Compile Data Set for Download or QSAR
Report error Found 2178 Enz. Inhib. hit(s) with Target = 'Vasopressin V2 receptor'
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM35723(N-[4-(7-Chloro-5-hydroxy-2,3,4,5-tetrahydro-benzo[...)
Affinity DataIC50: 0.00700nMAssay Description:Antagonist activity at human AVPR2 by PathHunter beta-arrestin assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/28/2022
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM301678(US10131692, Compound 10)
Affinity DataEC50:  0.0200nMAssay Description:Agonist activity at recombinant rat V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205308(CHEMBL1429 | (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino...)
Affinity DataEC50:  0.0300nMAssay Description:Agonist activity at recombinant rat V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM301689(US10131692, Compound 21)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at recombinant rat V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ge...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50044777(CHEBI:34543 | Arginine Vasopressin | Beta-Hypopham...)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at human vasopressin V2 expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2016
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50205304(dVDAVP | CHEMBL435323)
Affinity DataEC50:  0.0500nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301678(US10131692, Compound 10)
Affinity DataEC50:  0.0700nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301693(US10131692, Compound 25)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50525073(CHEMBL4454891)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301701(US10131692, Compound 33)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50525084(CHEMBL4528032)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301676(US10131692, Compound 8)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301669(US10131692, Compound 1)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301699(US10131692, Compound 31)
Affinity DataEC50:  0.100nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50525085(CHEMBL4536454)
Affinity DataEC50:  0.110nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301708(US10131692, Compound 40)
Affinity DataEC50:  0.120nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50525079(CHEMBL4532363)
Affinity DataEC50:  0.140nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50525077(CHEMBL4472007)
Affinity DataEC50:  0.170nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50525086(CHEMBL4459424)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50525078(CHEMBL4444891)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301681(US10131692, Compound 13)
Affinity DataEC50:  0.190nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50146577(spirobenzoxazines analogues | CHEMBL102311)
Affinity DataIC50: 0.200nMAssay Description:In vitro inhibitory concentration against [3H]AVP binding to cloned human vasopressin receptorMore data for this Ligand-Target Pair
In Depth
Date in BDB:
11/10/2009
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50205308(CHEMBL1429 | (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50525076(CHEMBL4571464)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205305(d[Arg4]AVP | CHEMBL375324)
Affinity DataKi:  0.200nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50205308(CHEMBL1429 | (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino...)
Affinity DataEC50:  0.200nMAssay Description:Agonist activity at human vasopressin V2 expressed in HEK293 cells after 5 hrs by firefly luciferase reporter gene assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
3/21/2016
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301680(US10131692, Compound 12)
Affinity DataEC50:  0.210nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301703(US10131692, Compound 35)
Affinity DataEC50:  0.210nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301686(US10131692, Compound 18)
Affinity DataEC50:  0.220nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301673(US10131692, Compound 5)
Affinity DataEC50:  0.220nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301709(US10131692, Compound 41)
Affinity DataEC50:  0.220nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301684(US10131692, Compound 27 | US10131692, Compound 16)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301679(US10131692, Compound 11)
Affinity DataEC50:  0.230nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301689(US10131692, Compound 21)
Affinity DataEC50:  0.25nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301682(US10131692, Compound 14)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205304(dVDAVP | CHEMBL435323)
Affinity DataKi:  0.260nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50525074(CHEMBL4555263)
Affinity DataEC50:  0.260nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301694(US10131692, Compound 26)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50525082(CHEMBL4451692)
Affinity DataEC50:  0.270nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50525081(CHEMBL4462616)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301671(US10131692, Compound 3)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301687(US10131692, Compound 19)
Affinity DataEC50:  0.290nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205300(d[Val4]AVP | CHEMBL221436)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Rat)
Ferring Research Institute

Curated by ChEMBL
LigandPNGBDBM50205308(CHEMBL1429 | (S)-1-((4R,7S,10S,13S,16S)-7-(2-amino...)
Affinity DataKi:  0.300nMAssay Description:Displacement of [3H]AVP from vasopressin V2 receptor in rat kidney membranesMore data for this Ligand-Target Pair
In Depth
Date in BDB:
12/9/2012
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM50525083(CHEMBL4439313)
Affinity DataEC50:  0.300nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301707(US10131692, Compound 39)
Affinity DataEC50:  0.310nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301675(US10131692, Compound 7)
Affinity DataEC50:  0.310nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301698(US10131692, Compound 30)
Affinity DataEC50:  0.320nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301672(US10131692, Compound 4)
Affinity DataEC50:  0.330nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
TargetVasopressin V2 receptor(Human)
University of Florida

Curated by ChEMBL
LigandPNGBDBM301692(US10131692, Compound 24)
Affinity DataEC50:  0.350nMAssay Description:Agonist activity at recombinant human V2 receptor expressed in HEK293 cells measured after 5 hrs by cAMP response element driven luciferase reporter ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/24/2021
Entry Details Article
PubMed
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