affinity DataEC50:  10nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630557(CHEMBL5424373)
Affinity DataEC50:  20nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630555(CHEMBL5417493)
Affinity DataEC50:  20nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630583(CHEMBL5407367)
Affinity DataEC50:  25nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630584(CHEMBL5404180)
Affinity DataEC50:  40nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50560410(CHEMBL4761268)
Affinity DataEC50:  50nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630567(CHEMBL5436011)
Affinity DataEC50:  50nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434026(CHEMBL2381196)
Affinity DataEC50:  50nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630582(CHEMBL5424215)
Affinity DataEC50:  54nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434038(CHEMBL2381198)
Affinity DataEC50:  63nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50560409(CHEMBL4781178)
Affinity DataEC50:  68nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630561(CHEMBL5439268)
Affinity DataEC50:  70nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630569(CHEMBL5412941)
Affinity DataEC50:  70nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50383675(CHEMBL2030074)
Affinity DataEC50:  77nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by BMAL1-luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50383675(CHEMBL2030074)
Affinity DataEC50:  77nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50383675(CHEMBL2030074)
Affinity DataEC50:  77nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630565(CHEMBL5434147)
Affinity DataEC50:  80nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50383674(CHEMBL2030073)
Affinity DataEC50:  97nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434025(CHEMBL2381197)
Affinity DataEC50:  100nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630588(CHEMBL5432192)
Affinity DataEC50:  110nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50383678(CHEMBL2030077)
Affinity DataEC50:  120nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630564(CHEMBL5435001)
Affinity DataEC50:  120nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50383673(CHEMBL2030072)
Affinity DataEC50:  120nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630578(CHEMBL5438917)
Affinity DataEC50:  123nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50383676(CHEMBL2030075)
Affinity DataEC50:  140nMAssay Description:Agonist activity at Rev-erbalpha assessed as repression of transcription by luciferase-reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
2/7/2013
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50383676(CHEMBL2030075)
Affinity DataEC50:  140nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by BMAL1-luciferase reporter assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50383676(CHEMBL2030075)
Affinity DataEC50:  140nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50560414(CHEMBL4763333)
Affinity DataEC50:  150nMAssay Description:Inverse agonist activity at Rev-Erb alpha LBD (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50630558(CHEMBL5429567)
Affinity DataEC50:  160nMAssay Description:Agonist activity at his6-tagged human REV-ERBalpha LBD (281 to 614 residues) expressed in Escherichia coli assessed as increase in SMRT corepressor p...More data for this Ligand-Target Pair
In Depth
Date in BDB:
12/20/2024
Entry Details
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434042(CHEMBL2381200)
Affinity DataEC50:  160nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434031(CHEMBL2381201)
Affinity DataEC50:  160nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434030(CHEMBL2381202)
Affinity DataEC50:  160nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434030(CHEMBL2381202)
Affinity DataEC50:  160nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434041(CHEMBL2381199)
Affinity DataEC50:  160nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434039(CHEMBL2381193)
Affinity DataEC50:  200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434039(CHEMBL2381193)
Affinity DataEC50:  200nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434036(CHEMBL2381204)
Affinity DataEC50:  200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434034(CHEMBL2381205)
Affinity DataEC50:  200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434037(CHEMBL2381208)
Affinity DataEC50:  200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434045(CHEMBL2381214)
Affinity DataEC50:  200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434037(CHEMBL2381208)
Affinity DataEC50:  200nMAssay Description:Agonist activity at Rev-Erb alpha (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434035(CHEMBL2381203)
Affinity DataEC50:  200nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM643202(US20240002380, Example 70)
Affinity DataIC50: 250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM50434033(CHEMBL2381209)
Affinity DataEC50:  250nMAssay Description:Agonist activity at biotinylated REV-ERBalpha (unknown origin) assessed as increase in biotinylated NCOR peptide recruitment after 1 hr by FRET assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/13/2014
Entry Details Article
PubMed
TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM643179(US20240002380, Example 5)
Affinity DataIC50: 250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM643200(US20240002380, Example 62)
Affinity DataIC50: 250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM643184(US20240002380, Example 17)
Affinity DataIC50: 250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

TargetNuclear receptor subfamily 1 group D member 1(Human)
The Scripps Research Institute

Curated by ChEMBL
LigandPNGBDBM643186(US20240002380, Example 22)
Affinity DataIC50: 250nMAssay Description:The capacity for compounds to function as ligands for either REV-ERBα or REV-ERBβ was assessed using a fluorescent resonance energy transfe...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/28/2024
Entry Details
US Patent

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