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Found 48 with Last Name = 'drakopoulos' and Initial = 'a'
TargetKappa-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511258(CHEMBL4438046)
Affinity DataKi:  1.10nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human KOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511255(CHEMBL4463414)
Affinity DataKi:  1.40nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human KOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511257(CHEMBL4577693)
Affinity DataKi:  1.80nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human KOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511256(CHEMBL4514226)
Affinity DataKi:  3.20nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human KOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511259(CHEMBL4459592)
Affinity DataKi:  8.60nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human KOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511259(CHEMBL4459592)
Affinity DataKi:  31nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human DOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511255(CHEMBL4463414)
Affinity DataKi:  39nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human DOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511255(CHEMBL4463414)
Affinity DataKi:  40nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human MOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511258(CHEMBL4438046)
Affinity DataKi:  100nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human MOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511258(CHEMBL4438046)
Affinity DataKi:  106nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human DOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511256(CHEMBL4514226)
Affinity DataKi:  110nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human MOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511257(CHEMBL4577693)
Affinity DataKi:  133nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human MOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511257(CHEMBL4577693)
Affinity DataKi:  193nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human DOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511256(CHEMBL4514226)
Affinity DataKi:  280nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human DOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511259(CHEMBL4459592)
Affinity DataKi:  380nMAssay Description:Displacement of [3H]-diprenorphine from recombinant human MOR transiently expressed in HEK293 cell membranes measured after 60 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465108(CHEMBL4277543)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes assessed as blockade of inward currents at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50033369(AMANTADINE | CHEMBL660 | SYMADINE | SYMMETREL)
Affinity DataIC50:  4.70E+3nMAssay Description:Inhibition of Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes assessed as blockade of inward currents at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465108(CHEMBL4277543)
Affinity DataIC50:  9.30E+3nMAssay Description:Inhibition of Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes assessed as blockade of inward currents at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50216627((alpha-methyl-1-adamantyl)methylamine | 1-Adamanta...)
Affinity DataIC50:  1.08E+4nMAssay Description:Inhibition of Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes assessed as blockade of inward currents at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50033369(AMANTADINE | CHEMBL660 | SYMADINE | SYMMETREL)
Affinity DataIC50:  1.25E+4nMAssay Description:Inhibition of Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes assessed as blockade of inward currents at...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465104(CHEMBL4284791)
Affinity DataIC50:  1.32E+4nMAssay Description:Inhibition of Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes assessed as blockade of inward currents at...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465104(CHEMBL4284791)
Affinity DataIC50:  2.43E+4nMAssay Description:Inhibition of Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes assessed as blockade of inward currents at...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)TBA
LigandPNGBDBM50465106(CHEMBL3392935)
Affinity DataKd:  340nMAssay Description:Binding affinity to C-terminal amidated influenza A virus A/Udorn/72 (H3N2) M2 transmembrane domain (22 to 46 residues) in DPC micelles at pH 8 asses...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)TBA
LigandPNGBDBM50465105(CHEMBL1235691)
Affinity DataKd:  320nMAssay Description:Binding affinity to C-terminal amidated influenza A virus A/Udorn/72 (H3N2) M2 transmembrane domain (22 to 46 residues) in DPC micelles at pH 8 asses...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)TBA
LigandPNGBDBM50216627((alpha-methyl-1-adamantyl)methylamine | 1-Adamanta...)
Affinity DataKd:  510nMAssay Description:Binding affinity to C-terminal amidated influenza A virus A/Udorn/72 (H3N2) M2 transmembrane domain (22 to 46 residues) in DPC micelles at pH 8 asses...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)TBA
LigandPNGBDBM50465108(CHEMBL4277543)
Affinity DataKd:  130nMAssay Description:Binding affinity to C-terminal amidated influenza A virus A/Udorn/72 (H3N2) M2 transmembrane domain (22 to 46 residues) in DPC micelles at pH 8 asses...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511259(CHEMBL4459592)
Affinity DataKd:  19nMAssay Description:Binding affinity to recombinant human KOR transiently expressed in CHOK1 cells measured after 20 mins by TIRF microscopic analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511255(CHEMBL4463414)
Affinity DataKd:  9.5nMAssay Description:Binding affinity to recombinant human KOR transiently expressed in CHOK1 cells measured after 20 mins by TIRF microscopic analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
Julius Maximilian University of W£Rzburg

Curated by ChEMBL
LigandPNGBDBM50511257(CHEMBL4577693)
Affinity DataKd:  4.80nMAssay Description:Binding affinity to recombinant human KOR transiently expressed in CHOK1 cells measured after 20 mins by TIRF microscopic analysisMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465105(CHEMBL1235691)
Affinity DataKd:  3.20E+3nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465104(CHEMBL4284791)
Affinity DataKd:  4.59E+3nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel by isothermal calorimetric titrationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465108(CHEMBL4277543)
Affinity DataKd:  1.30E+4nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465107(CHEMBL4292664)
Affinity DataKd:  3.43E+3nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel by isothermal calorimetric titrationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465107(CHEMBL4292664)
Affinity DataKd:  8.80E+4nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage c...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50033369(AMANTADINE | CHEMBL660 | SYMADINE | SYMMETREL)
Affinity DataKd:  2.10E+5nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 M2 proton channel S31N mutant expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50216627((alpha-methyl-1-adamantyl)methylamine | 1-Adamanta...)
Affinity DataKd:  510nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel by isothermal calorimetric titrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465107(CHEMBL4292664)
Affinity DataKd: >1.00E+4nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 M2 proton channel S31N mutant by isothermal calorimetric titrationMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50033369(AMANTADINE | CHEMBL660 | SYMADINE | SYMMETREL)
Affinity DataKd:  9.00E+3nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50216627((alpha-methyl-1-adamantyl)methylamine | 1-Adamanta...)
Affinity DataKd:  7.00E+3nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50216627((alpha-methyl-1-adamantyl)methylamine | 1-Adamanta...)
Affinity DataKd: >1.00E+7nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 M2 proton channel S31N mutant expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465108(CHEMBL4277543)
Affinity DataKd:  4.44E+5nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 M2 proton channel S31N mutant expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50033369(AMANTADINE | CHEMBL660 | SYMADINE | SYMMETREL)
Affinity DataKd:  2.17E+3nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel by isothermal calorimetric titrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465106(CHEMBL3392935)
Affinity DataKd:  340nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel by isothermal calorimetric titrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465108(CHEMBL4277543)
Affinity DataKd:  130nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel by isothermal calorimetric titrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465107(CHEMBL4292664)
Affinity DataKd:  1.80E+6nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 M2 proton channel S31N mutant expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (strain A/Puerto Rico/8/1934 H1N...)TBA
LigandPNGBDBM50033369(AMANTADINE | CHEMBL660 | SYMADINE | SYMMETREL)
Affinity DataKd:  2.17E+3nMAssay Description:Binding affinity to C-terminal amidated influenza A virus A/Udorn/72 (H3N2) M2 transmembrane domain (22 to 46 residues) in DPC micelles at pH 8 asses...More data for this Ligand-Target Pair
In DepthDetails PubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465105(CHEMBL1235691)
Affinity DataKd:  320nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel by isothermal calorimetric titrationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMatrix protein 2(Influenza A virus (A/Udorn/307/1972(H3N2)))
National and Kapodistrian University of Athens

Curated by ChEMBL
LigandPNGBDBM50465106(CHEMBL3392935)
Affinity DataKd:  3.90E+3nMAssay Description:Binding affinity to Influenza A virus A/Udorn/72 wild-type M2 proton channel expressed in Xenopus laevis oocytes at pH 5.5 by two-electrode voltage c...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed