Compile Data Set for Download or QSAR
Report error Found 7 Enz. Inhib. hit(s) with Target = 'Sodium channel protein type 1 subunit alpha [1489-1708]'
TargetSodium channel protein type 1 subunit alpha [1489-1708](Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50118518(CHEMBL3617066)
Affinity DataKd:  290nMAssay Description:Inhibition of mouse NaV1.1 channel by two-electrode voltage-clamp methodMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/1/2016
Entry Details Article
PubMed
TargetSodium channel protein type 1 subunit alpha [1489-1708](Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50130535(CHEMBL3632695)
Affinity DataIC50: 670nMAssay Description:Inhibition of mouse NaV1.1 by IonWorks quattro automated electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetSodium channel protein type 1 subunit alpha [1489-1708](Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50130524(CHEMBL3634332)
Affinity DataIC50: 690nMAssay Description:Inhibition of mouse NaV1.1 by IonWorks quattro automated electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetSodium channel protein type 1 subunit alpha [1489-1708](Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50130510(CHEMBL3632698)
Affinity DataIC50: 2.40E+3nMAssay Description:Inhibition of mouse NaV1.1 by IonWorks quattro automated electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetSodium channel protein type 1 subunit alpha [1489-1708](Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50130521(CHEMBL3634329)
Affinity DataIC50: 3.10E+3nMAssay Description:Inhibition of mouse NaV1.1 by IonWorks quattro automated electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetSodium channel protein type 1 subunit alpha [1489-1708](Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50117271(CHEMBL558 | 2-(2,6-Dimethyl-phenoxy)-1-methyl-ethy...)
Affinity DataIC50: 2.10E+4nMAssay Description:Inhibition of mouse NaV1.1 by IonWorks quattro automated electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed
TargetSodium channel protein type 1 subunit alpha [1489-1708](Mouse)
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50130527(CHEMBL3634334)
Affinity DataIC50: 3.40E+4nMAssay Description:Inhibition of mouse NaV1.1 by IonWorks quattro automated electrophysiology assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/17/2016
Entry Details Article
PubMed