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Found 30 with Last Name = 'celik' and Initial = 'f'
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246510(1-(4-(1,3,7,7-Tetramethyl-5-oxo-1,2,3,4,5,6,7,8-oc...)
Affinity DataIC50:  6.31E+4nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246507(1-(4-Fluorophenyl)-3-(4-(1,3,7,7-tetramethyl-5-oxo...)
Affinity DataIC50:  6.62E+4nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246508(1-Phenyl-3-(4-(1,3,7,7-tetramethyl-5-oxo-1,2,3,4,5...)
Affinity DataIC50:  8.89E+4nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246513(1-(3-Fluorophenyl)-3-(4-(1,3,7,7-tetramethyl-5-oxo...)
Affinity DataIC50:  8.92E+4nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246510(1-(4-(1,3,7,7-Tetramethyl-5-oxo-1,2,3,4,5,6,7,8-oc...)
Affinity DataIC50:  1.06E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246513(1-(3-Fluorophenyl)-3-(4-(1,3,7,7-tetramethyl-5-oxo...)
Affinity DataIC50:  1.30E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246512(1-(2,4-Dichlorophenyl)-3-(4-(1,3,7,7-tetramethyl-5...)
Affinity DataIC50:  1.32E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246505(1-Phenyl-3-(4-(1,3,7,7-tetramethyl-5-oxo-1,2,3,4,5...)
Affinity DataIC50:  1.35E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246508(1-Phenyl-3-(4-(1,3,7,7-tetramethyl-5-oxo-1,2,3,4,5...)
Affinity DataIC50:  1.36E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246507(1-(4-Fluorophenyl)-3-(4-(1,3,7,7-tetramethyl-5-oxo...)
Affinity DataIC50:  1.42E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246512(1-(2,4-Dichlorophenyl)-3-(4-(1,3,7,7-tetramethyl-5...)
Affinity DataIC50:  1.51E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246505(1-Phenyl-3-(4-(1,3,7,7-tetramethyl-5-oxo-1,2,3,4,5...)
Affinity DataIC50:  1.53E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246506(1-(4-Methoxyphenyl)-3-(4-(1,3,7,7-tetramethyl-5-ox...)
Affinity DataIC50:  1.53E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246509(1-(4-Nitrophenyl)-3-(4-(1,3,7,7-tetramethyl-5-oxo-...)
Affinity DataIC50:  1.55E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246506(1-(4-Methoxyphenyl)-3-(4-(1,3,7,7-tetramethyl-5-ox...)
Affinity DataIC50:  1.57E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246511(1-(3-Methoxyphenyl)-3-(4-(1,3,7,7-tetramethyl-5-ox...)
Affinity DataIC50:  1.64E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 2(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246511(1-(3-Methoxyphenyl)-3-(4-(1,3,7,7-tetramethyl-5-ox...)
Affinity DataIC50:  1.70E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCarbonic anhydrase 1(Homo sapiens (Human))
Sakarya University

LigandPNGBDBM246509(1-(4-Nitrophenyl)-3-(4-(1,3,7,7-tetramethyl-5-oxo-...)
Affinity DataIC50:  1.98E+5nMAssay Description:For the inhibition studies of sulphanilamide, different concentrationsof these compounds were added to the enzyme. Activity percentage values of CA f...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group E member 1(Homo sapiens)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50584388(CHEMBL5089826)
Affinity DataEC50:  1.20E+3nMAssay Description:Agonist activity at human Gal4-fused TLX LBD expressed in human HEK293T cells coexpressing Gal4-VP16 assessed as repressor activity of receptor by me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group E member 1(Homo sapiens)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50584389(CHEMBL5080383)
Affinity DataEC50:  251nMAssay Description:Agonist activity at human Gal4-fused TLX LBD expressed in human HEK293T cells coexpressing Gal4-VP16 assessed as repressor activity of receptor by me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group E member 1(Homo sapiens)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50584383(CHEMBL5080162 | EN300-5601139)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity at human Gal4-fused TLX LBD expressed in human HEK293T cells coexpressing Gal4-VP16 assessed as repressor activity of receptor by me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group E member 1(Homo sapiens)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50584389(CHEMBL5080383)
Affinity DataEC50:  250nMAssay Description:Agonist activity at human Gal4-fused TLX LBD expressed in human HEK293T cells coexpressing Gal4-VP16 assessed as repressor activity of receptor by me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group E member 1(Homo sapiens)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50584389(CHEMBL5080383)
Affinity DataEC50:  700nMAssay Description:Agonist activity at human full length Gal4-fused TLX transfected in human HEK293T cells coexpressing pFR-TAE-Luc assessed as repressor activity of re...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group E member 1(Homo sapiens)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50584389(CHEMBL5080383)
Affinity DataKd:  1.60E+3nMAssay Description:Binding affinity to recombinant TLX LBD (unknown origin) by differential scanning fluorometryMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group E member 1(Homo sapiens)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50584387(CHEMBL5088898)
Affinity DataEC50:  3.00E+3nMAssay Description:Agonist activity at human Gal4-fused TLX LBD expressed in human HEK293T cells coexpressing Gal4-VP16 assessed as repressor activity of receptor by me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group E member 1(Homo sapiens)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50584385(CHEMBL5077720)
Affinity DataEC50:  1.10E+4nMAssay Description:Agonist activity at human Gal4-fused TLX LBD expressed in human HEK293T cells coexpressing Gal4-VP16 assessed as repressor activity of receptor by me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group E member 1(Homo sapiens)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50584384(CHEMBL5090226 | US20240067625, Compound 30)
Affinity DataEC50:  1.00E+3nMAssay Description:Agonist activity at human Gal4-fused TLX LBD expressed in human HEK293T cells coexpressing Gal4-VP16 assessed as repressor activity of receptor by me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group E member 1(Homo sapiens)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50584383(CHEMBL5080162 | EN300-5601139)
Affinity DataEC50:  2.00E+4nMAssay Description:Agonist activity at human Gal4-fused TLX LBD expressed in human HEK293T cells coexpressing Gal4-VP16 assessed as repressor activity of receptor by me...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group E member 1(Homo sapiens)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50584389(CHEMBL5080383)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonist activity at TLX (unknown origin) assessed as induction of receptor oligomerization using sGFP-labeled TLX LBD as acceptor and biotin TLX LBD ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNuclear receptor subfamily 2 group E member 1(Homo sapiens)
Goethe University Frankfurt

Curated by ChEMBL
LigandPNGBDBM50584386(CHEMBL5071695)
Affinity DataEC50:  5.00E+3nMAssay Description:Agonist activity at human Gal4-fused TLX LBD expressed in human HEK293T cells coexpressing Gal4-VP16 assessed as repressor activity of receptor by me...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed