Compile Data Set for Download or QSAR
Report error Found 110 Enz. Inhib. hit(s) with Target = 'tRNA (guanine-N(1)-)-methyltransferase'
TargettRNA (guanine-N(1)-)-methyltransferase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519348(CHEMBL4517402)
Affinity DataKd:  3.10E+3nMAssay Description:Binding affinity to full length Staphylococcus aureus tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surface pla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataKd:  1.04E+4nMAssay Description:Binding affinity to full length Mycobacterium tuberculosis tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surfac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519348(CHEMBL4517402)
Affinity DataKd:  190nMAssay Description:Binding affinity to full length Mycobacterium tuberculosis tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surfac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Mycobacterium tuberculosis (strain ATCC 25618 / H3...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataKd:  1.01E+4nMAssay Description:Binding affinity to full length Mycobacterium tuberculosis tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surfac...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataKd:  3.30E+3nMAssay Description:Binding affinity to full length Staphylococcus aureus tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surface pla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50009672(AdoHcy | S-[1-(adenin-9-yl)-1,5-dideoxy-beta-D-rib...)
Affinity DataKd:  5.90E+3nMAssay Description:Binding affinity to Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataKd:  91nMAssay Description:Binding affinity to Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Staphylococcus aureus (strain NCTC 8325 / PS 47))
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataKd:  2.75E+4nMAssay Description:Binding affinity to full length Staphylococcus aureus tRNA (guanine(37)-N1)-methyltransferase expressed in Escherichia coli BL21 (DE3) by surface pla...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519348(CHEMBL4517402)
Affinity DataKd:  1.60nMAssay Description:Binding affinity to Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) ...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM225673(GTC000445A)
Affinity DataKd:  1.30E+3nMAssay Description:Binding affinity to Escherichia coli TrmD by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613254(CHEMBL5271824)
Affinity DataKd:  4.20E+5nMAssay Description:Binding affinity to Escherichia coli TrmD by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613255(CHEMBL5283966)
Affinity DataKd:  2.60E+5nMAssay Description:Binding affinity to Escherichia coli TrmD by surface plasmon resonance assayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225676(GTC000449A)
Affinity DataIC50: 5.01nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2017
Entry Details
D3R
PDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225677(GTC000450A)
Affinity DataIC50: 5.01nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2017
Entry Details
D3R
PDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613268(CHEMBL5275681)
Affinity DataIC50: 9nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613266(CHEMBL5268562)
Affinity DataIC50: 11nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613282(CHEMBL5270264)
Affinity DataIC50: 13nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519348(CHEMBL4517402)
Affinity DataIC50: 24nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519370(CHEMBL4513615)
Affinity DataIC50: 25nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613267(CHEMBL5276443)
Affinity DataIC50: 27nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613281(CHEMBL5270195)
Affinity DataIC50: 36nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613279(CHEMBL5290255)
Affinity DataIC50: 37nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613283(CHEMBL5271729)
Affinity DataIC50: 38nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613280(CHEMBL5276347)
Affinity DataIC50: 39nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613269(CHEMBL5291180)
Affinity DataIC50: 50nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519348(CHEMBL4517402)
Affinity DataIC50: 60nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 Rosetta (DE3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519358(CHEMBL4447065)
Affinity DataIC50: 80nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519366(CHEMBL4463176)
Affinity DataIC50: 85nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613284(CHEMBL5269867)
Affinity DataIC50: 96nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519347(CHEMBL4555967)
Affinity DataIC50: 110nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519357(CHEMBL4543513)
Affinity DataIC50: 110nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM225684(GTC000457A)
Affinity DataIC50: 110nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613285(CHEMBL5277663)
Affinity DataIC50: 120nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519346(CHEMBL4580116)
Affinity DataIC50: 130nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613270(CHEMBL5288117)
Affinity DataIC50: 130nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519367(CHEMBL4437560)
Affinity DataIC50: 140nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613257(CHEMBL5268458)
Affinity DataIC50: 140nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519354(CHEMBL4469887)
Affinity DataIC50: 150nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225678(GTC000451A)
Affinity DataIC50: 158nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2017
Entry Details
D3R
PDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataIC50: 180nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225684(GTC000457A)
Affinity DataIC50: 200nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2017
Entry Details
D3R
PDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Haemophilus influenzae (strain ATCC 51907 / DSM 11...)
D3R/Abbott

LigandPNGBDBM225687(GTC000460A)
Affinity DataIC50: 200nMAssay Description:ScintillationProximity_AssayMore data for this Ligand-Target Pair
In Depth
Date in BDB:
5/10/2017
Entry Details
D3R
PDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519355(CHEMBL4460223)
Affinity DataIC50: 210nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519348(CHEMBL4517402)
Affinity DataIC50: 260nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 Rosetta (DE3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613265(CHEMBL5279532)
Affinity DataIC50: 270nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613260(CHEMBL5289815)
Affinity DataIC50: 310nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Escherichia coli (strain K12))
Infex Therapeutics

Curated by ChEMBL
LigandPNGBDBM50613278(CHEMBL5287055)
Affinity DataIC50: 310nMAssay Description:Inhibition of Escherichia coli TrmDMore data for this Ligand-Target Pair
In Depth
Date in BDB:
4/22/2024
Entry Details
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519349(CHEMBL2431997)
Affinity DataIC50: 330nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 Rosetta (DE3...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMedPDB3D3D Structure (crystal)
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519352(CHEMBL4458857)
Affinity DataIC50: 370nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
TargettRNA (guanine-N(1)-)-methyltransferase(Pseudomonas aeruginosa (strain ATCC 15692 / PAO1 /...)
Singapore-Mit Alliance For Research and Technology

Curated by ChEMBL
LigandPNGBDBM50519363(CHEMBL4544475)
Affinity DataIC50: 380nMAssay Description:Inhibition of Pseudomonas aeruginosa tRNA (guanine(37)-N1)-methyltransferase (Leu5 to Asp25 residues) expressed in Escherichia coli BL21 (DE3) Rosett...More data for this Ligand-Target Pair
In Depth
Date in BDB:
2/23/2021
Entry Details Article
PubMed
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