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Found 203 with Last Name = 'emer' and Initial = 'e'
LigandPNGBDBM50117636(CHEMBL3613642)
Affinity DataIC50:  57nMAssay Description:Antagonist activity at mouse TRPV4 receptor expressed in HEK293 cells assessed as inhibition of 4alpha-PDD-stimulated calcium flux after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Renovis

Curated by ChEMBL
LigandPNGBDBM50311785(CHEMBL1079421 | Phenmedipham)
Affinity DataIC50:  77nMAssay Description:Inhibition of rat FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117636(CHEMBL3613642)
Affinity DataIC50:  120nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of 4alpha-PDD-stimulated calcium flux after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Renovis

Curated by ChEMBL
LigandPNGBDBM50311785(CHEMBL1079421 | Phenmedipham)
Affinity DataIC50:  152nMAssay Description:Inhibition of human FAAH-mediated hydrolysis of [3H]AEAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117640(CHEMBL3613639)
Affinity DataIC50:  260nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117636(CHEMBL3613642)
Affinity DataIC50:  320nMAssay Description:Antagonist activity at mouse TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117639(CHEMBL3613640)
Affinity DataIC50:  370nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Renovis

Curated by ChEMBL
LigandPNGBDBM50311785(CHEMBL1079421 | Phenmedipham)
Affinity DataIC50:  377nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117639(CHEMBL3613640)
Affinity DataIC50:  380nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117646(CHEMBL3613628)
Affinity DataIC50:  390nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117640(CHEMBL3613639)
Affinity DataIC50:  390nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117636(CHEMBL3613642)
Affinity DataIC50:  420nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Renovis

Curated by ChEMBL
LigandPNGBDBM50311786(Amperozide | CHEMBL1079935)
Affinity DataIC50:  455nMAssay Description:Inhibition of human FAAH-mediated hydrolysis of [3H]AEAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117638(CHEMBL3613641)
Affinity DataIC50:  490nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117638(CHEMBL3613641)
Affinity DataIC50:  540nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117636(CHEMBL3613642)
Affinity DataIC50:  570nMAssay Description:Antagonist activity at human TRPV4 expressed in HEK293 cells assessed as inhibition of 20% hypotonic solution-induced Ca2+ influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase Su(var)3-9(Drosophila melanogaster)
Ludwig-Maximillians University Of Munich

Curated by ChEMBL
LigandPNGBDBM50315537(CHEMBL1089316 | chaetocin)
Affinity DataIC50:  600nMAssay Description:Inhibition of Drosophila melanogaster SU(VAR)3-9More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117636(CHEMBL3613642)
Affinity DataIC50:  660nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117645(CHEMBL3613629)
Affinity DataIC50:  710nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117650(CHEMBL3613638)
Affinity DataIC50:  800nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117652(CHEMBL3613636)
Affinity DataIC50:  910nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117647(CHEMBL3613627)
Affinity DataIC50:  930nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117637(CHEMBL3613643)
Affinity DataIC50:  930nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117645(CHEMBL3613629)
Affinity DataIC50:  940nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117646(CHEMBL3613628)
Affinity DataIC50:  1.05E+3nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117651(CHEMBL3613637)
Affinity DataIC50:  1.28E+3nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117654(CHEMBL3613634)
Affinity DataIC50:  1.32E+3nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1(Homo sapiens (Human))
Renovis

Curated by ChEMBL
LigandPNGBDBM50311786(Amperozide | CHEMBL1079935)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition of human FAAHMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117644(CHEMBL3613630)
Affinity DataIC50:  1.94E+3nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117636(CHEMBL3613642)
Affinity DataIC50:  2.10E+3nMAssay Description:Antagonist activity at rat TRPV4 expressed in HEK293 cells assessed as inhibition of 20% hypotonic solution-induced Ca2+ influxMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117653(CHEMBL3613635)
Affinity DataIC50:  2.11E+3nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117644(CHEMBL3613630)
Affinity DataIC50:  2.17E+3nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase EHMT2(Mus musculus)
Ludwig-Maximillians University Of Munich

Curated by ChEMBL
LigandPNGBDBM50315537(CHEMBL1089316 | chaetocin)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of mouse G9aMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305208(3-Methyl-4-phenylbut-3-en-2-one oxime | CHEMBL6037...)
Affinity DataIC50:  2.70E+3nMAssay Description:Antagonist activity at human TRPA1 expressed in HEK293 cells assessed as [45]Ca2+ influx by microbeta plate countMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50305207(4-(4-chlorophenyl)-3-methylbut-3-en-2-one oxime | ...)
Affinity DataIC50:  2.80E+3nMAssay Description:Antagonist activity at human TRPA1 expressed in HEK293 cells assessed as [45]Ca2+ influx by microbeta plate countMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117637(CHEMBL3613643)
Affinity DataIC50:  2.92E+3nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone-lysine N-methyltransferase, H3 lysine-9 specific dim-5(Neurospora crassa)
Ludwig-Maximillians University Of Munich

Curated by ChEMBL
LigandPNGBDBM50315537(CHEMBL1089316 | chaetocin)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of Neurospora crassa DIM5More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117647(CHEMBL3613627)
Affinity DataIC50:  3.90E+3nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50519637(CHEMBL4550375)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of monoamino oxidase B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50117641(CHEMBL3613633)
Affinity DataIC50:  4.22E+3nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117649(CHEMBL3613625)
Affinity DataIC50:  4.30E+3nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117648(CHEMBL3613626)
Affinity DataIC50:  4.93E+3nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50519636(BMN 195 | BMN-195 | Ezutromid | SMT-C1100 | SMTC-1...)
Affinity DataIC50:  5.40E+3nMAssay Description:Inhibition of CYP1A2 in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117641(CHEMBL3613633)
Affinity DataIC50:  5.74E+3nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117648(CHEMBL3613626)
Affinity DataIC50:  6.49E+3nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117649(CHEMBL3613625)
Affinity DataIC50:  8.53E+3nMAssay Description:Antagonist activity at human TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 m...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMultidrug and toxin extrusion protein 1(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50519637(CHEMBL4550375)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibition of MATE1 (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
LigandPNGBDBM50117636(CHEMBL3613642)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human TRPV1 receptor expressed in HEK293 cells assessed as inhibition of capsaicin-stimulated calcium flux after 10 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117642(CHEMBL3613632)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50117643(CHEMBL3613631)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat TRPV4 receptor expressed in HEK293 cells assessed as inhibition of EC80 of 4alpha-PDD-stimulated calcium flux after 10 min...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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