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Found 1487 with Last Name = 'bian' and Initial = 'a'
TargetMu-type opioid receptor(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50474150(CHEMBL58362)
Affinity DataKi:  0.0100nMAssay Description:Binding affinity to mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50472720(CHEMBL41721)
Affinity DataKi:  0.220nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196014(3-(2-(trifluoromethyl)benzyl)-N-cyclopentyl-5-phen...)
Affinity DataKi:  0.600nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataKi:  0.650nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106372(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  0.710nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50472720(CHEMBL41721)
Affinity DataKi:  0.720nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50072775(2-((1R,2R,5R)-5-hydroxy-2-(3-hydroxypropyl)cyclohe...)
Affinity DataKi:  0.980nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196002(3-(2-fluorobenzyl)-N-cyclohexyl-5-phenyl-3H-[1,2,3...)
Affinity DataKi:  1.15nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106373(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  1.40nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196009(3-benzyl-N-cyclohexyl-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  1.90nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106374(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  2.10nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276769(CHEMBL514399 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  2.20nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106376(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  2.30nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276770(CHEMBL456211 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  2.5nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50284000((2-Methyl-1-pentyl-1H-indol-3-yl)-naphthalen-1-yl-...)
Affinity DataKi:  3nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptidyl-prolyl cis-trans isomerase FKBP5(Homo sapiens (Human))
Max Institute Of Psychiatry

Curated by ChEMBL
LigandPNGBDBM36609(Rapamycin C-7, analog 4 | SIROLIMUS | US11603377, ...)
Affinity DataKi:  3nMAssay Description:Binding affinity to human FKBP51 by competitive fluorescence polarization assayMore data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50474150(CHEMBL58362)
Affinity DataKi:  3nMAssay Description:Binding affinity to delta opioid receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195990(3-(2-fluorobenzyl)-5-phenyl-N-propyl-3H-[1,2,3]tri...)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Temple University

Curated by ChEMBL
LigandPNGBDBM50000092((-)-(etorphine) | (-)-morphine | (1S,5R,13R,14S)-1...)
Affinity DataKi:  3.5nMAssay Description:Displacement of [3H]DAMGO from mu opoid receptor in Dunkin-Hartley guinea pig brain after 1.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM21281((11R)-2-methyl-11-(morpholin-4-ylmethyl)-3-(naphth...)
Affinity DataKi:  3.5nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195996(3-(3-(2-fluorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  3.70nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM106370(9-(ortho-fluorobenzyl)-2-phenyl-azaadenine (1bis))
Affinity DataKi:  3.80nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196018(3-(2-fluorobenzyl)-N-butyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195995(1-(3-(2-fluorobenzyl)-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  4.80nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195992(3-benzyl-N-cyclobutyl-5-phenyl-3H-[1,2,3]triazolo[...)
Affinity DataKi:  5nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106375(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  5.5nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106378(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  5.5nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276243(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyrimid...)
Affinity DataKi:  5.60nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50060617((5Z,8Z,11Z,14Z)-2-Methyl-icosa-5,8,11,14-tetraenoi...)
Affinity DataKi:  5.80nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196015(3-(2-(trifluoromethyl)benzyl)-N-butyl-5-phenyl-3H-...)
Affinity DataKi:  6.5nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196003(3-(2-fluorobenzyl)-N-cyclopentyl-5-phenyl-3H-[1,2,...)
Affinity DataKi:  6.70nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196030(3-(2-(trifluoromethyl)benzyl)-N-cyclohexyl-5-pheny...)
Affinity DataKi:  6.80nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50492099(CHEMBL2396991)
Affinity DataKi:  7nMAssay Description:Binding affinity to mu opioid receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Temple University

Curated by ChEMBL
LigandPNGBDBM50492099(CHEMBL2396991)
Affinity DataKi:  7nMAssay Description:Binding affinity to kappa opioid receptor (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276242(4-amino-N-(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,...)
Affinity DataKi:  7.10nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Temple University

Curated by ChEMBL
LigandPNGBDBM50474152(CHEBI:6956 | CHEMBL299031)
Affinity DataKi:  7.20nMAssay Description:Displacement of [3H]DAMGO from mu opoid receptor in Dunkin-Hartley guinea pig brain after 1.5 hrs by liquid scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195999(1-(3-benzyl-5-phenyl-3H-[1,2,3]triazolo[4,5-d]pyri...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276707(CHEMBL458346 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  7.5nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196020(3-(2-(trifluoromethyl)benzyl)-N-cyclopropyl-5-phen...)
Affinity DataKi:  7.80nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276772(CHEMBL456011 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  8nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50072757((5Z,8Z,11Z,14Z)-Icosa-5,8,11,14-tetraenoic acid (2...)
Affinity DataKi:  8.5nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50472724(5''-F-delta8-THC | CHEMBL75330)
Affinity DataKi:  8.70nMAssay Description:Binding affinity towards cloned human cannabinoid receptor 2More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196011(3-(2-chlorobenzyl)-N-cyclopentyl-5-phenyl-3H-[1,2,...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

LigandPNGBDBM106371(N-[9-(ortho-fluorobenzyl)-2-phenyl-9H-8-azapurin-6...)
Affinity DataKi:  9.20nMpH: 7.4Assay Description:For A1 adenosine receptors, 40 mg of protein were incubated for 60 min at 25°C with [3H]DPCPX 0.5 nM (Kd = 0.4 nM) and increasing concentrations...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50284000((2-Methyl-1-pentyl-1H-indol-3-yl)-naphthalen-1-yl-...)
Affinity DataKi:  9.5nMAssay Description:Binding affinity towards cloned human Cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(GUINEA PIG)
Temple University

Curated by ChEMBL
LigandPNGBDBM50474153(CHEMBL61630)
Affinity DataKi:  9.80nMAssay Description:Displacement of [3H]DAMGO from guinea pig brain mu opoid receptor after 3 hrs by liquid scintillation counting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Università

Curated by ChEMBL
LigandPNGBDBM50276867(CHEMBL459772 | N-(3-benzyl-5-phenyl-3H-[1,2,3]tria...)
Affinity DataKi:  10nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in Wistar rat brain cortex by liquid scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50195997(3-(2-chlorobenzyl)-N-cyclopropyl-5-phenyl-3H-[1,2,...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Università

Curated by ChEMBL
LigandPNGBDBM50196022(3-benzyl-N-cyclopentyl-5-phenyl-3H-[1,2,3]triazolo...)
Affinity DataKi:  11nMAssay Description:Displacement of [3H]DPCPX from bovine cerbral cortex adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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