1687 SMILES Strings for Epithelial discoidin domain-containing receptor 1

Compound Name
SMILES String
Brc1cccc2N(CC(=O)N3C4CCC3COC4)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Brc1cccc2N(CC(=O)N3C4CCC3COC4)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c12 |THB:8:10:12.13:15.17.16|
Brc1cccc2N(CC(=O)N3C4CCC3COC4)C(=O)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)c12 |THB:8:10:12.13:15.17.16|
Brc1cccc2N(CC(=O)N3CC4CCCN4C(=O)C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Brc1cccc2N(CC(=O)N3CCC4CCCC34)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Brc1cccc2N(CC(=O)N3CCCCC3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Brc1cccc2N(CC(=O)N3CCC[C@H]3C#N)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12 |r|
Brc1cccc2N(CC(=O)N3CCN4CCCC4C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Brc1cccc2N(CC(=O)N3CCOc4ccccc34)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Brc1cccc2N(CC(=O)N3CCc4[nH]ccc4C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Brc1cccc2N(CC(=O)N3CCc4ccccc34)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Brc1cccc2N(CC(=O)N3CCn4cccc4C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Brc1cccc2N(CC(=O)N3C[C@@H]4CCC[C@@H]4C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12 |r|
Brc1cccc2N(CC(=O)Nc3ccccc3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Brc1cccc2N(CC(=O)Nc3ccccc3CN3CCOCC3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Brc1cccc2N(CC(=O)Nc3ccccn3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
CC(=O)Nc1ccc(cc1)-n1nc2c(c1-c1oc3cc(ccc3c1C)C(=O)NC1CCCCC1)c(N)n[nH]c2=O |(51.49,-18.77,;50.72,-17.43,;49.18,-17.44,;51.48,-16.1,;50.71,-14.77,;49.16,-14.77,;48.39,-13.44,;49.16,-12.1,;50.69,-12.1,;51.47,-13.42,;48.39,-10.77,;46.87,-10.62,;46.55,-9.13,;47.87,-8.36,;49,-9.38,;50.51,-9.05,;51.13,-7.64,;52.66,-7.8,;53.79,-6.78,;55.25,-7.24,;55.58,-8.74,;54.44,-9.77,;52.98,-9.3,;51.66,-10.08,;51.5,-11.61,;56.39,-6.2,;56.06,-4.7,;57.86,-6.67,;58.99,-5.63,;60.47,-6.11,;61.6,-5.08,;61.28,-3.57,;59.82,-3.1,;58.67,-4.13,;47.87,-6.82,;49.2,-6.06,;46.54,-6.04,;45.21,-6.82,;45.21,-8.36,;43.88,-9.14,)|
CC(=O)Nc1ccc(cc1)-n1nc2c(c1-c1oc3cc(ccc3c1C)C(=O)Nc1ccc(cc1)C(F)(F)F)c(N)n[nH]c2=O |(31.09,-19.53,;30.32,-18.2,;28.77,-18.2,;31.08,-16.86,;30.3,-15.53,;28.76,-15.53,;27.99,-14.2,;28.76,-12.86,;30.29,-12.86,;31.07,-14.18,;27.99,-11.53,;26.47,-11.38,;26.15,-9.89,;27.47,-9.12,;28.6,-10.14,;30.11,-9.81,;30.73,-8.4,;32.26,-8.56,;33.39,-7.53,;34.85,-8,;35.18,-9.5,;34.04,-10.53,;32.58,-10.06,;31.26,-10.84,;31.1,-12.37,;35.99,-6.96,;35.66,-5.46,;37.46,-7.43,;38.6,-6.39,;40.06,-6.86,;41.2,-5.83,;40.87,-4.32,;39.4,-3.86,;38.26,-4.89,;42.01,-3.28,;43.48,-3.75,;41.68,-1.78,;43.09,-2.18,;27.47,-7.58,;28.8,-6.81,;26.14,-6.8,;24.81,-7.58,;24.81,-9.12,;23.48,-9.89,)|
CC(=O)Nc1ccc(cc1)-n1nc2c(c1-c1oc3cc(ccc3c1C)C(=O)Nc1cccc(c1)C(F)(F)F)c(N)n[nH]c2=O |(21.52,-24.11,;22.28,-22.79,;23.81,-22.79,;21.52,-21.47,;20,-21.46,;19.22,-20.12,;17.69,-20.12,;16.92,-21.45,;17.68,-22.79,;19.22,-22.8,;15.38,-21.44,;14.48,-22.67,;13.03,-22.2,;13.04,-20.67,;14.49,-20.21,;14.97,-18.74,;14.07,-17.49,;14.98,-16.25,;14.66,-14.76,;15.8,-13.73,;17.26,-14.21,;17.58,-15.71,;16.43,-16.73,;16.43,-18.27,;17.68,-19.18,;15.48,-12.23,;14.02,-11.75,;16.63,-11.2,;16.31,-9.69,;17.46,-8.66,;17.14,-7.16,;15.67,-6.68,;14.53,-7.72,;14.85,-9.22,;13.06,-7.24,;11.92,-8.28,;11.56,-6.84,;12.73,-5.74,;11.71,-19.89,;11.72,-18.35,;10.36,-20.65,;10.36,-22.19,;11.69,-22.97,;11.68,-24.51,)|
CC(=O)Nc1ccc(cc1)-n1nc2c(c1-c1oc3cc(ccc3c1C)C(=O)Nc1ccccc1)c(N)n[nH]c2=O |(11.01,-19.24,;10.24,-17.91,;8.7,-17.92,;11,-16.57,;10.23,-15.24,;8.69,-15.24,;7.91,-13.91,;8.68,-12.58,;10.22,-12.57,;11,-13.89,;7.91,-11.25,;6.39,-11.09,;6.07,-9.6,;7.39,-8.83,;8.53,-9.85,;10.03,-9.52,;10.66,-8.11,;12.19,-8.27,;13.32,-7.25,;14.77,-7.71,;15.1,-9.21,;13.96,-10.24,;12.51,-9.77,;11.18,-10.55,;11.03,-12.09,;15.91,-6.67,;15.59,-5.17,;17.38,-7.14,;18.52,-6.1,;19.99,-6.58,;21.13,-5.54,;20.8,-4.03,;19.32,-3.57,;18.19,-4.61,;7.39,-7.29,;8.73,-6.53,;6.06,-6.51,;4.73,-7.29,;4.73,-8.83,;3.4,-9.61,)|
CC(=O)Nc1cccc(c1)-n1nc2c(c1-c1oc3cc(ccc3c1C)C(=O)Nc1cccc(c1)C(F)(F)F)c(N)n[nH]c2=O |(29.34,-40.21,;27.79,-40.21,;27.03,-41.55,;27.02,-38.88,;27.79,-37.54,;29.33,-37.54,;30.1,-36.19,;29.32,-34.87,;27.79,-34.88,;27.02,-36.21,;27.01,-33.55,;25.5,-33.39,;25.18,-31.9,;26.49,-31.13,;27.63,-32.15,;29.13,-31.82,;29.76,-30.42,;31.29,-30.57,;32.42,-29.55,;33.88,-30.01,;34.2,-31.52,;33.07,-32.54,;31.61,-32.07,;30.28,-32.85,;30.13,-34.39,;35.02,-28.97,;34.69,-27.47,;36.48,-29.44,;37.62,-28.4,;39.09,-28.88,;40.23,-27.84,;39.9,-26.34,;38.42,-25.87,;37.29,-26.91,;38.09,-24.37,;39.22,-23.32,;36.62,-23.9,;37.68,-22.87,;26.49,-29.59,;27.83,-28.83,;25.16,-28.81,;23.83,-29.59,;23.83,-31.13,;22.5,-31.91,)|
CC(=O)c1ccc(Nc2nccc3c(NC(=O)c4csc5c(N)ncnc45)c(C)ccc23)cc1
CC(C)(C)NS(=O)(=O)c1cncc(c1)-c1ccn2nc(N)nc2c1
CC(C)(C)OC(=O)N1CC2(CCN2C(=O)CN2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)C2=O)C1
CC(C)(C)OC(=O)N1CCN(C[C@@H]1C(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O |r|
CC(C)(C)OC(=O)N1CCN(C[C@H]1C(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O |r|
CC(C)(C)OC(=O)N1CC[C@@H](C1)NC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
CC(C)(C)OC(=O)N1CC[C@H](C1)NC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
CC(C)(C)c1cc(NC(=O)Nc2ccc(Nc3ncnc4ccccc34)cc2)n(n1)-c1cccc(N)c1
CC(C)(C)c1cc(NC(=O)Nc2ccc(cc2)-c2cn3c(n2)sc2cc(OCCN4CCOCC4)ccc32)no1
CC(C)(C)c1cc(NC(=O)Nc2ccc(cc2)-n2nc(-c3ccc(OCCN4CCOCC4)cc3)c3c(N)ncnc23)no1
CC(C)(C)c1cc(NC(=O)Nc2cccc(Nc3ncnc4ccccc34)c2)n(n1)-c1cccc(N)c1
CC(C)(C)c1cnc(CSc2cnc(NC(=O)C3CCNCC3)s2)o1
CC(C)(C)c1nsc(CN2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)C2=O)n1
CC(C)(CO)NC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
CC(C)(NC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)C#N
CC(C)CNC(=O)c1ccc(C)c(c1)C#Cc1cnc2ccnn2c1
CC(C)COC(=O)N1CCC(C1)c1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
CC(C)COC(=O)N1CCN(CC1)c1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
CC(C)N(CC(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
CC(C)NC(=O)c1ccc(C)c(c1)C#Cc1cnc2ccnn2c1
CC(C)OC(=O)N1CCC(C1)c1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
CC(C)OC(=O)N1CCN(CC1)c1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
CC(C)Oc1cccc(NC(=O)c2ccc(C)c(c2)C#Cc2cnc3ccnn3c2)c1
CC(C)S(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CC(C)S(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)cc(cc2c1=O)C(F)(F)F
CC(C)S(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Br)cc(cc2c1=O)C(F)(F)F
CC(C)S(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Cl)cc(cc2c1=O)C(F)(F)F
CC(C)S(=O)(=O)c1ccc(Cl)cc1Nn1cnc2ccc(OC(F)(F)F)cc2c1=O
CC(C)Sc1ccc(Cl)cc1Cn1cnc2c(Cl)cc(cc2c1=O)C(F)(F)F
CC(C)[C@@H]1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1 |r|
CC(C)[C@H]1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1 |r|
CC(C)c1cc(CN2CCN(C)CC2)cc(NC(=O)c2ccc3C(C)CN(Cc3c2)c2cncnc2)c1
CC(C)c1cc(CN2CCN(C)CC2)cc(NC(=O)c2ccc3C(C)CN(Cc3c2)c2cncnc2)c1 |w:23.24|
CC(C)c1cc(NC(=O)c2ccc3C[C@H](Cc3c2)N(C)c2cncnc2)cc(c1)-n1cnc(C)c1 |r|
CC(C)c1ccc(cc1-c1cccc(c1)-c1cnc2cnccn12)C(=O)Nc1cccc(c1)C(F)(F)F
CC(C)c1ccc(cc1C#Cc1cnc2ccccn12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CC(C)c1ccc(cc1C#Cc1cnc2cccnn12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CC(C)c1ccc(cc1C#Cc1cnc2cnccn12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CC(C)n1nc(-c2cc3cc(O)ccc3[nH]2)c2c(N)ncnc12
CC(N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)C(=O)NCC(F)(F)F
CC(NC(=O)c1cc(n[nH]1)-c1ccccc1)c1ccc(cc1)C(=O)N[C@@H](CCC1CCCCC1)C(=O)NC1CCCN(C1)S(C)(=O)=O |r|
CC(NC(=O)c1cc(n[nH]1)-c1ccccc1)c1ccc(cc1)C(=O)N[C@@H](CCC1CCCCC1)C(=O)N[C@@H]1CCCN(C1)S(C)(=O)=O |r|
CC(NC(=O)c1cc(n[nH]1)-c1ccccc1)c1ccc(cc1)C(=O)N[C@@H](CCC1CCCCC1)C(=O)N[C@H]1CCCN(C1)S(C)(=O)=O |r|
CC(NC(=O)c1cnc2ccccn12)c1ccc(cc1)C(=O)N[C@H](CCC1CCCCC1)C(=O)NC1CCCN(C1)S(C)(=O)=O |r|
CC(NC(=O)c1cnn(C)c1N)c1ccc(cc1)C(=O)N[C@@H](CCC1CCCCC1)C(=O)NC1CCCN(C1)S(C)(=O)=O |r|
CC1(C)CCCN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3n2)c2c1ccc(F)c2Cl
CC1(C)CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
CC1(C)CNc2cc(NC(=O)c3cccnc3NCc3ccncc3)ccc12
CC1(C)COCCN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
CC1(C)N(CC(=O)NCC(F)(F)F)C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)N1c1ccccc1
CC1(C)OCC(=O)Nc2cc(Nc3nc(NCC(F)(F)F)c4occc4n3)ccc12
CC1(F)CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
CC1(O)CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
CC1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(Oc3ccc(cc3)-c3n[nH]c4ncnc(N)c34)c2)CC1
CC1CN(C(=O)CN2C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c3c2cccc3Br)c2ccccc12
CC1CN(C(=O)CN2C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c3c2cccc3Br)c2ccccc12 |w:1.0|
CC1CN(CCS1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
CC1CN(Cc2cc(NC(=O)Nc3cc(CN4CCN(C)CC4)cc(c3)C(F)(F)F)ccc12)c1cncnc1
CC1CN(Cc2cc(NC(=O)c3cc(CN4CCN(C)CC4)cc(c3)C(F)(F)F)ccc12)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CCN2CCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CCN2CCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN(C)C)cc(c1)C(F)(F)F)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN(C)C)cc(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN(C)CCN(C)C)cc(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCCCC2)cc(c1)C(F)(F)F)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCCCC2)cc(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)c(C)c(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)c(Cl)c(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)c(F)c(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)-c1ccccc1)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)-c1ccccc1)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(C)(C)C)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(C)(C)C)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)c1cccnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C1CC1)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C1CC1)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C1CCCC1)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C1CCCCC1)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C1CCCCC1)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(CC2)C(=O)CC2(CCC#C)N=N2)cc(c1)C(F)(F)F)c1cncnc1 |c:35|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(CC2)C2CCCCC2)cc(c1)C(F)(F)F)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(CC2)C2CCCCC2)cc(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(CCC(=O)NCCCNC(=O)OC3CCC\C=C\CC3)CC2)cc(c1)C(F)(F)F)c1cncnc1 |t:40|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(CCC3(CCC#C)N=N3)CC2)cc(c1)C(F)(F)F)c1cncnc1 |c:31|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCOCC2)cc(c1)C(F)(F)F)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCOCC2)cc(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCSCC2)cc(c1)C(F)(F)F)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCSCC2)cc(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CC[C@@H](C2)N(C)C)cc(c1)C(F)(F)F)c1cncnc1 |r,w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CC[C@H](C2)N(C)C)cc(c1)C(F)(F)F)c1cncnc1 |r,w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(cc(c1)C(F)(F)F)N1CCN(C)CC1)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(cc(c1)C(F)(F)F)N1CCN(C)CC1)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cc(ccc1CN1CCN(C)CC1)C(F)(F)F)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1ccc(CN2CCN(C)CC2)c(c1)C(F)(F)F)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1ccc(CN2CCN(C)CC2)c(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1CN(Cc2cc(ccc12)C(=O)Nc1cccc(CN2CCN(C)CC2)c1)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cccc(c1)C(F)(F)F)c1cncnc1
CC1CN(Cc2cc(ccc12)C(=O)Nc1cccc(c1)C(F)(F)F)c1cncnc1 |w:1.0|
CC1Cc2ccc(cc2CN1c1cncnc1)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CC1Cc2ccc(cc2CN1c1cncnc1)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F |w:1.0|
CC1N(CC(=O)NCC(F)(F)F)C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)N1c1ccccc1
CCC(=O)N1CCC(C1)Nc1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
CCC(=O)Nc1cc(Nc2ncc(C(=O)Nc3cc(NC(=O)c4cc(OC)c(OC)c(OC)c4)ccc3C)c(NC)n2)ccc1C
CCC(CC)N1CCN(Cc2cc3ncn(Nc4cc(Cl)ccc4S(=O)(=O)CC)c(=O)c3cc2Br)CC1
CCC1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1 |w:2.1|
CCCCNC(=O)c1ccc(C)c(c1)C#Cc1cnc2ccnn2c1
CCCCNC(=O)c1ccc2c(C)c(oc2c1)-c1n(nc2c1c(N)n[nH]c2=O)-c1ccc(NC(C)=O)cc1 |(82.23,-6.25,;80.77,-5.78,;79.63,-6.81,;78.16,-6.34,;77.02,-7.37,;75.55,-6.91,;75.22,-5.4,;74.41,-7.94,;74.74,-9.45,;73.6,-10.48,;72.14,-10.01,;70.81,-10.79,;70.66,-12.32,;69.67,-9.76,;70.29,-8.35,;71.82,-8.5,;72.95,-7.48,;68.16,-10.08,;67.55,-11.48,;66.03,-11.32,;65.71,-9.83,;67.03,-9.07,;67.03,-7.53,;68.36,-6.76,;65.7,-6.75,;64.37,-7.53,;64.37,-9.07,;63.03,-9.84,;68.32,-12.81,;67.55,-14.15,;68.32,-15.48,;69.86,-15.47,;70.64,-16.81,;69.87,-18.14,;70.65,-19.47,;68.33,-18.15,;70.63,-14.13,;69.85,-12.8,)|
CCCCOC(=O)N1CCC(C1)c1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
CCCCOC(=O)N1CCN(CC1)c1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
CCCN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1)c1cncnc1 |r|
CCCNC(=O)[C@H](CCC1CCCCC1)NC(=O)c1ccc(CNC(=O)c2cc(n[nH]2)-c2ccccc2)cc1 |r|
CCCNC(=O)[C@H](CCC1CCCCC1)NC(=O)c1ccc(CNC(=O)c2cnn(c2N)-c2ccccc2)cc1 |r|
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(Cl)cc23)c1F
CCCS(=O)(=O)Nc1ccc(F)c(C(=O)c2c[nH]c3ncc(cc23)-c2ccc(Cl)cc2)c1F
CCCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
CCCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCCSc1ccccc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CCCc1ccc(Cl)cc1Nn1cnc2c(Cl)cc(cc2c1=O)C(F)(F)F
CCN(CC)CCNC(=O)c1c(C)[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c1C
CCN(CCO)CCCOc1ccc2c(Nc3cc(CC(=O)Nc4cccc(F)c4)n[nH]3)ncnc2c1
CCN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1)c1cncnc1 |r|
CCN1CCN(CC1)c1cc(cc(c1)C(F)(F)F)C(=O)Nc1cccc(Nc2ccc3c(OC)cccc3n2)c1
CCN1CCN(CC1)c1ccc(Nc2ncc3scc(-c4cccc(NS(C)(=O)=O)c4)c3n2)cc1
CCN1CCN(Cc2c(Br)cc3c([nH]c(=O)n(Cc4cc(Cl)ccc4S(=O)(=O)CC)c3=O)c2Br)CC1
CCN1CCN(Cc2cc(NC(=O)c3ccc4C(C)CN(Cc4c3)c3cncnc3)cc(c2)C(F)(F)F)CC1
CCN1CCN(Cc2cc(NC(=O)c3ccc4C(C)CN(Cc4c3)c3cncnc3)cc(c2)C(F)(F)F)CC1 |w:17.17|
CCN1CCN(Cc2cc(OC(F)(F)F)cc(c2)C(=O)NCc2cc(Cl)ccc2S(=O)(=O)CC)CC1
CCN1CCN(Cc2cc3[nH]c(=O)n(Cc4cc(Cl)ccc4S(=O)(=O)CC)c(=O)c3cc2C(F)(F)F)CC1
CCN1CCN(Cc2cc3[nH]c(=O)n(Cc4cc(Cl)ccc4S(=O)(=O)CC)c(=O)c3cc2OC(F)(F)F)CC1
CCN1CCN(Cc2ccc(NC(=O)Nc3ccc(Oc4cc(NC)ncn4)cc3)cc2C(F)(F)F)CC1
CCN1CCN(Cc2ccc(NC(=O)c3cccc(c3)-c3ccc4nc(NC(=O)C5CC5)sc4n3)cc2C(F)(F)F)CC1
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(NCc3cnc4[nH]ccc4c3OC)c2)CC1
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(Oc3ccc(cc3)-c3n[nH]c4ncnc(N)c34)c2)CC1
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(Oc3ccc4CC(=O)Nc4c3)c2)CC1
CCN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(Oc3ccc4NC(=O)Cc4c3)c2)CC1
CCNC(=O)[C@H](CCC1CCCCC1)NC(=O)c1ccc(CNC(=O)c2cnn(c2N)-c2ccccc2)cc1 |r|
CCN[C@H]1CCCN(Cc2c(Br)c3ncn(Cc4cc(Cl)ccc4S(=O)(=O)CC)c(=O)c3cc2C(F)(F)F)C1 |r|
CCN[C@H]1CCCN(Cc2c(Cl)c3ncn(Cc4cc(Cl)ccc4S(=O)(=O)CC)c(=O)c3cc2C(F)(F)F)C1 |r|
CCN[C@H]1CCCN(Cc2c(Cl)cc(cc2C(F)(F)F)C(=O)NCc2cc(Cl)ccc2S(=O)(=O)CC)C1 |r|
CCN[C@H]1CCCN(Cc2c(cc3c(ncn(Cc4cc(Cl)ccc4S(=O)(=O)CC)c3=O)c2C#N)C(F)(F)F)C1 |r|
CCOC(=O)N1CCC(C1)c1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
CCOC(=O)N1CCN(CC1)c1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
CCOc1cc(=O)[nH]cc1-c1ccc(CC(=O)Nc2cc(on2)C(C)(C)C(F)(F)F)c(F)c1
CCOc1cc2ncc(C#N)c(Nc3ccc(F)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)C
CCOc1cc2ncc(C#N)c(Nc3ccc(OCc4ccccn4)c(Cl)c3)c2cc1NC(=O)\C=C\CN(C)C
CCOc1ccc(c(NNC(=O)c2cc(Cl)cc(c2)C(F)(F)F)c1)S(=O)(=O)CC |$;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;$|
CCOc1cccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
CCS(=O)(=O)N1CCC(C1)Nc1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
CCS(=O)(=O)c1c(C)cc(Cl)cc1CNC(=O)c1cc(Cl)c(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1c(C)cc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1c(C)cc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1c(CNC(=O)c2cc(Cl)c(CN3CCC[C@@H](C3)NC)c(c2)C(F)(F)F)cc(Cl)cc1OC |r|
CCS(=O)(=O)c1c(Cl)cc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1c(Cl)cc(Cl)cc1CNC(=O)c1ccc(CN2CCN(C)CC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1c(Cl)cc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1c(Cl)cc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(C)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1c(Cl)cc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCNCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1c(Cn2c(=O)[nH]c3c(Cl)c(CN4CCC[C@@H](N)C4)c(cc3c2=O)C(F)(F)F)cc(Cl)cc1OC |r|
CCS(=O)(=O)c1cc(C)c(C)cc1CNC(=O)c1cc(Cl)c(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1cc(C)c(C)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1cc(C)c(Cl)cc1CNC(=O)c1cc(Cl)c(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1cc(C)c(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1cc(C)ccc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1cc(C)ccc1Cn1cnc2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1cc(Cl)c(Cl)cc1NNC(=O)c1cc(Cl)cc(c1)C(F)(F)F |$;;;;;;;;;;;;;HN;;;;;;;;;;;;;;$|
CCS(=O)(=O)c1cc(OC)c(Cl)cc1NNC(=O)c1cc(Cl)c(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r,$;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(Br)cc1CNC(=O)c1cc(Cl)cc(OC(F)(F)F)c1
CCS(=O)(=O)c1ccc(Br)cc1CNC(=O)c1cc(Cl)cc(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Br)cc1CNC(=O)c1cccc(OC(F)(F)F)c1
CCS(=O)(=O)c1ccc(Br)cc1CNC(=O)c1cccc(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Br)cc1Cn1c(=O)[nH]c2c(Cl)cc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Br)cc1Cn1c(=O)[nH]c2c(Cl)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Br)cc1Cn1c(=O)[nH]c2ccc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Br)cc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Br)cc1Cn1cnc2c(Cl)cc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Br)cc1Cn1cnc2c(Cl)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Br)cc1Cn1cnc2ccc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Br)cc1Cn1cnc2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(C)cc1CNC(=O)c1cc(Cl)c(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(C)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1c[nH]c(=O)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCC[C@@H](C2)NC(=O)CCN)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCC[C@@H](C2)NC(=O)CN)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCC[C@@H](C2)NC(=O)CNC)c(c1)C(F)(F)F |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCC[C@@H](N)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCC[C@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCC[C@H](N)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCN(C)CC2)c(Br)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCN(C)CC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCN(CC2)C(C)C)c(Br)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCN(CC2)C2CCOCC2)c(Br)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCNCC2)c(Br)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCNCC2)c(OC(F)(F)F)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CCNCC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CC[C@@H](CN)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CC[C@@H](CNC)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CC[C@H](C2)NS(=O)(=O)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)c(CN2CC[C@H](N)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)cc(Br)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)cc(CN2CCN(C)CC2)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)cc(CN2CCN(CC2)C(C)C)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)cc(CN2CCN(CC2)C2CCOCC2)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)cc(CN2CCNCC2)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)cc(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)cc(c1)N1CCN(C)CC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)cc(c1)N1CCN(CC1)C(C)C
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)cc(c1)N1CCN(CC1)C1CCOCC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Br)cc(c1)N1CCNCC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(C#N)c(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(C#N)c(CN2CCN(C)CC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(C#N)c(CN2CCNCC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(C)c(CN2CCC[C@@H](C2)NC)c(Cl)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(C)c(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
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CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(CN2CC[C@H](C2)N(C)C)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(CN2CC[C@H](C2)NC(C)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(CN2CC[C@H](C2)NC(N)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(CN2CC[C@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(CN2CC[C@H](C2)NS(C)(=O)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(CN2CC[C@H](CNC)C2)c(OC(F)(F)F)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(CN2CC[C@H](N)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(CN2C[C@@H](N)C3(CC3)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(CNCCCN)c(c1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(CNCCCNCCCN(C)C)c(c1)C(F)(F)F |$;;;;;;;;;;;;;;;;;;;;;;HN;;;;HN;;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(Cc2cccc(N)c2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(N2CCN(C)CC2)c(OC(F)(F)F)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(N2CCNCC2)c(OC(F)(F)F)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)c(OC(C)=O)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)cc(CN2CCN(C)CC2)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)cc(CN2CCN(CC2)C(C)C)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)cc(CN2CCN(CC2)C2CCOCC2)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)cc(CN2CCNCC2)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)cc(Cl)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)cc(OC(F)(F)F)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)cc(OC)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)cc(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(F)cc(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCC(CC1)N(C)C
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCC(CC1)N1CCCC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCC(CC1)N1CCOCC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCC(CC1)NC(C)=O
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCC(CC1)NS(C)(=O)=O
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCC(N)CC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCC(O)CC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCN(C)CC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCN(CC(F)(F)F)CC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCN(CC1)C(C)C
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCN(CC1)C1CCOCC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCNC(C)(C)C1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCNCC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CCOCC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CC[C@@H](C1)NC(C)=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CC[C@@H](C1)NS(C)(=O)=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CC[C@@H](N)C1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CC[C@H](C1)NC(C)=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CC[C@H](C1)NS(C)(=O)=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC(F)(F)F)cc(c1)N1CC[C@H](N)C1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC)c(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC)c(CN2CCN(C)CC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC)c(CN2CCNCC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(OC)c(CN2CC[C@@H](N)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(cc(Cl)c1F)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(cc(c1)C(F)(F)F)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(cc(c1)C(F)(F)F)N1CCN(C)CC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(cc(c1)C(F)(F)F)N1CCN(CC1)C(C)C
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(cc(c1)C(F)(F)F)N1CCN(CC1)C1CCOCC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(cc(c1)C(F)(F)F)N1CCNCC1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(ccc1F)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cc(ccn1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(Br)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CC2CCN(C)CC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CC2CCNCC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCCC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCCC[C@@H]2CN)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCCC[C@@H]2CNC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCCC[C@@H]2NC(=O)CCN)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCCC[C@@H]2NC(=O)CN(C)C)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCCC[C@@H]2NC(=O)CN)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCCC[C@@H]2NC(=O)CNC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCCC[C@@H]2NC(=O)[C@@H](C)N)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCCC[C@@H]2NC(=O)[C@H](C)N)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCCC[C@H]2CNC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)N(C)C)c(OC(F)(F)F)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)N(C)C)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)NC(=O)C(C)(C)N)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)NC(=O)CN)c(OC(F)(F)F)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)NC(C)=O)c(OC(F)(F)F)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)NC(C)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)NC(N)=O)c(OC(F)(F)F)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)NC(N)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)NC)c(OC(F)(F)F)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)NS(C)(=O)=O)c(OC(F)(F)F)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](C2)NS(C)(=O)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](CN(C)C)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](CN)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](CNC(=O)CN)C2)c(c1)C(F)(F)F |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](CNC(C)=O)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](CNS(C)(=O)=O)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](N)C2)c(OC(F)(F)F)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H](N)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H]2CN(C)C)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H]2CN)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@@H]2CNC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@H](C2)N(C)C)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@H](C2)NC(C)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@H](C2)NC(N)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@H](C2)NS(C)(=O)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@H](CN(C)C)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@H](CNC(C)=O)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@H](CNS(C)(=O)=O)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@H](N)C2)c(OC(F)(F)F)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@H](N)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@H]2CN(C)C)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@H]2CN)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCC[C@H]2CNC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCN(C)CC2)c(Br)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCN(C)CC2)c(Cl)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCN(C)CC2)c(OC(F)(F)F)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCN(C)CC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCN(CC2)C(=O)CN)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCN(CC2)C(C)C)c(Br)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCN(CC2)C(C)C)c(Cl)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCN(CC2)C(C)C)c(OC(F)(F)F)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCN(CC2)C(C)C)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCN(CC2)C2CCOCC2)c(Br)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCN(CC2)C2CCOCC2)c(Cl)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCN(CC2)C2CCOCC2)c(OC(F)(F)F)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCN(CC2)C2CCOCC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCNCC2)c(Br)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCNCC2)c(Cl)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCNCC2)c(OC(F)(F)F)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CCNCC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@@H](C2)N(C)C)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@@H](C2)NC(C)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@@H](C2)NS(C)(=O)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@@H](CN(C)C)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@@H](CN)C2)c(OC(F)(F)F)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@@H](CN)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@@H](CNC(C)=O)C2)c(c1)C(F)(F)F |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@@H](CNC)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@@H](CNS(C)(=O)=O)C2)c(c1)C(F)(F)F |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@@H](N)C2)c(Br)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@@H](N)C2)c(OC(F)(F)F)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@@H](N)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@@H](O)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)N(C)C)c(Br)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)N(C)C)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)N(C)S(C)(=O)=O)c(Br)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)N(C)S(C)(=O)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)NC(=O)CN)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)NC(=O)OC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)NC(C)=O)c(Br)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)NC(C)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)NC(N)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)NC)c(Br)c1 |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)NC)c(c1)C(F)(F)F |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)NS(C)(=O)=O)c(Br)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)NS(C)(=O)=O)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](C2)OC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](CN(C)C)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](CN)C2)c(OC(F)(F)F)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](CN)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](CNC(C)=O)C2)c(c1)C(F)(F)F |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](CNC)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](CNS(C)(=O)=O)C2)c(c1)C(F)(F)F |r,$;;;;;;;;;;;;;;;;;;;;;;;;;;HN;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](N)C2)c(OC(F)(F)F)c1 |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(CN2CC[C@H](N)C2)c(c1)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(Cc2cccc(N)c2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(Cc2ccncc2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(N)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(N2CCNCC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(NC2CCNCC2)c(OC)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(OC2CCCNC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccc(OC2CCNCC2)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cccc(OC(F)(F)F)c1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cccc(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cccc(n1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1ccnc(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cnc(N)c(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cncc(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1cnn(c1-n1cccc1)-c1ccccc1
CCS(=O)(=O)c1ccc(Cl)cc1CNC(=O)c1nc(C)oc1C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CCC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CCC[C@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CCN(C)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CCN(C)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CCN(CC3)C(C)C)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CCN(CC3)C3CCOCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CCNCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CCNCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CC[C@@H](CN)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CC[C@@H](N)C3)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CC[C@H](C3)N(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CC[C@H](C3)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CC[C@H](C3)NC(C)=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CC[C@H](C3)NC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CC[C@H](C3)NC)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CC[C@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CC[C@H](C3)NS(C)(=O)=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CC[C@H](C3)NS(C)(=O)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)cc(C)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)cc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(C#N)c(CN3CCC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(C)c(CN3CCC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(C=C)c(CN3CCC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(CN3CCN(C)CC3)cc(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(CN3CCN(C)CC3)cc(Cl)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(CN3CCN(CC3)C(=O)OC(C)(C)C)cc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(CN3CCN(CC3)C(=O)OC(C)(C)C)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(CN3CCNCC3)cc(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(CN3CCNCC3)cc(Cl)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(CN3CCNCC3)cc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(CN3CCNCC3)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(C3OCCO3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(C=C)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(C=O)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC(C3)NC(=O)OC(C)(C)C)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC(C3)NC(C)=O)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC(C3)NS(=O)(=O)N(C)C)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC(C3)NS(=O)(=O)NC)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC(C3)NS(C)(=O)=O)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC(C3)NS(N)(=O)=O)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC(N)C3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC(C3)C(N)=O)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC(CC3)C(N)=O)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC(CN)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC(N)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCCC(C3)NC(=O)C(C)N)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCCC(C3)NC(=O)CCN)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCCC(C3)NC(=O)CN)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCCC(C3)NC(=O)CNC)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCCCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCCC[C@@H]3C(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCCC[C@@H]3CN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCCC[C@H]3C(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCCC[C@H]3CN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)C(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)N(C)C(=O)OC(C)(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)N(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)NC(=O)OC(C)(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)NC(=O)OC(C)(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)NC(C)=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)NC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)NC)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)NCCNC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)NCCO)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)NS(C)(=O)=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)NS(C)(=O)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](C3)OCCN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](CN(C)C(=O)OC(C)(C)C)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](CN(C)C)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](CN)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](CNC(=O)OC(C)(C)C)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](CNC(C)=O)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](CNC)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](CNS(C)(=O)=O)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](N)C3)c(C)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](N)C3)c(C=C)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](N)C3)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](O)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3C(=O)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3C(=O)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3CN(C)C(=O)OC(C)(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3CN(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3CN(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3CN)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3CN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3CNC(=O)OC(C)(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3CNC(C)=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3CNC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3CNC)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3CNC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3CNS(C)(=O)=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H]3CNS(C)(=O)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@]3(C)C(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)C(=O)NC3CCNCC3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)C(=O)NCCN(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)C(=O)NCCN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)C(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)C(O)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)N(C)C(=O)OC(C)(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)N(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)NC(=O)C3CCNCC3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)NC(=O)OC(C)(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)NC(=O)OC(C)(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)NC(=O)OCCN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)NC(C)=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)NC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)NC)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)NS(C)(=O)=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](C3)NS(C)(=O)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](CN(C)C(=O)OC(C)(C)C)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](CN(C)C)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](CN)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](CNC(=O)OC(C)(C)C)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](CNC(C)=O)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](CNC)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](CNS(C)(=O)=O)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](N)C3)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3C(=O)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3C(=O)NC(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3C(=O)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3C(=O)OC(C)(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3C(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3C(O)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CN(C)C(=O)OC(C)(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CN(C)C(=O)OC(C)(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CN(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CN(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CN)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CNC(=O)OC(C)(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CNC(=O)OC(C)(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CNC(C)=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CNC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CNC)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CNC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CNS(C)(=O)=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CNS(C)(=O)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@H]3CO)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(C)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(C)CC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(C)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC#C)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC#N)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC(F)(F)F)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC(F)F)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC(N)=O)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC3)C(=O)CCN)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC3)C(=O)CN)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC3)C(C)C)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC3)C(C)C)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC3)C(N)=O)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC3)C3CCOCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC3)C3CCOCC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC3)C3COC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCN(CC3)S(=O)(=O)NC)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCNC(=O)C3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCNCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCNCC3)c(Cl)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCNCC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCNCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](C3)C(=O)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](C3)C(=O)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](C3)C(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](C3)N(C)C(=O)OC(C)(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](C3)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](C3)NC(=O)OC(C)(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](C3)NC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](C3)NS(C)(=O)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](CN(C)C)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](CN)C3)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](CN)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](CNC(=O)OC(C)(C)C)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](CNC(C)=O)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](CNC)C3)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](CNC)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](CNS(C)(=O)=O)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](CO)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](N)C3)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@@H](O)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)C(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)N(C)C(=O)CN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)N(C)C(=O)OC(C)(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)N(C)C(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)N(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)N(C)S(C)(=O)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)N3CCCC3=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC(=O)C(C)(C)N)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC(=O)C(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC(=O)C3CCCC3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC(=O)CC3CCCCC3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC(=O)CCN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC(=O)CN(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC(=O)CN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC(=O)CNC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC(=O)[C@@H](C)N)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC(=O)[C@H](C)N)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NC3COC3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NCC#C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NCC#N)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NCC(F)(F)F)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NCC(F)F)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NCC(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NS(=O)(=O)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NS(=O)(=O)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](C3)NS(C)(=O)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](CN(C)C)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](CN)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](CNC(=O)OC(C)(C)C)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](CNC(C)=O)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](CNC)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](CNS(C)(=O)=O)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CC[C@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3C[C@@H](CCN)NC3=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CN3C[C@@H](CCNS(C)(=O)=O)NC3=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(CO)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)c(COS(C)(=O)=O)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)cc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(F)c(CN3CCN(C)CC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(F)c(CN3CCN(C)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(F)c(CN3CCNCC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(F)c(CN3CCNCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2c(OC)c(CN3CCC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(Br)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(C(O)CO)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(C)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCC(C3)N3CCC(F)(F)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCC(C3)N3CCC(F)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCC(C3)N3CCCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCC(C3)N3CCCCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCC(C3)N3CCN(C)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCC(C3)N3CCOCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCC(C3)OC)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCC(C3)OCC=C)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCC(C3)OCCOC)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCC[C@@H](N)C3)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCC[C@H](C3)N(C)C)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCC[C@H](C3)NC)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(C)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(C)CC3)c(Cl)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(C)CC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(C)CC3)c(cc2c1=O)C#N
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(C)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(CC3)C(C)=O)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(CC3)C(C)C)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(CC3)C(C)C)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(CC3)C(C)C)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(CC3)C3CCC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(CC3)C3CCCCC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(CC3)C3CCOCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(CC3)C3CCOCC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(CC3)C3CCOCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(CC3)S(C)(=O)=O)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCN(CC3)S(C)(=O)=O)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCNCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCNCC3)c(Cl)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCNCC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CCNCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@@H](C3)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@@H](C3)NC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@@H](CN(C)C)C3)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@@H](CN)C3)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@@H](CN)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@@H](CNC)C3)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@@H](N)C3)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@@H](N)C3)c(Cl)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@@H](N)C3)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@@H](O)C3)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)N(C)C(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)N(C)C)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)N(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)NC(=O)OC(C)(C)C)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)NC(C)=O)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)NC(C)=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)NC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)NC)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)NC)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)NS(=O)(=O)N(C)C)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](C3)NS(C)(=O)=O)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](N)C3)c(Cl)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(CN3CC[C@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(Cc3ccncc3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(NC3CCNCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2cc(OC3CCNCC3)c(Cl)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2ccc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1c(N)nc2c(CN3CCNCC3)cc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1ccc2c(Br)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1ccc2c(Cl)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1ccc2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Br)c(CN3CCC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Br)c(CN3CCN(CC3)C3CCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Br)c(CN3CCN(CC3)C3CCCCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Br)c(CN3CCNCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Br)c(CN3CC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Br)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(C#N)c(CN3CCC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(C#N)c(CN3CC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(C#N)c(CN3CC[C@H](C3)NC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(C#N)c(CN3CC[C@H](C3)NS(C)(=O)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(C)c(CN3CCC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(CN3CCN(C)CC3)cc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(CN3CCN(C)CC3)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(CN3CCN(CC3)C(C)C)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(CN3CCN(CC3)C3CCOCC3)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(CN3CCN(CC3)C3CNC3)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(CN3CCNCC3)cc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(CN3CCNCC3)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(C3OCCO3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(C=O)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC(C3)C(N)=O)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](C3)C(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](C3)N(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](C3)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](C3)N(CCN)CCN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](C3)NC(=O)CCN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](C3)NC(=O)CN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](C3)NC(=O)CNC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](C3)NC(=O)[C@@H](C)N)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](C3)NC(=O)[C@H](C)N)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](C3)NC)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](C3)NCCN)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](C3)NCCO)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@@H]3C(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@H](C3)C(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@H](C3)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@H](N)C3)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCC[C@H]3C(N)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCN(C)CC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCN(C)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCN(CC3)C(C)C)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCN(CC3)C3CCOCC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCN4CCC[C@@H]4C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCN4CCC[C@H]4C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCNC(=O)C3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCNCC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CCNCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@@H](CN(C)C)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@@H](CN)C3)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@@H](CN)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@@H](CNC)C3)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@@H](CNC)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@@H](N)C3)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@H](C3)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@H](C3)N3CCCC3=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@H](C3)NC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@H](C3)NC)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@H](C3)NS(C)(=O)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@H](CN(C)C)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@H](CN)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@H](CNC(=O)OC(C)(C)C)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(CN3CC[C@H](CNC)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)c(COS(C)(=O)=O)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(Cl)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(F)c(CN3CCN(C)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(F)c(CN3CCNCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2c(OC)c(CN3CCC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CC(C3)N3CCCCC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCC(CC3)N3CCCC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCC(CC3)N3CCOCC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCC(F)(F)CC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCC[C@@H](C3)NC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCC[C@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCN(C)CC3)c(Cl)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCN(C)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCN(CC#C)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCN(CC(F)(F)F)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCN(CC3)C(C)C)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCN(CC3)C(C)C)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCN(CC3)C3CCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCN(CC3)C3CCN(C)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCN(CC3)C3CCOCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCNCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCNCC3)c(Cl)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCNCC3)c(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CCNCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CC[C@@H](C3)NC(C)=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CC[C@@H](C3)NC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CC[C@@H](N)C3)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CC[C@H](C3)N(C)C)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CC[C@H](C3)N(C)C)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CC[C@H](C3)NC(C)=O)c(OC(F)(F)F)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CC[C@H](C3)NC(C)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2cc(CN3CC[C@H](C3)NS(C)(=O)=O)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2ccc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Cn1cnc2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1NNC(=O)c1c[nH]nc1C(F)(F)F |$;;;;;;;;;;;;HN;;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1NNC(=O)c1cc(C)[nH]c(=O)c1 |$;;;;;;;;;;;;HN;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1NNC(=O)c1ccc(NC2CCNCC2)c(OC)c1 |$;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1NNC(=O)c1nc(oc1C(F)(F)F)-c1ccccc1 |$;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(Cl)cc1Nn1c(=O)[nH]c2c(Br)cc(C)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1c(=O)[nH]c2c(Cl)c(CN3CCN(C)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Nn1c(=O)[nH]c2c(Cl)c(CN3CCNCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Br)c(CN3CCN(C)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Br)c(CN3CCN(CC3)C(C)C)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Br)c(CN3CCN(CC3)C3CCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Br)c(CN3CCN(CC3)C3CCCCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Br)c(CN3CCNCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Br)cc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Br)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(C)cc(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Cl)c(CN3CCN(C)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Cl)c(CN3CCN(C)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Cl)c(CN3CCN(CC3)C(C)C)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Cl)c(CN3CCN(CC3)C3CCOCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Cl)c(CN3CCNCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Cl)c(CN3CCNCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Cl)cc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2c(Cl)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CC(C)OC(C)C3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCC(C3)N3CCCCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCC(N)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCCOCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(C)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(C)CC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)C(C)=O)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)C(C)C)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)C(C)C)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)C(CO)CO)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)C3CCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)C3CCCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)C3CCCCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)C3CCOCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)C3CCOCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)C3CCSCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)C3CNC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)C3COC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)S(=O)(=O)C(C)C)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)S(=O)(=O)C(F)(F)F)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)S(=O)(=O)N(C)C)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CC3)S(C)(=O)=O)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(CCOC)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(Cc4cc[nH]n4)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(Cc4ccoc4)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCN(Cc4ccsc4)CC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCNCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCNCC3)c(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CCOCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CC[C@@H](C3)N(C)C)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CC[C@@H](C3)NC(C)=O)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CC[C@@H](N)C3)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CC[C@@H](O)C3)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CC[C@H](C3)N(C)C(C)=O)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CC[C@H](C3)N(C)C)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CC[C@H](C3)NC(C)=O)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN3CC[C@H](C3)NC)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CNCCN3CCCCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CNCCN3CCOCC3)c(Br)cc2c1=O
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN[C@@H]3CCNC3)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2cc(CN[C@H]3CCNC3)c(Br)cc2c1=O |r|
CCS(=O)(=O)c1ccc(Cl)cc1Nn1cnc2ccc(OC(F)(F)F)cc2c1=O
CCS(=O)(=O)c1ccc(F)cc1CNC(=O)c1cccc(c1)C(F)(F)F
CCS(=O)(=O)c1ccc(F)cc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(F)cc1Cn1cnc2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(F)cc1NNC(=O)c1cccc(c1)C(F)(F)F |$;;;;;;;;;;;;HN;;;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(OC(F)(F)F)cc1NNC(=O)c1ccc(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r,$;;;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(OC)cc1Cn1c(=O)[nH]c2c(Br)c(CN3CCC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(OC)cc1Cn1c(=O)[nH]c2c(OC)c(CN3CCC[C@@H](C3)NC)c(cc2c1=O)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(OC)cc1Cn1cnc2c(Br)cc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccc(cc1CNC(=O)c1cc(Cl)cc(c1)C(F)(F)F)C#N
CCS(=O)(=O)c1ccc(cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCC[C@@H](N)C3)c(cc2c1=O)C(F)(F)F)C(F)(F)F |r|
CCS(=O)(=O)c1ccc(cc1Cn1c(=O)[nH]c2c(Cl)c(CN3CCNCC3)c(cc2c1=O)C(F)(F)F)C#N
CCS(=O)(=O)c1ccc(cc1Cn1c(=O)[nH]c2cc(CN3CCNCC3)c(cc2c1=O)C(F)(F)F)C#N
CCS(=O)(=O)c1ccc(cc1Cn1ccc2ccc(OC(F)(F)F)cc2c1=O)C#N
CCS(=O)(=O)c1ccc(cc1Cn1ccc2ccc(cc2c1=O)C(F)(F)F)C#N
CCS(=O)(=O)c1ccc(cc1Cn1cnc2c(Br)cc(cc2c1=O)C(F)(F)F)C#N
CCS(=O)(=O)c1ccc(cc1Cn1cnc2c(Cl)c(CN3CCNCC3)c(cc2c1=O)C(F)(F)F)C#N
CCS(=O)(=O)c1ccc(cc1Cn1cnc2cc(CN3CCNCC3)c(cc2c1=O)C(F)(F)F)C#N
CCS(=O)(=O)c1ccc(cc1NNC(=O)c1cc(Cl)cc(c1)C(F)(F)F)C#N |$;;;;;;;;;;;HN;;;;;;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(cc1NNC(=O)c1cc(Cl)cc(c1)C(F)(F)F)C(F)(F)F |$;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;$|
CCS(=O)(=O)c1ccc(cc1Nn1c(=O)[nH]c2c(Br)cc(cc2c1=O)C(F)(F)F)C#N
CCS(=O)(=O)c1ccc(cc1Nn1cnc2c(Br)cc(OC(F)(F)F)cc2c1=O)C#N
CCS(=O)(=O)c1ccc(cc1Nn1cnc2c(Br)cc(cc2c1=O)C(F)(F)F)C#N
CCS(=O)(=O)c1ccc(cc1Nn1cnc2c(Cl)c(CN3CCNCC3)c(cc2c1=O)C(F)(F)F)C#N
CCS(=O)(=O)c1ccc(cc1Nn1cnc2c(Cl)cc(OC(F)(F)F)cc2c1=O)C#N
CCS(=O)(=O)c1ccc(cc1Nn1cnc2c(Cl)cc(cc2c1=O)C(F)(F)F)C#N
CCS(=O)(=O)c1ccc(cc1Nn1cnc2cc(CN3CCNCC3)c(OC(F)(F)F)cc2c1=O)C#N
CCS(=O)(=O)c1ccc(cc1Nn1cnc2ccc(cc2c1=O)C(F)(F)F)C#N
CCS(=O)(=O)c1ccccc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccccc1Cn1cnc2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1ccncc1CNC(=O)c1cc(Cl)cc(c1)C(F)(F)F
CCS(=O)(=O)c1ccncc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1cnc(Cl)cc1Nn1cnc2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)c1cnccc1CNC(=O)c1cc(Cl)cc(c1)C(F)(F)F
CCS(=O)(=O)c1cnccc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)n1cccc1CNC(=O)c1cc(Cl)c(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r|
CCS(=O)(=O)n1cccc1CNC(=O)c1cccc(c1)C(F)(F)F
CCS(=O)(=O)n1cccc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CCS(=O)(=O)n1cccc1Cn1cnc2ccc(cc2c1=O)C(F)(F)F
CCS(=O)c1ccc(Cl)cc1CNC(=O)c1cc(Cl)cc(c1)C(F)(F)F
CCS(=O)c1ccc(Cl)cc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CCS(=O)c1ccncc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CCSc1ccc(Cl)cc1CNC(=O)c1cc(Br)cc(c1)C(F)(F)F
CCSc1ccc(Cl)cc1CNC(=O)c1cc(Cl)cc(OC(F)(F)F)c1
CCSc1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)cc(C)cc2c1=O
CCSc1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)cc(OC(F)(F)F)cc2c1=O
CCSc1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Br)cc(cc2c1=O)C(F)(F)F
CCSc1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)cc(OC(F)(F)F)cc2c1=O
CCSc1ccc(Cl)cc1Cn1c(=O)[nH]c2c(Cl)cc(cc2c1=O)C(F)(F)F
CCSc1ccc(Cl)cc1Cn1cnc2c(CN3CCNCC3)cc(OC(F)(F)F)cc2c1=O
CCSc1ccc(Cl)cc1Nn1cnc2c(C)cc(Br)cc2c1=O
CCSc1ccc(F)cc1CNC(=O)c1cccc(c1)C(F)(F)F
CCSc1ccc(F)cc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CCSc1ccc(F)cc1Cn1cnc2ccc(cc2c1=O)C(F)(F)F
CCSc1ccc(F)cc1NNC(=O)c1cccc(c1)C(F)(F)F |$;;;;;;;;;;HN;;;;;;;;;;;;;$|
CCSc1ccc(OC(F)(F)F)cc1NNC(=O)c1ccc(CN2CCC[C@@H](C2)NC)c(c1)C(F)(F)F |r,$;;;;;;;;;;;;;;HN;;;;;;;;;;;;;;;;;;;;;;$|
CCSc1ccc(OC(F)(F)F)cc1Nn1cnc2c(Br)cc(cc2c1=O)C(F)(F)F
CCSc1ccc(OC)cc1Cn1cnc2c(Br)cc(cc2c1=O)C(F)(F)F
CCSc1ccc(cc1Nn1c(=O)[nH]c2c(Br)cc(cc2c1=O)C(F)(F)F)C#N
CCSc1ccccc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CC[C@@H]1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1 |r|
CC[C@H](CO)Nc1nc(NCc2ccccc2)c2ncn(C(C)C)c2n1 |r|
CC[C@H]1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1 |r|
CC[C@H]1N(C2CCCC2)c2nc(Nc3ccc(cc3OC)C(=O)NC3CCN(C)CC3)ncc2N(C)C1=O |r|
CCc1c(CN2CCC[C@@H](C2)NC)c(cc2c1[nH]c(=O)n(Cc1cc(Cl)ccc1S(=O)(=O)CC)c2=O)C(F)(F)F |r|
CCc1c(CN2CCC[C@@H](C2)NC)c(cc2c1ncn(Cc1cc(Cl)ccc1S(=O)(=O)CC)c2=O)C(F)(F)F |r|
CCc1cc(CN2CCN(C)CC2)cc(NC(=O)c2ccc3C(C)CN(Cc3c2)c2cncnc2)c1
CCc1cc(CN2CCN(C)CC2)cc(NC(=O)c2ccc3C(C)CN(Cc3c2)c2cncnc2)c1 |w:22.23|
CCc1cc(NC(=O)c2ccc3C[C@H](Cc3c2)N(C)c2cncnc2)cc(c1)-n1cnc(C)c1 |r|
CCc1cc(cc(Cl)c1CN1CCC[C@@H](C1)NC)C(=O)NCc1cc(Cl)ccc1S(=O)(=O)CC |r|
CCc1cc(cc(c1)-c1cc(ccc1CC)C(=O)Nc1cccc(c1)C(F)(F)F)-c1cnc2cnccn12
CCc1cc(cc(c1CN1CCC[C@@H](C1)NC)C(F)(F)F)C(=O)NCc1cc(Cl)ccc1S(=O)(=O)CC |r|
CCc1cc2c([nH]c(=O)n(Cc3cc(Cl)ccc3S(=O)(=O)CC)c2=O)c(Cl)c1CN1CCC[C@@H](N)C1 |r|
CCc1ccc(cc1-c1cc(C)cc(c1)-c1cnc2cnccn12)C(=O)Nc1cc(F)cc(c1)C(F)(F)F
CCc1ccc(cc1-c1cc(C)cc(c1)-c1cnc2cnccn12)C(=O)Nc1cc(ccc1F)C(F)(F)F
CCc1ccc(cc1-c1cc(C)cc(c1)-c1cnc2cnccn12)C(=O)Nc1ccc(F)c(c1)C(F)(F)F
CCc1ccc(cc1-c1cc(C)cc(c1)-c1cnc2cnccn12)C(=O)Nc1cccc(c1)C(F)(F)F
CCc1ccc(cc1-c1cc(C)cc(c1)-c1cnc2cnccn12)C(=O)Nc1cccc(c1F)C(F)(F)F
CCc1ccc(cc1-c1cc(Cl)cc(c1)-c1cnc2cnccn12)C(=O)Nc1cccc(c1)C(F)(F)F
CCc1ccc(cc1-c1cc(F)cc(c1)-c1cnc2cnccn12)C(=O)Nc1cccc(c1)C(F)(F)F
CCc1ccc(cc1-c1cc(OC)cc(c1)-c1cnc2cnccn12)C(=O)Nc1cccc(c1)C(F)(F)F
CCc1ccc(cc1-c1cc(cc(c1)-c1cnc2cnccn12)C#N)C(=O)Nc1cccc(c1)C(F)(F)F
CCc1ccc(cc1-c1cc(cc(c1)-c1cnc2cnccn12)C(C)C)C(=O)Nc1cccc(c1)C(F)(F)F
CCc1ccc(cc1-c1cc(cc(c1)C(C)(C)C)-c1cnc2cnccn12)C(=O)Nc1cccc(c1)C(F)(F)F
CCc1ccc(cc1-c1cc(ccc1C)-c1cnc2cnccn12)C(=O)Nc1cccc(c1)C(F)(F)F
CCc1ccc(cc1-c1ccc(C)c(c1)-c1cnc2cnccn12)C(=O)Nc1cccc(c1)C(F)(F)F
CCc1ccc(cc1-c1cccc(-c2cnc3cnccn23)c1C)C(=O)Nc1cccc(c1)C(F)(F)F
CCc1ccc(cc1-c1cccc(c1)-c1cnc2ccnn2c1)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1-c1cccc(c1)-c1cnc2cnccn12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1-c1cccc(c1)-c1cnc2cnccn12)C(=O)Nc1ccc(cc1)C(F)(F)F
CCc1ccc(cc1-c1cccc(c1)-c1cnc2cnccn12)C(=O)Nc1cccc(CN2CCN(C)CC2)c1
CCc1ccc(cc1-c1cccc(c1)-c1cnc2cnccn12)C(=O)Nc1cccc(c1)C(F)(F)F
CCc1ccc(cc1-c1cccc(c1)-c1cnc2cnccn12)C(=O)Nc1ccccc1
CCc1ccc(cc1-c1cccc(c1)-c1cnc2cnccn12)C(=O)Nc1ccccc1C(F)(F)F
CCc1ccc(cc1C#Cc1ccc2ccnn2c1)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1C#Cc1ccco1)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1C#Cc1ccoc1)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1C#Cc1ccsc1)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1C#Cc1cnc(C)n1C)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1C#Cc1cnc(N)nc1)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1C#Cc1cnc(NC)nc1)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1C#Cc1cnc(nc1)N(C)C)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1C#Cc1cnc2ccccn12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1C#Cc1cnc2cccnn12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1C#Cc1cnc2cnccn12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1C#Cc1cncn1C)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc(cc1C#Cc1cncnc1)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F
CCc1ccc2n(C)c(C)c(C(=O)Nc3ccc(Oc4ncnc5cc(OC)c(OC)cc45)c(F)c3)c(=O)c2c1
CCc1cccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)c12
CCc1nc(C)c(o1)C(=O)NNc1cc(Cl)ccc1S(=O)(=O)CC |$;;;;;;;;;;;HN;;;;;;;;;;;;$|
CCn1c(nc2c(ncc(OC[C@H]3CCCNC3)c12)C#CC(C)(C)O)-c1nonc1N |r|
CCn1cc(-c2ccc3N(CCc3c2)C(=O)Cc2cccc(OC(F)(F)F)c2)c2c(N)ncnc12
CCn1cc(cn1)N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
CCn1ccc(n1)N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
CCn1nc(C#Cc2cc(ccc2C)C(=O)Nc2ccc(CN3CCN(C)CC3)c(c2)C(F)(F)F)c2c(N)ncnc12
CN(C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br)c1cc(C)on1
CN(C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2C)C(C)(C)C
CN(C)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
CN(C)CC(=O)N1CCC(CC1)c1ccc(NC(=O)c2ncc([nH]2)C#N)c(c1)C1=CCCCC1 |t:31|
CN(C)CCC1CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
CN(C)CCN(CC(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
CN(C)CCN(CC(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
CN(C)CCN(Cc1ccc(cc1)C(=O)Nc1ccc(C)c(Nc2nccc(n2)-c2cccnc2)c1)C(=O)c1cccnc1
CN(C)CCNC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
CN(C)CCOC(=O)N1CCN(CC1)c1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
CN(C)C[C@@H]1CCn2cc(C3=C(C(=O)NC3=O)c3cn(CCO1)c1ccccc31)c1ccccc21 |r,t:10|
CN(C)C\C=C\C(=O)Nc1cc(ccc1C)-n1c2c(ccc3ccc(cc23)-c2cnn(C)c2)ccc1=O
CN(C)C\C=C\C(=O)Nc1cc2c(Nc3ccc(F)c(Cl)c3)ncnc2cc1O[C@H]1CCOC1 |r|
CN(C)[C@@H]1CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O |r|
CN(C)[C@@H]1CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
CN(C)[C@@H]1CN(C[C@@H]1F)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3n2)c2c1ccc(F)c2Cl |r|
CN(C)[C@H]1CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
CN(C)c1ccc2c(Oc3ccc(NC(=O)NCc4ccc(nc4)C(F)(F)F)cc3)ncnc2c1
CN(C)c1cccc(NC(=O)c2ccc(C)c(c2)C#Cc2cnc3ccnn3c2)c1
CN(CC#N)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
CN(CC(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cc3cn[nH]c3cn2)C1=O
CN(CC(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
CN(CC(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
CN(CC1COC1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
CN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(C)cc(c1)-n1cnc(C)c1)c1cncnc1 |r|
CN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(cc(c1)-n1cnc(C)c1)C1CCCCC1)c1cncnc1 |r|
CN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(cc(c1)C(C)(C)C)-n1cnc(C)c1)c1cncnc1 |r|
CN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1)c1cncnc1 |r|
CN([C@@H]1Cc2ccc(cc2C1)C(=O)Nc1cc(cc(c1)C12CC3CC(CC(C3)C1)C2)-n1cnc(C)c1)c1cncnc1 |r,TLB:18:20:23:27.25.26,THB:25:24:21:27.26.28,25:26:23.24.29:21,28:26:23:29.20.21,28:20:23:27.25.26|
CN(c1ccc2c(C)n(C)nc2c1)c1ccnc(Nc2ccc(C)c(c2)S(N)(=O)=O)n1
CN1CCC(CC1)n1nc(C#Cc2cc(NC(=O)c3cccc(c3)C(F)(F)F)ccc2C)c2c(N)ncnc12
CN1CCCC(N2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)C2=O)C1=O
CN1CCN(C(C1)C(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
CN1CCN(CC1(C)C)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
CN1CCN(CC1(C)C)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
CN1CCN(CC1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
CN1CCN(CC1)c1cc(Nc2cc(C)n[nH]2)nc(Sc2ccc(NC(=O)C3CC3)cc2)n1
CN1CCN(CC1)c1ccc2nc([nH]c2c1)-c1c(N)c2c(F)cccc2[nH]c1=O
CN1CCN(CC1C(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
CN1CCN(CC1C(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
CN1CCN(C[C@@H]1C(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O |r|
CN1CCN(C[C@H]1C(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O |r|
CN1CCN(Cc2cc(C)cc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ccnn4c3)c2)CC1
CN1CCN(Cc2cc(Cl)cc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ccnn4c3)c2)CC1
CN1CCN(Cc2cc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ccnn4c3)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4cnccn34)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3ccc(C4CC4)c(c3)C#Cc3cnc4cnccn34)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3ccc(Cl)c(c3)C#Cc3cnc4ccnn4c3)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3ccc(c(c3)C#Cc3cnc4cnccn34)C(C)(C)C)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3ccc4CCN(Cc4c3)c3ccccc3)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3ccc4CCN(Cc4c3)c3cccnc3)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3ccc4CCN(Cc4c3)c3ccncn3)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3ccc4CCN(Cc4c3)c3cnc4ccccc4c3)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3ccc4CCN(Cc4c3)c3cncnc3)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3ccc4CCN(Cc5cncnc5)Cc4c3)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3ccc4c(CN(CC4(C)C)c4cncnc4)c3)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(NC(=O)c3cccc(c3)C#Cc3cnc4ccnn4c3)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(Nc3noc4c(C#Cc5cnc6cccnn56)c(C)ccc34)cc(c2)C(F)(F)F)CC1
CN1CCN(Cc2cc(cc(c2)C(F)(F)F)C(=O)Nc2ccc3CCN(Cc3c2)c2cncnc2)CC1
CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4cccnn34)cc2C(F)(F)F)CC1
CN1CCN(Cc2ccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ccnn4c3)cc2C(F)(F)F)CC1
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nc(cs3)-c3cccnc3)c2)CC1
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)CC1
CN1CCN(Cc2ccc(cc2)C(=O)Nc2ccc(C)c(Oc3ccc(cc3)-c3n[nH]c4ncnc(N)c34)c2)CC1
CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(OC3CCN(CC3)C(=O)c3ccc(C)nc3)c2)CC1
CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2ccc(C)c(Oc3ccc(cc3)-c3n[nH]c4ncnc(N)c34)c2)CC1
CN1CCN(Cc2ccc(cc2C(F)(F)F)C(=O)Nc2cccc(Oc3ccc(cc3)-c3n[nH]c4ncnc(N)c34)c2)CC1
CN1CCN(Cc2ccc(cc2I)C(=O)Nc2ccc(C)c(Oc3ccc(cc3)-c3n[nH]c4ncnc(N)c34)c2)CC1
CN1CCN(Cc2cccc(NC(=O)c3ccc(C)c(c3)C#Cc3cnc4ccnn4c3)c2)CC1
CN1CCN(Cc2cccc(c2)C(=O)Nc2ccc(C)c(Oc3ccc(cc3)-c3n[nH]c4ncnc(N)c34)c2)CC1
CN1CCN(Cc2cccc(c2)[C@H]2C[C@@H]2NC(=O)CN2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)C2=O)CC1 |r|
CN1CCN(Cc2ccccc2C2CC2NC(=O)CN2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)C2=O)CC1
CN1CCNC(=O)CCCCOc2cc(C#Cc3cnc4ccc1nn34)c(C)c(c2)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1
CN1CC[C@@H]([C@H](O)C1)c1c(O)cc(O)c2c1oc(cc2=O)-c1ccccc1Cl |r|
CNC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
CNC(=O)Cc1cccc(CNC(=O)CN2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)C2=O)c1
CNC(=O)c1c(F)cccc1Nc1nc(Nc2cc3N(CCc3cc2OC)C(=O)CN(C)C)nc2[nH]ccc12
CNC(=O)c1cc(Oc2ccc(NC(=O)Nc3ccc(Cl)c(c3)C(F)(F)F)cc2)ccn1
CNC(=O)c1ccccc1Sc1ccc2c(\C=C\c3ccccn3)n[nH]c2c1
CNS(=O)(=O)Nc1cccc(Cc2c(C)c3cc(Cl)c(OC(=O)N(C)C)cc3oc2=O)c1
CN[C@@H]1C[C@H]2O[C@@](C)([C@@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r|
CN[C@H]1CCCN(Cc2c(Cl)cc(cc2C(F)(F)F)C(=O)NCc2cc(Cl)ccc2S(=O)(=O)C(C)C)C1 |r|
CN[C@H]1CCCN(Cc2c(Cl)cc(cc2C(F)(F)F)C(=O)NCc2cc(Cl)ccc2S(=O)(=O)C2CCCC2)C1 |r|
CN[C@H]1CCCN(Cc2c(Cl)cc(cc2C(F)(F)F)C(=O)NCc2cc(Cl)ccc2S(=O)(=O)c2ccccc2)C1 |r|
CN[C@H]1C[C@@H]2O[C@](C)([C@H]1OC)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13
CNc1nc(Nc2ccc(C)c(N)c2)ncc1C(=O)Nc1cc(NC(=O)c2cccc(c2)C(F)(F)F)ccc1C
CNc1nc(Nc2ccc(C)c(NC(=O)C=C)c2)ncc1C(=O)Nc1cc(NC(=O)c2cc(OC)c(OC)c(OC)c2)ccc1C
CNc1ncc2c(nn(CC3CCCC3)c2n1)-c1ccc(cc1)N1CCN(C)CC1
CNc1ncc2c(nn(CC3CCCC3)c2n1)-c1ccc(nc1)N1CCN(C)CC1
COC(=O)N1CCC(C1)c1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
COC(=O)N1CCN(CC1)c1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
COC(=O)[C@@H]1CC(F)(F)CN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2c1cccc2C |r|
COC(=O)[C@@H]1CC(F)(F)CN1C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
COC(=O)c1ccc2\C(=C(\Nc3ccc(cc3)N(C)C(=O)CN3CCN(C)CC3)c3ccccc3)C(=O)Nc2c1
COC(=O)c1cccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
COC(=O)c1cccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)c12
COC(=O)c1n[nH]c2ccc(cc12)C(=O)N1CCC2(CC1)C(=O)N(CC(=O)NCC(F)(F)F)c1ccc(F)c(Cl)c21
COC1CCN(C1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1ccc(F)c2Cl
COC1CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
COCC(=O)NC\C=C\c1ccc2ncnc(Nc3ccc(Oc4ccc(C)nc4)c(C)c3)c2c1
COCC1CCCN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1ccc(F)c2Cl
COCCOc1cc2ncnc(Nc3cccc(c3)C#C)c2cc1OCCOC
COC[C@H]1CCCN1C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O |r|
CO[C@@H]1[C@@H](C[C@H]2O[C@]1(C)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1 |r|
CO[C@@H]1[C@@H](C[C@H]2O[C@]1(C)n1c3ccccc3c3c4[C@H](O)NC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1 |r|
COc1c(Cl)cc2c3ccncc3[nH]c2c1NC(=O)c1cccnc1C
COc1cc(CN2CCN(C)CC2)cc(NC(=O)c2ccc(C)c(c2)C#Cc2cnc3ccnn3c2)c1
COc1cc(Nc2c(cnc3cc(OCCCN4CCN(C)CC4)c(OC)cc23)C#N)c(Cl)cc1Cl
COc1cc(Nc2ncc(F)c(Nc3ccc4OC(C)(C)C(=O)Nc4n3)n2)cc(OC)c1OC
COc1cc(Oc2ccnc3cc(OC)c(OC)cc23)ccc1NC(=O)NC(C)c1nccs1
COc1cc(cc(OC)c1OC)-c1cncc(c1C)-c1ccc(cc1)N1CCNCC1
COc1cc(ccc1Nc1ncc(Cl)c(Nc2ccccc2S(=O)(=O)C(C)C)n1)N1CCC(CC1)N1CCN(C)CC1
COc1cc2c(Nc3ccc(Br)cc3F)ncnc2cc1OCC1CCN(C)CC1
COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)NC4=CCC(F)C=C4)cc3F)ccnc2cc1OCCCN1CCOCC1 |c:26,t:21|
COc1cc2c(Oc3ccc(NC(=O)C4(CC4)C(=O)Nc4ccc(F)cc4)cc3F)ccnc2cc1OCCCN1CCOCC1
COc1cc2c(Oc3ccc(Nc4nn(C)cc4C(=O)NC4CCCCC4)cc3F)ccnc2cc1OCCCN1CCOCC1
COc1cc2c(Oc3ccc4[nH]c(C)cc4c3F)ncnc2cc1OCCCN1CCCC1
COc1cc2c(ncnc2cc1OCCCN1CCCCC1)N1CCN(CC1)C(=O)Nc1ccc(OC(C)C)cc1
COc1cc2ncc(-c3cccc(NC4CCNC4)n3)n2cc1-c1cnn(C)c1
COc1cc2nccc(Oc3ccc(NC(=O)Cc4ccc(Cl)c(c4)C(F)(F)F)cc3)c2cc1OC
COc1cc2ncccc2cc1NC(=O)c1csc2cncnc12
COc1cc2ncnc(Nc3ccc(F)c(Cl)c3)c2cc1OCCCN1CCOCC1
COc1ccc(COc2ccc(Cc3cnc(N)nc3N)cc2OC)cc1
COc1ccc(F)c(F)c1C(=O)c1cnc(NC2CCN(CC2)S(C)(=O)=O)nc1N
COc1ccc(NC(=O)c2ccc(C)c(c2)C#Cc2cnc3ccnn3c2)cc1
COc1ccc(cc1\C=C\c1ccc(Cl)cc1)C(=O)NC[C@@H](O)CO |r|
COc1ccc(cc1\C=C\c1ccc(Cl)cc1)C(=O)NC[C@H](O)CO |r|
COc1ccc2N(CC(=O)N3CCC[C@H]3C(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c2n1 |r|
COc1ccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c2n1
COc1cccc(NC(=O)c2ccc(C)c(c2)C#Cc2cnc3ccnn3c2)c1
COc1cccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)c12
COc1cccc2nc(Nc3cccc(NC(=O)c4ccc(N5CCN(C)CC5)c(c4)C(F)(F)F)c3)ccc12
COc1ccccc1NC(=O)c1ccc(C)c(c1)C#Cc1cnc2ccnn2c1
COc1cncc(CNc2cc(ccc2C)C(=O)Nc2cccc(c2)C(F)(F)F)c1
CS(=O)(=O)CCNCc1ccc(o1)-c1ccc2ncnc(Nc3ccc(OCc4cccc(F)c4)c(Cl)c3)c2c1
CS(=O)(=O)N1CCCC(C1)NC(=O)[C@H](CCC1CCCCC1)NC(=O)c1ccc(CNC(=O)c2cc(n[nH]2)-c2ccccc2)cc1 |r|
CS(=O)(=O)N1CCCC(C1)NC(=O)[C@H](CCC1CCCCC1)NC(=O)c1ccc(CNC(=O)c2cnc3ccccn23)cc1
CS(=O)(=O)N1CCCC(C1)NC(=O)[C@H](CCC1CCCCC1)NC(=O)c1ccc(CNc2ncnc3n(ncc23)-c2ccccc2)cc1 |r|
CS(=O)(=O)N1CCCC(C1)NC(=O)[C@H](CCC1CCCCC1)NC(=O)c1ccc(CNc2ncnc3n(nnc23)-c2ccccc2)cc1
CS(=O)(=O)N1CCC[C@@H](C1)NC(=O)[C@H](CCC1CCCCC1)NC(=O)c1ccc(CNC(=O)c2cnn(c2N)-c2ccccc2)cc1 |r|
CS(=O)(=O)N1CCN(Cc2cc3nc(nc(N4CCOCC4)c3s2)-c2cccc3[nH]ncc23)CC1
CS(=O)(=O)c1ccc(F)cc1CNC(=O)c1cccc(c1)C(F)(F)F
CS(=O)(=O)c1ccc(F)cc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CS(=O)(=O)c1ccc(F)cc1Cn1cnc2ccc(cc2c1=O)C(F)(F)F
CS(=O)(=O)n1cccc1Cn1c(=O)[nH]c2ccc(cc2c1=O)C(F)(F)F
CS(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1
CSc1ccc(F)cc1CNC(=O)c1cccc(c1)C(F)(F)F
CSc1cccc(Nc2ncc3cc(-c4c(Cl)cccc4Cl)c(=O)n(C)c3n2)c1 |(-12.18,1.86,;-10.84,1.09,;-9.51,1.86,;-9.51,3.4,;-8.18,4.17,;-6.84,3.4,;-6.84,1.86,;-5.51,1.08,;-4.18,1.85,;-4.18,3.39,;-2.84,4.16,;-1.51,3.4,;-.18,4.17,;1.16,3.4,;2.49,4.17,;2.49,5.71,;1.16,6.48,;3.83,6.48,;5.16,5.71,;5.16,4.17,;3.83,3.39,;3.83,1.85,;1.16,1.86,;2.49,1.09,;-.18,1.09,;-.18,-.45,;-1.51,1.86,;-2.84,1.08,;-8.18,1.08,)|
C[C@@H](N(C)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2C)C(F)(F)F |r|
C[C@@H](N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)C(=O)NCC(F)(F)F |r|
C[C@@H](NC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2C)C(F)(F)F |r|
C[C@@H](NC(=O)Nc1ccccc1)c1ccc(C)c(NC(=O)c2cnc3ccccn23)c1 |r|
C[C@@H](O)COc1cn2ncnc(Oc3ccc4[nH]c(C)cc4c3F)c2c1C
C[C@@H](Oc1cc(cnc1N)-c1cnn(c1)C1CCNCC1)c1c(Cl)ccc(F)c1Cl |r|
C[C@@H](Oc1cc(sc1C(N)=O)-n1cnc2ccc(CN3CCN(C)CC3)cc12)c1ccccc1C(F)(F)F |r|
C[C@@H]1CCN(C[C@@H]1N(C)c1ncnc2[nH]ccc12)C(=O)CC#N |r|
C[C@@H]1CN(Cc2cc(NC(=O)c3cc(CN4CCN(C)CC4)cc(c3)C(F)(F)F)ccc12)c1cncnc1 |r|
C[C@@H]1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1 |r|
C[C@@H]1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1 |r|
C[C@@H]1CN(Cc2cc(ccc12)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1)c1cncnc1 |r|
C[C@H](N(C)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2C)C(F)(F)F |r|
C[C@H](N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)C(=O)NCC(F)(F)F |r|
C[C@H](NC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2C)C(F)(F)F |r|
C[C@H](NC(=O)Nc1ccccc1)c1ccc(C)c(NC(=O)c2cnc3ccccn23)c1 |r|
C[C@H]1CN(C[C@@H](C)O1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2C |r|
C[C@H]1CN(C[C@@H]1O)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
C[C@H]1CN(C[C@H]1O)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
C[C@H]1CN(Cc2cc(NC(=O)c3cc(CN4CCN(C)CC4)cc(c3)C(F)(F)F)ccc12)c1cncnc1 |r|
C[C@H]1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1 |r|
C[C@H]1CN(Cc2cc(ccc12)C(=O)Nc1cc(CN2CCN(C)CC2)cc(c1)C(F)(F)F)c1cncnc1 |r|
C[C@H]1CN(Cc2cc(ccc12)C(=O)Nc1cc(cc(c1)C(F)(F)F)-n1cnc(C)c1)c1cncnc1 |r|
C[C@]12O[C@H](C[C@]1(O)CO)n1c3ccccc3c3c4C(=O)NCc4c4c5ccccc5n2c4c13 |r|
C\C=C\C(=O)N1CCN(CC1)c1cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)nc(C)n1
Cc1[nH]c(\C=C2/C(=O)Nc3ccc(F)cc23)c(C)c1C(=O)NC[C@H](O)CN1CCOCC1
Cc1[nH]c(\C=C2/C(=O)Nc3ccc(cc23)S(=O)(=O)Cc2c(Cl)cccc2Cl)c(C)c1C(=O)N1CCC[C@@H]1CN1CCCC1 |r|
Cc1c(oc2cc(ccc12)C(=O)Nc1cccc(c1)C(F)(F)F)-c1n(nc2c1c(N)n[nH]c2=O)-c1ccc(C)cc1 |(51.37,-34.33,;51.52,-32.79,;50.38,-31.77,;51,-30.36,;52.53,-30.51,;53.66,-29.49,;55.12,-29.95,;55.45,-31.46,;54.31,-32.48,;52.85,-32.01,;56.26,-28.91,;55.93,-27.41,;57.73,-29.38,;58.86,-28.35,;60.33,-28.82,;61.47,-27.78,;61.14,-26.28,;59.66,-25.81,;58.53,-26.85,;59.33,-24.31,;60.47,-23.26,;57.86,-23.84,;58.92,-22.81,;48.87,-32.09,;48.25,-33.49,;46.74,-33.33,;46.42,-31.84,;47.73,-31.07,;47.73,-29.53,;49.07,-28.77,;46.4,-28.76,;45.07,-29.53,;45.07,-31.07,;43.74,-31.85,;49.03,-34.82,;48.26,-36.15,;49.03,-37.48,;50.57,-37.48,;51.35,-38.81,;51.34,-36.14,;50.56,-34.81,)|
Cc1c(oc2cc(ccc12)C(=O)Nc1cccc(c1)C(F)(F)F)-c1n(nc2c1c(N)n[nH]c2=O)-c1ccc(F)cc1 |(10.15,-36.25,;10.3,-34.72,;9.15,-33.69,;9.78,-32.28,;11.31,-32.44,;12.44,-31.41,;13.9,-31.87,;14.22,-33.38,;13.08,-34.41,;11.63,-33.94,;15.03,-30.84,;14.71,-29.33,;16.5,-31.3,;17.64,-30.27,;19.11,-30.74,;20.25,-29.7,;19.92,-28.2,;18.44,-27.73,;17.31,-28.77,;18.11,-26.23,;19.24,-25.19,;16.64,-25.76,;17.7,-24.73,;7.65,-34.01,;7.03,-35.41,;5.51,-35.25,;5.19,-33.76,;6.51,-33,;6.51,-31.46,;7.85,-30.69,;5.18,-30.68,;3.85,-31.46,;3.85,-33,;2.52,-33.77,;7.8,-36.74,;7.03,-38.08,;7.81,-39.41,;9.35,-39.4,;10.12,-40.74,;10.12,-38.06,;9.34,-36.73,)|
Cc1c(oc2cc(ccc12)C(=O)Nc1cccc(c1)C(F)(F)F)-c1n(nc2c1c(N)n[nH]c2=O)-c1ccccc1 |(72.02,-33.45,;72.18,-31.91,;71.03,-30.89,;71.65,-29.48,;73.19,-29.63,;74.32,-28.61,;75.77,-29.07,;76.1,-30.58,;74.96,-31.61,;73.51,-31.13,;76.91,-28.04,;76.58,-26.53,;78.38,-28.5,;79.52,-27.47,;80.99,-27.94,;82.12,-26.9,;81.8,-25.4,;80.32,-24.93,;79.19,-25.97,;79.98,-23.43,;81.12,-22.38,;78.52,-22.96,;79.57,-21.93,;69.52,-31.21,;68.91,-32.61,;67.39,-32.45,;67.07,-30.96,;68.39,-30.2,;68.39,-28.65,;69.73,-27.89,;67.06,-27.88,;65.73,-28.65,;65.73,-30.2,;64.4,-30.97,;69.68,-33.94,;68.91,-35.27,;69.68,-36.61,;71.23,-36.6,;71.99,-35.26,;71.22,-33.93,)|
Cc1cc(C)cc(NC(=O)c2ccc(C)c(c2)C#Cc2cnc3ccnn3c2)c1
Cc1cc(Cl)cc(NC(=O)c2ccc(C)c(c2)C#Cc2cnc3ccnn3c2)c1
Cc1cc(F)c(cc1Cl)N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
Cc1cc(N2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)C2=O)n(C)n1
Cc1cc(NC(=O)Nc2cc(nn2-c2ccc(Cl)cc2)C(C)(C)C)ccc1Nc1ncnc2NC(=O)C(C)(C)Oc12
Cc1cc(Nc2noc3c(C#Cc4cnc5cccnn45)c(C)ccc23)cc(c1)C(F)(F)F
Cc1cc(cc2cn[nH]c12)C(=O)N1CCC2(CC1)N(CN(CC(=O)NCC(F)(F)F)C2=O)c1ccccc1
Cc1cc(nn1C)N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
Cc1ccc(-c2cn([C@@H]3CC[C@H](N)CC3)c3ncnc(N)c23)c(F)c1 |r,wU:8.7,11.11,(2.17,7.19,;1.77,5.71,;.28,5.31,;-.11,3.82,;.97,2.74,;.58,1.25,;1.48,0,;.58,-1.24,;.97,-2.73,;-.11,-3.82,;.28,-5.31,;1.77,-5.71,;2.17,-7.19,;2.86,-4.62,;2.46,-3.13,;-.89,-.77,;-2.22,-1.54,;-3.56,-.77,;-3.56,.77,;-2.22,1.54,;-2.22,3.08,;-.89,.77,;2.47,3.14,;3.56,2.05,;2.86,4.62,)|
Cc1ccc(F)c(NC(=O)Nc2ccc(cc2)-c2cccc3[nH]nc(N)c23)c1
Cc1ccc(N2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)C2=O)c(F)c1
Cc1ccc(NC(=O)c2ccc(C)c(c2)C#Cc2cnc3ccnn3c2)cc1
Cc1ccc(NC(=O)c2ccc(C)c(c2)C(F)(F)F)cc1C#Cc1nn([C@H]2CC[C@H](O)CC2)c2ncnc(N)c12 |r,wU:26.27,wD:29.31,(-5.46,5.4,;-3.98,5.8,;-3.58,7.29,;-2.09,7.69,;-1,6.6,;.49,7,;1.57,5.91,;1.18,4.42,;3.06,6.31,;3.46,7.79,;4.95,8.19,;6.04,7.1,;7.53,7.5,;5.64,5.62,;4.15,5.22,;6.73,4.53,;8.22,4.93,;6.33,3.04,;7.82,3.44,;-1.4,5.11,;-2.89,4.71,;-3.29,3.22,;-3.68,1.74,;-4.08,.25,;-3.18,-1,;-4.08,-2.24,;-3.68,-3.73,;-2.2,-4.13,;-1.8,-5.62,;-2.89,-6.7,;-2.49,-8.19,;-4.38,-6.31,;-4.77,-4.82,;-5.55,-1.77,;-6.88,-2.54,;-8.22,-1.77,;-8.22,-.23,;-6.88,.54,;-6.88,2.08,;-5.55,-.23,)|
Cc1ccc(NC(=O)c2ccc(CN3CCCC3)c(c2)C(F)(F)F)cc1Oc1ccc(cc1)-c1n[nH]c2ncnc(N)c12
Cc1ccc(NC(=O)c2ccc(CN3CCCCC3)c(c2)C(F)(F)F)cc1Oc1ccc(cc1)-c1n[nH]c2ncnc(N)c12
Cc1ccc(NC(=O)c2ccc(CN3CCOCC3)c(Br)c2)cc1Oc1ccc(cc1)-c1n[nH]c2ncnc(N)c12
Cc1ccc(NC(=O)c2ccc(CN3CCOCC3)c(Cl)c2)cc1Oc1ccc(cc1)-c1n[nH]c2ncnc(N)c12
Cc1ccc(NC(=O)c2ccc(CN3CCOCC3)c(F)c2)cc1Oc1ccc(cc1)-c1n[nH]c2ncnc(N)c12
Cc1ccc(NC(=O)c2ccc(CN3CCOCC3)c(c2)C(F)(F)F)cc1Oc1ccc(cc1)-c1n[nH]c2ncnc(N)c12
Cc1ccc(NC(=O)c2cccc(c2)C(F)(F)F)cc1OC1CCN(CC1)C(=O)c1ccncc1
Cc1ccc(NC(=O)c2ccnc(c2)C(F)(F)F)cc1-c1cc(OCCO)nc(c1)N1CCOCC1
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1ccc(OCCN2CCOCC2)c2ccccc12)C(C)(C)C
Cc1ccc(cc1)-n1nc(cc1NC(=O)Nc1nc(CCOCc2ccncc2)cs1)C(C)(C)C
Cc1ccc(cc1-c1cccc(c1)-c1cnc2cnccn12)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)NC1CCCC1
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)NC1CCCCC1
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)Nc1cc(CN2CCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)Nc1cc(CN2CCCCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)Nc1cc(CN2CCOCC2)cc(c1)C(F)(F)F
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)Nc1ccc(Cl)cc1
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)Nc1ccc(cc1)C(F)(F)F
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)Nc1cccc(Br)c1
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)Nc1cccc(Cl)c1
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)Nc1cccc(I)c1
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)Nc1cccc(c1)-n1ccnc1
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)Nc1ccccc1
Cc1ccc(cc1C#Cc1cnc2ccnn2c1)C(=O)Nc1ccccc1Cl
Cc1ccc(cc1NC(=O)C1(CC1)c1ncnc2[nH]cnc12)C(=O)Nc1ccc(Cl)c(c1)C(F)(F)F
Cc1ccc(cc1NCc1cccnc1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1NCc1cncc(c1)-c1ccc[nH]1)C(=O)Nc1ccc(C)c(c1)C(F)(F)F
Cc1ccc(cc1NCc1cncc(c1)-c1ccc[nH]1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1NCc1cncc(c1)-c1ccn(C)n1)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1NCc1cncc(c1)C(N)=O)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc(cc1Nc1cncc(c1)C(N)=O)C(=O)Nc1cccc(c1)C(F)(F)F
Cc1ccc2c(Nc3cc(CN4CCCC4)cc(c3)C(F)(F)F)noc2c1C#Cc1cnc2cccnn12
Cc1ccc2c(Nc3cc(CN4CCOCC4)cc(c3)C(C)(C)C#N)noc2c1C#Cc1cnc2cccnn12
Cc1ccc2c(Nc3cc(CN4CCOCC4)cc(c3)C(F)(F)F)noc2c1C#Cc1cnc2cccnn12
Cc1ccc2c(Nc3cc(CNC4CC4)cc(c3)C(F)(F)F)noc2c1C#Cc1cnc2cccnn12
Cc1ccc2c(Nc3cc(Cn4ccnc4)cc(c3)C(F)(F)F)noc2c1C#Cc1cnc2cccnn12
Cc1ccc2c(Nc3cc(cc(c3)C(C)(C)C#N)C(F)(F)F)noc2c1C#Cc1cnc2cccnn12
Cc1ccc2c(Nc3ccc(Cl)cc3)nccc2c1NC(=O)c1csc2c(N)ncnc12
Cc1ccc2c(Nc3ccc(F)c(Cl)c3)nccc2c1NC(=O)c1csc2c(N)ncnc12
Cc1ccc2c(Nc3cccc(Cl)c3)nccc2c1NC(=O)c1csc2c(N)ncnc12
Cc1ccc2c(Nc3cccc(Cl)c3F)nccc2c1NC(=O)c1csc2c(N)ncnc12
Cc1ccc2c(Nc3cccc(OC(F)(F)F)c3)noc2c1C#Cc1cnc2cccnn12
Cc1ccc2c(Nc3cccc(c3)C(C)(C)C#N)noc2c1C#Cc1cnc2cccnn12
Cc1ccc2c(Nc3cccc(c3)C(F)(F)F)noc2c1C#Cc1cnc2cccnn12
Cc1ccc2c(Nc3cncc(c3)C(F)(F)F)noc2c1C#Cc1cnc2cccnn12
Cc1cccc(CN2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)C2=O)n1
Cc1cccc(Cl)c1NC(=O)c1cnc(Nc2cc(nc(C)n2)N2CCN(CC2)C(=O)Oc2ccccc2)s1
Cc1cccc(NC(=O)c2ccc(C)c(c2)C#Cc2cnc3ccnn3c2)c1
Cc1cccc2N(CC(=O)N3CC(O)C(C)(C)C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)N3CC(O)C(F)(F)C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)N3CCC(C)(F)C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)N3CCC(C3)C#N)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)N3CCC(F)(F)C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)N3CCC(O)(C3)C(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)N3CCC[C@H]3C(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3cc4cn[nH]c4cn3)c12 |r|
Cc1cccc2N(CC(=O)N3CCC[C@H]3C(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c12 |r|
Cc1cccc2N(CC(=O)N3CCC[C@H]3C(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)c12 |r|
Cc1cccc2N(CC(=O)N3CCOC(C3)C(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)NC(C)(C)C#N)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)NC(C)(C)C)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)NC(C)(C)CO)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)NC3(C)COC3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)NC3(CC3)C(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)NC3CCCCC3(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)NC3CCCc4ccccc34)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)NC3CCc4ccccc34)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c12
Cc1cccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)c12
Cc1cccc2N(CC(=O)NCCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(CCC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1cccc2N(Cc3nc(no3)C3CC3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Cc1ccccc1NC(=O)c1ccc(C)c(c1)C#Cc1cnc2ccnn2c1
Cc1cn(cn1)-c1cc(NC(=O)c2ccc(C)c(Nc3nccc(n3)-c3cccnc3)c2)cc(c1)C(F)(F)F
Cc1cn(cn1)-c1cc(NC(=O)c2ccc3CC(C)(Cc3c2)Nc2cncnc2)cc(c1)C(F)(F)F
Cc1cn(cn1)-c1cc(NC(=O)c2ccc3CN(Cc3c2)c2cncnc2)cc(c1)C(F)(F)F
Cc1cn(cn1)-c1cc(NC(=O)c2ccc3CN(Cc4cncnc4)Cc3c2)cc(c1)C(F)(F)F
Cc1cn(cn1)-c1cc(NC(=O)c2ccc3C[C@@H](Cc3c2)Nc2cncnc2)cc(c1)C(F)(F)F |r|
Cc1cn(cn1)-c1cc(NC(=O)c2ccc3C[C@H](Cc3c2)Nc2cncnc2)cc(c1)C(F)(F)F |r|
Cc1cn(cn1)-c1cc(Nc2noc3c(C#Cc4cnc5cccnn45)c(C)ccc23)cc(c1)C(F)(F)F
Cc1cn(cn1)-c1cccc(NC(=O)c2ccc(C)c(c2)C#Cc2cnc3ccnn3c2)c1
Cc1cnc(Nc2ccc(OCCN3CCCC3)cc2)nc1Nc1cccc(c1)S(=O)(=O)NC(C)(C)C
Cc1cnc2c(NCCN)nc3ccc(C)cc3n12
Cc1n[nH]c2ccc(cc12)-c1cncc(OC[C@@H](N)Cc2ccccc2)c1 |r|
Cc1n[nH]c2ccc(cc12)C(=O)N1CCC2(CC1)N(CN(CC(=O)NCC(F)(F)F)C2=O)c1ccccc1
Cc1nc(C)c(s1)N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
Cc1nc(CN2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)C2=O)cs1
Cc1nc(NC2CCN(C2)C(=O)C=C)cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)n1
Cc1nc(NC2CCN(C2)S(C)(=O)=O)cc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)n1
Cc1nc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)cc(n1)C1CCN(C1)C(=O)OCC=C
Cc1nc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)cc(n1)C1CCN(C1)C(=O)OCc1ccccc1
Cc1nc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)cc(n1)C1CCN(C1)C(=O)Oc1ccccc1
Cc1nc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)cc(n1)N1CCN(CC1)C(=O)C=C
Cc1nc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)cc(n1)N1CCN(CC1)C(=O)OCC=C
Cc1nc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)cc(n1)N1CCN(CC1)C(=O)OCCCl
Cc1nc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)cc(n1)N1CCN(CC1)C(=O)OCCN1CCOCC1
Cc1nc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)cc(n1)N1CCN(CC1)C(=O)OCc1ccccc1
Cc1nc(Nc2ncc(s2)C(=O)Nc2c(C)cccc2Cl)cc(n1)N1CCN(CCO)CC1
Cc1nc2n(ncc2cc1Nc1c(F)cccc1Cl)-c1csc(c1)C(=O)NC1COC1
Cc1nnc(CN2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)C2=O)o1
Cc1noc(CN2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)C2=O)n1
Cc1noc(n1)[C@@H]1CNC[C@H]1NC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O |r|
Cc1oc(nc1CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)C(C)(C)C
Clc1ccc(Nc2nnc(Cc3ccncc3)c3ccccc23)cc1
Clc1cccc(Cl)c1C(=O)Nc1cn[nH]c1C(=O)NC1CCNCC1
Clc1cccc(c1)N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
Clc1cccc2N(Cc3nc(no3)C3CC3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
Clc1ccccc1NC(=O)NCc1cccnc1
Cn1c(Nc2ccc(cc2)C(F)(F)F)nc2cc(Oc3ccnc(c3)-c3ncc([nH]3)C(F)(F)F)ccc12
Cn1c2nc(NC(CCO)CCO)ncc2cc(Oc2ccc(F)cc2F)c1=O
Cn1c2nc(NC3CCOCC3)ncc2cc(Oc2ccc(F)cc2F)c1=O
Cn1c2nc(Nc3ccc4[nH]ccc4c3)ncc2cc(c1=O)S(=O)(=O)c1ccc(F)cc1F
Cn1cc(C2=C(C(=O)NC2=O)c2cn(C3CCN(Cc4ccccn4)CC3)c3ccccc23)c2ccccc12 |t:4|
Cn1cc(cn1)-c1ccc2nnc(Sc3ccc4ncccc4c3)n2n1
Cn1ccc(n1)-c1cncc(CNc2cc(ccc2F)C(=O)Nc2cccc(OC(F)(F)F)c2)c1
Cn1ccnc1CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
Cn1cnc2c(F)c(Nc3ccc(Br)cc3Cl)c(cc12)C(=O)NOCCO
Cn1nc(cc1NC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)C(F)(F)F
Cn1ncc(C(=O)NCc2ccc(cc2)C(=O)N[C@@H](CCC2CCCCC2)C(=O)NC2CCCN(C2)S(C)(=O)=O)c1N |r|
Cn1nccc1CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
FC(F)(F)C1(CC1)NC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
FC(F)(F)C1CCN(C1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cc3cn[nH]c3cn2)c2c1cccc2Br
FC(F)(F)C1CCN(C1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
FC(F)(F)C1CCN(C1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3n2)c2c1cccc2Br
FC(F)(F)C1CCN(C1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2c1cccc2Br
FC(F)(F)C1CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC(F)(F)C1CN(CCO1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
FC(F)(F)C1CN(CCO1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3n2)c2c1cccc2Br
FC(F)(F)C1CN(CCO1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2c1cccc2Br
FC(F)(F)C1CN(CCO1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC(F)(F)C1CN(Cc2ccccc2)CCN1C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
FC(F)(F)C1CNCCN1C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
FC(F)(F)CC1CCCN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
FC(F)(F)CC1CCCN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3n2)c2c1ccc(Cl)c2Cl
FC(F)(F)CC1CCCN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3n2)c2c1ccc(Cl)c2Cl |w:5.4|
FC(F)(F)CN(C1CC1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC(F)(F)CN1CCC(N2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)C2=O)C1=O
FC(F)(F)CN1CCCC(N2C(=O)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)c3c2cccc3Cl)C1=O |w:10.9|
FC(F)(F)CN1CC[C@@H](N2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)C2=O)C1=O |r|
FC(F)(F)CN1CC[C@H](N2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)C2=O)C1=O |r|
FC(F)(F)CNC(=O)C(CN1CCOCC1)N1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2c1cccc2Cl
FC(F)(F)CNC(=O)C(CN1CCOCC1)N1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2c1cccc2Cl |w:8.8|
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(C2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Cl
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(C2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Cl |w:13.12|
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(C2)C(=O)c2ccc3[nH]ncc3n2)c2c1cccc2Cl
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(C2)C(=O)c2cnc3[nH]ncc3c2)c2c1cccc2Cl
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cc3cn[nH]c3cn2)c2c1ccc(Cl)c2Cl
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cc3cn[nH]c3cn2)c2c1cccc2Br
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1ccc(Cl)c2Cl
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2C1CC1
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Cl
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2ccccc12
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3n2)c2c1ccc(Cl)c2Cl
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3n2)c2c1cccc2Br
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2c1ccc(Cl)c2Cl
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2c1cccc2Br
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2c1cccc2C#N
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2c1cccc2C(F)(F)F
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2c1cccc2Cl
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2cc(Br)ccc12
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2cc(Cl)ccc12
FC(F)(F)CNC(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ncc3[nH]ncc3n2)c2c1cccc2Br
FC(F)(F)CNC(=O)CN1C(=O)C2(CN(C2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
FC(F)(F)CNC(=O)CN1C(=O)C2(CN(C2)C(=O)c2ccc3[nH]ncc3n2)c2c1cccc2Br
FC(F)(F)CNC(=O)CN1CN(c2ccc(Cl)c(Cl)c2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2ccc(Cl)cc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2cccc(Br)c2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2cccc(Cl)c2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2cccc(c2)C#N)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2cccc(c2)C(F)(F)F)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cc3cn[nH]c3cn2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3n2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]nnc3c2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3cn[nH]c3c2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3cncn3c2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3nnnn3c2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC(F)(F)CNC(=O)CN1CN(c2cccnc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC(F)(F)Cn1ccc(NC(=O)CN2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)C2=O)n1
FC(F)(F)Oc1cc(Cl)c2ncn(Nc3cc(Cl)ccc3CC3CCCC3)c(=O)c2c1
FC(F)(F)Oc1ccc2ncn(Nc3cc(Cl)ccc3CC3CC3)c(=O)c2c1
FC(F)(F)Oc1ccc2ncn(Nc3cc(Cl)ccc3CC3CCC3)c(=O)c2c1
FC(F)(F)Oc1ccc2ncn(Nc3cc(Cl)ccc3S(=O)(=O)C3CC3)c(=O)c2c1
FC(F)(F)Oc1ccc2ncn(Nc3cc(Cl)ccc3S(=O)(=O)C3CCCC3)c(=O)c2c1
FC(F)(F)Oc1cccc(NC(=O)CN2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)C2=O)c1
FC(F)(F)[C@@H]1CCCN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cc3cn[nH]c3cn2)c2c1cccc2Br |r|
FC(F)(F)[C@@H]1CCCN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br |r|
FC(F)(F)[C@@H]1CCCN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Cl |r|
FC(F)(F)[C@@H]1CCCN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2nc(Cl)ccc12 |r|
FC(F)(F)[C@@H]1CCCN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3n2)c2c1cccc2Br |r|
FC(F)(F)[C@@H]1CCCN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2c1cccc2Br |r|
FC(F)(F)[C@@H]1CCCN1C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
FC(F)(F)[C@@H]1CN(CCN1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O |r|
FC(F)(F)[C@@H]1CN(CCO1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cc3cn[nH]c3cn2)C1=O |r|
FC(F)(F)[C@@H]1CN(CCO1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O |r|
FC(F)(F)[C@@H]1CN(CCO1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3n2)C1=O |r|
FC(F)(F)[C@@H]1CN(CCO1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
FC(F)(F)[C@H]1CCCN1C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
FC(F)(F)[C@H]1CN(CCN1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O |r|
FC(F)(F)[C@H]1CN(CCO1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cc3cn[nH]c3cn2)C1=O |r|
FC(F)(F)[C@H]1CN(CCO1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O |r|
FC(F)(F)[C@H]1CN(CCO1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3n2)C1=O |r|
FC(F)(F)[C@H]1CN(CCO1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
FC(F)(F)c1c(cnn1-c1ccccc1)C(=O)NCc1ccc(cc1)C(=O)NCCCC1CCCCC1
FC(F)(F)c1cc(Br)c2ncn(Nc3cc(Cl)ccc3S(=O)(=O)C3CC3)c(=O)c2c1
FC(F)(F)c1cc(Cl)c2ncn(Nc3cc(Cl)ccc3CC3CCC3)c(=O)c2c1
FC(F)(F)c1cc(Cl)c2ncn(Nc3cc(Cl)ccc3CC3CCCC3)c(=O)c2c1
FC(F)(F)c1cc(Cl)c2ncn(Nc3cc(Cl)ccc3S(=O)(=O)C3CC3)c(=O)c2c1
FC(F)(F)c1cc(Cl)cc(c1)C(=O)NCc1cc(Cl)ccc1S(=O)c1ccccc1
FC(F)(F)c1cc(Cl)cc(c1)C(=O)NCc1cc(Cl)ccc1Sc1ccccc1
FC(F)(F)c1cc(NC(=O)Nc2ccc3N(c4ccncc4)C(=O)c4cccnc4Oc3c2)ccc1Cl
FC(F)(F)c1ccc(Cl)c(c1)N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
FC(F)(F)c1ccc2[nH]c(=O)n(Cc3cc(Cl)ccc3S(=O)c3ccccc3)c(=O)c2c1
FC(F)(F)c1ccc2[nH]c(=O)n(Cc3cc(Cl)ccc3Sc3ccccc3)c(=O)c2c1
FC(F)(F)c1cccc(NC(=O)CN2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)C2=O)n1
FC(F)(F)c1cccc(c1)N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC(F)CNC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC1(F)CC11CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC1(F)CCCN(C1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
FC1(F)CCN(C1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cc3cn[nH]c3cn2)c2c1cccc2Br
FC1(F)CCN(C1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
FC1(F)CCN(C1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3n2)c2c1cccc2Br
FC1(F)CCN(C1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)c2c1cccc2Br
FC1(F)CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC1(F)CCN(CC1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
FC1(F)CN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
FC1CCN(C1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1ccc(F)c2Cl
FC1CCN(C1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
FCC1CN(CC1C(F)(F)F)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
FCCNC(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
FC[C@@H]1CC(F)(F)CN1C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br |r|
F[C@@H]1CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
F[C@H]1CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
F[C@H]1CN(C[C@H]1F)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br |r|
Fc1cc(Cl)cc(c1)N1CN(CC(=O)NCC(F)(F)F)C(=O)C11CCN(CC1)C(=O)c1cnc2[nH]ncc2c1
Fc1cc(Cl)ccc1N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
Fc1cc(ccc1N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)C(F)(F)F
Fc1ccc(Br)c2c1N(CC(=O)NCC(F)(F)F)C(=O)C21CCN(CC1)C(=O)c1cnc2[nH]ncc2c1
Fc1ccc(C(=O)NOCC2CC2)c(Nc2ccc(I)cc2Cl)c1F
Fc1ccc(Cl)cc1N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
Fc1ccc(Nc2ncnc3cc(OCCCN4CCOCC4)c(NC(=O)C=C)cc23)cc1Cl
Fc1ccc(Sc2ccc3c(-c4c(Cl)cccc4Cl)c(=O)ncn3n2)c(F)c1 |(-1.69,6.87,;-1.69,5.33,;-.36,4.56,;-.36,3.02,;-1.69,2.25,;-1.69,.71,;-3.03,-.06,;-3.03,-1.6,;-4.36,-2.37,;-5.75,-1.54,;-7.08,-2.31,;-7.08,-3.85,;-5.75,-4.62,;-4.42,-3.85,;-5.75,-6.16,;-7.08,-6.93,;-8.42,-6.16,;-8.42,-4.62,;-9.75,-3.85,;-8.42,-1.54,;-9.75,-2.31,;-8.42,,;-7.08,.77,;-5.75,,;-4.36,.71,;-3.03,3.02,;-4.36,2.25,;-3.03,4.56,)|
Fc1ccc(cc1)-c1noc(CN2CN(c3ccccc3)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)C2=O)n1
Fc1ccc(cc1)N1CN(CC(=O)NCC(F)(F)F)C(=O)C11CCN(CC1)C(=O)c1cnc2[nH]ncc2c1
Fc1ccc(cc1N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)C(F)(F)F
Fc1ccc2N(CC(=O)N3CC(C3)C(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c2c1Cl
Fc1ccc2N(CC(=O)N3CC(F)(F)C(F)(F)C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c2c1Cl
Fc1ccc2N(CC(=O)N3CC(F)(F)C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c2c1Cl
Fc1ccc2N(CC(=O)N3CC4(CCC4(F)F)C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c2c1Cl
Fc1ccc2N(CC(=O)N3CC4CCCC4C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c2c1Cl
Fc1ccc2N(CC(=O)N3CCC4(COC4)C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c2c1Cl
Fc1ccc2N(CC(=O)N3CCC4CCCC34)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c2c1Cl
Fc1ccc2N(CC(=O)N3CCC4CCCC34)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c2c1Cl |w:12.12,15.15|
Fc1ccc2N(CC(=O)N3CCCC3C#N)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c2c1Cl
Fc1ccc2N(CC(=O)N3CCCC3CC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c2c1Cl
Fc1ccc2N(CC(=O)N3CCC[C@@H]3C(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c2c1Cl |r|
Fc1ccc2N(CC(=O)N3CCC[C@@H]3CC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c2c1Cl |r|
Fc1ccc2N(CC(=O)N3CCC[C@H]3C(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c2c1Cl |r|
Fc1ccc2N(CC(=O)N3CCC[C@H]3C(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c2c1Cl |r|
Fc1ccc2N(CC(=O)N3CCC[C@H]3CC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c2c1Cl |r|
Fc1ccc2N(CC(=O)N3CCN4CCCC4C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c2c1Cl
Fc1ccc2N(CC(=O)N3CCOC(C3)C(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c2c1Cl
Fc1ccc2N(CC(=O)N3CCOC(C3)C(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c2c1Cl |w:13.15|
Fc1ccc2N(CC(=O)N3C[C@@H]4CCC[C@@H]4C3)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c2c1Cl |r|
Fc1ccc2N(CC(=O)NC3(CC3)C#N)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c2c1Cl
Fc1ccc2N(CC(=O)NC3CC3(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c2c1Cl
Fc1ccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3cc4cn[nH]c4cn3)c2c1Cl
Fc1ccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c2c1Br
Fc1ccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c2c1Cl
Fc1ccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4n3)c2c1Cl
Fc1ccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)c2c1
Fc1ccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)c2c1Br
Fc1ccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)c2c1Cl
Fc1ccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)c2c1F
Fc1ccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ncc4[nH]ncc4n3)c2c1Cl
Fc1ccc2N(CCc2c1)C(=O)CN1C(=O)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)c2c1cccc2Br
Fc1ccc2c(c1)N(CC(=O)NCC(F)(F)F)C(=O)C21CCN(CC1)C(=O)c1cnc2[nH]ncc2c1
Fc1cccc(c1)N1CN(CC(=O)NCC(F)(F)F)C(=O)C11CCN(CC1)C(=O)c1cnc2[nH]ncc2c1
Fc1cccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3cnc4[nH]ncc4c3)c12
Fc1ccccc1N1CN(CC(=O)NCC(F)(F)F)C(=O)C11CCN(CC1)C(=O)c1cnc2[nH]ncc2c1
Fc1ccccc1N1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
N#CC[C@H](C1CCCC1)n1cc(cn1)-c1ncnc2[nH]ccc12 |r|
NC(=O)C1CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
NC(=O)c1ccc(cc1)-c1nc(c([nH]1)-c1ccc2OCOc2c1)-c1ccccn1
NC(=O)c1n[nH]c2ccc(cc12)C(=O)N1CCC2(CC1)C(=O)N(CC(=O)NCC(F)(F)F)c1cccc(Cl)c21
NCC1CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O
N[C@@H]1CCCN(Cc2c(Cl)c3[nH]c(=O)n(Cc4cc(Cl)ccc4S(=O)(=O)c4ccccc4)c(=O)c3cc2C(F)(F)F)C1 |r|
Nc1c(cnn1-c1ccccc1)C(=O)NCc1ccc(cc1)C(=O)NCCCC1CCCCC1
Nc1c(cnn1-c1ccccc1)C(=O)NCc1ccc(cc1)C(=O)N[C@@H](CCC1CCCCC1)C(=O)NC1CCCN(C1)C(=O)C1CC1 |r|
Nc1c(cnn1-c1ccccc1)C(=O)NCc1ccc(cc1)C(=O)N[C@@H](CCC1CCCCC1)C(=O)NC1CCCN(C1)C1COC1 |r|
Nc1n[nH]c2cc(ccc12)C(=O)N1CC2(C1)C(=O)N(CC(=O)NCC(F)(F)F)c1cccc(Br)c21
Nc1n[nH]c2cc(ccc12)C(=O)N1CCC2(CC1)C(=O)N(CC(=O)NCC(F)(F)F)c1ccc(F)c(Cl)c21
Nc1n[nH]c2cc(ccc12)C(=O)N1CCC2(CC1)N(CN(CC(=O)NCC(F)(F)F)C2=O)c1ccccc1
Nc1n[nH]c2ccc(cc12)C(=O)N1CCC2(CC1)N(CN(CC(=O)NCC(F)(F)F)C2=O)c1ccccc1
Nc1nc(-c2cccc(c2CO)-n2ccc3cc(cc(F)c3c2=O)C2CC2)c2cc([nH]c2n1)C1=CCN(CC1)C1COC1 |t:39|
Nc1nc(N)c2nc(-c3cccc(O)c3)c(nc2n1)-c1cccc(O)c1
Nc1nc(Nc2ccc(cc2)S(N)(=O)=O)nn1C(=O)c1c(F)cccc1F
Nc1nc(Nc2ccc3CC[C@@H](CCc3c2)N2CCCC2)nn1-c1cc2CCCc3ccccc3-c2nn1 |r|
Nc1ncc(cn1)C(=O)N1CCC2(CC1)N(CN(CC(=O)NCC(F)(F)F)C2=O)c1ccccc1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)N1CCC(C1)C#N
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)N1CCC(C1)n1cncn1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)N1CCOCC1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)N1C[C@@H]2CN(Cc3ccccc3)C[C@@H]2C1 |r|
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)NCCN1CCOCC1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)N[C@@H]1CNC[C@H]1c1ccccc1 |r|
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)N[C@H]1CNC[C@@H]1c1ccccc1 |r|
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)N[C@H]1C[C@@H]1c1ccccc1 |r|
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)Nc1cccc(c1)N1CCOCC1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)Nc1ccccc1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)Nc1ccccn1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)Nc1cccnc1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O)Nc1ccncc1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]nnc3c2)C1=O)N1CCOCC1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3cn[nH]c3c2)C1=O)Nc1ccccc1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)N1CCC(C1)C#N
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)N1CCC(C1)N1CCCC1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)N1CCCC1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)N1CCCC11COC1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)N1CCN(C2CC2)C(=O)C1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)N1CCN(CC1)C1CC1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)N1CCOCC1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)N1CCS(=O)(=O)CC1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)N1C[C@@H]2CN(Cc3ccccc3)C[C@@H]2C1 |r|
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)NC12CC3CC(CC(C3)C1)C2 |TLB:35:36:33.34.39:40,39:34:41:38.40.37,39:38:33.34.35:41,THB:35:34:40:36.41.37|
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)NC1COC1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)N[C@H]1C[C@@H]1c1cccc(CN2CCOCC2)c1 |r|
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)Nc1cccc(n1)C#N
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)Nc1ccccc1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)Nc1ccccc1CN1CCOCC1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)Nc1ccccn1
O=C(CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O)Nc1ncc(s1)C#N
O=C(N1CCC2(CC1)N(CN(C1CCN(C1=O)c1ccccc1)C2=O)c1ccccc1)c1cnc2[nH]ncc2c1
O=C(N1CCC2(CC1)N(CN(C1CCN(C3CC3)C1=O)C2=O)c1ccccc1)c1cnc2[nH]ncc2c1
O=C(N1CCC2(CC1)N(CN(C2=O)c1ccc(cc1)C#N)c1ccccc1)c1cnc2[nH]ncc2c1
O=C(N1CCC2(CC1)N(CN(C2=O)c1ccccc1)c1ccccc1)c1ccc2[nH]ncc2c1
O=C(N1CCC2(CC1)N(CN(Cc1cccc(n1)C#N)C2=O)c1ccccc1)c1cnc2[nH]ncc2c1
O=C(N1CCC2(CC1)N(CN(Cc1nc(no1)C1CC1)C2=O)c1ccccc1)c1ccc2[nH]ncc2c1
O=C(N1CCC2(CC1)N(CN(Cc1nnc(s1)C1CC1)C2=O)c1ccccc1)c1ccc2[nH]ncc2c1
O=C(N1CCNCC1)c1ccc(\C=C\c2n[nH]c3ccccc23)cc1
O=C(NCc1cccc(NC(=O)c2cnc3ccccn23)c1)Nc1ccccc1
O=C(\C=C1/Nc2cc(ccc2NC1=O)C#N)c1cccc2ccccc12
O=C(\C=C1/Nc2ccccc2NC1=O)c1cccc2ccccc12
OC(=O)c1ccc(Nc2ncc3CN=C(c4cc(Cl)ccc4-c3n2)c2c(F)cccc2F)cc1 |c:13|
OC(=O)c1n[nH]c2ccc(cc12)C(=O)N1CCC2(CC1)C(=O)N(CC(=O)NCC(F)(F)F)c1ccc(F)c(Cl)c21
OCCN(CC(F)(F)F)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2ccc3[nH]ncc3c2)C1=O
OCCn1cc(c(n1)-c1ccncc1)-c1ccc2C(CCc2c1)N=O
OCc1cccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
O[C@@H]1CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
O[C@H]1CCN(C1)C(=O)CN1CN(c2ccccc2)C2(CCN(CC2)C(=O)c2cnc3[nH]ncc3c2)C1=O |r|
Oc1ccc(cc1)-c1nc(c([nH]1)-c1ccc(F)cc1)-c1ccncc1
Oc1cccc(Nc2ccnc3cc(sc23)-c2cccc(CN3CCOCC3)c2)c1
Oc1cccc(c1)-c1nc(N2CCOCC2)c2oc3ncccc3c2n1
Oc1cccc2N(CC(=O)NCC(F)(F)F)C(=O)C3(CCN(CC3)C(=O)c3ccc4[nH]ncc4c3)c12
[H][C@@]12CCCN1CCN(Cc1c(Cl)c3[nH]c(=O)n(Cc4cc(Cl)ccc4S(=O)(=O)CC)c(=O)c3cc1C(F)(F)F)C2 |r|
[H][C@@]12C[C@@H]([C@H](OC)[C@@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13)N(C)C(=O)c1ccccc1 |TLB:11:10:9:4.3.2,17:33:9:4.3.2,THB:24:32:9:4.3.2,5:4:9:10.31.33.32,30:31:9:4.3.2|
[H][C@@]12C[C@@]3(CC(=O)c4cc(O)ccc4O)C(=O)O[C@@H](OC)[C@@]3(C)[C@]1([H])OC=C(C=O)[C@H]2C\C=C(/CC(=O)c1cc(O)ccc1O)C(O)=O |r,t:29|
[H][C@]12CCCN1CCN(Cc1c(Cl)c3[nH]c(=O)n(Cc4cc(Cl)ccc4S(=O)(=O)CC)c(=O)c3cc1C(F)(F)F)C2 |r|
[H][C@]12C[C@@H](NCCOCCOCCOCCNC(=O)CCC3=[N+]4C(C=C3)=Cc3c(C)cc(C)n3[B-]4(F)F)[C@@H](OC)[C@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13 |r,c:24,26,t:21|
[H][C@]12C[C@H]([C@@H](OC)[C@](C)(O1)n1c3ccccc3c3c4CNC(=O)c4c4c5ccccc5n2c4c13)N(C)CCOCCOCCOCCNC(=O)CCC1=[N+]2C(C=C1)=Cc1c(C)cc(C)n1[B-]2(F)F |r,c:63,65,t:60|
[H][C@]12C[C@]3(CC(=O)c4cc(O)ccc4O)C(=O)O[C@H](OC)[C@]3(C)[C@@]1([H])OC=C(C=O)[C@@H]2C\C=C(/CC(=O)c1cc(O)ccc1O)C(O)=O |r,t:29|