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Found 292 with Last Name = 'falchi' and Initial = 'f'
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM13530(4-[(4-methylpiperazin-1-yl)methyl]-N-[4-methyl-3-[...)
Affinity DataKi:  13nMMore data for this Ligand-Target Pair
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50262718(CHEMBL476304 | N-(5-(4-methoxybenzyl)thiazol-2-yl)...)
Affinity DataKi:  16nMAssay Description:Inhibition of Abl kinase (unknown origin) by cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50224371(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-6-(e...)
Affinity DataKi:  40nMAssay Description:Inhibition of human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50230100(4-fluoro-N-(5-(4-fluorobenzylthio)-1,3,4-thiadiazo...)
Affinity DataKi:  44nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86859(CAS_1327207 | N-(5-(4-bromobenzylthio)-1,3,4-thiad...)
Affinity DataKi:  47nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50262723(CHEMBL517822 | N-(5-(2,5-dichlorobenzyl)thiazol-2-...)
Affinity DataKi:  50nMAssay Description:Inhibition of Abl kinase (unknown origin) by cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50262722(CHEMBL517047 | Thiophene-2-carboxylic acid [5-(3-m...)
Affinity DataKi:  59nMAssay Description:Inhibition of Abl kinase (unknown origin) by cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50224388(CHEMBL238561 | N-(3-bromophenyl)-1-(2-chloro-2-phe...)
Affinity DataKi:  60nMAssay Description:Inhibition of human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86863(CAS_4390766 | N-(5-(3-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  64nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50262667(CHEMBL477139 | N-(6-methoxy-8H-indeno[1,2-d]thiazo...)
Affinity DataKi:  68nMAssay Description:Inhibition of Abl kinase (unknown origin) by cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86875(CAS_685639 | N-(5-(benzylthio)-1,3,4-thiadiazol-2-...)
Affinity DataKi:  70nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50089575(CHEMBL3578214)
Affinity DataKi:  70nMAssay Description:Inhibition of human recombinant full-length Fyn using Src substrate peptide after 15 mins incubation by MicroBeta liquid scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86874(CAS_44454498 | N-(5-(3-chlorobenzylthio)-1,3,4-thi...)
Affinity DataKi:  73nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50224377(1-(2-chloro-2-phenylethyl)-N-(2-fluorobenzyl)-6-(m...)
Affinity DataKi:  80nMAssay Description:Inhibition of human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86857(CAS_44454939 | N-(5-(4-nitrobenzylthio)-1,3,4-thia...)
Affinity DataKi:  83nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86868(CAS_3643794 | N-(5-(4-bromobenzylthio)-1,3,4-thiad...)
Affinity DataKi:  89nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50224387(1-(2-chloro-2-phenylethyl)-N-(2-chlorobenzyl)-6-(m...)
Affinity DataKi:  90nMAssay Description:Inhibition of human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50343427(CHEMBL1775039 | N-Benzyl-1-(2-chloro-2-phenylethyl...)
Affinity DataKi:  90nMAssay Description:Inhibition of AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50262664(CHEMBL504598 | N-(5-benzylthiazol-2-yl)thiophene-2...)
Affinity DataKi:  90nMAssay Description:Inhibition of Abl kinase (unknown origin) by cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86856(CAS_44454904 | N-(5-(4-nitrobenzylthio)-1,3,4-thia...)
Affinity DataKi:  92nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Fyn(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50089569(CHEMBL3578215)
Affinity DataKi:  95nMAssay Description:Inhibition of human recombinant full-length Fyn using Src substrate peptide after 15 mins incubation by MicroBeta liquid scintillation counting analy...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50262715(CHEMBL518430 | N-(5-(3-chlorobenzyl)thiazol-2-yl)t...)
Affinity DataKi:  97nMAssay Description:Inhibition of Abl kinase (unknown origin) by cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50224372(1-(2-chloro-2-phenylethyl)-N-(4-fluorobenzyl)-6-(m...)
Affinity DataKi:  100nMAssay Description:Inhibition of human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86860(CAS_3320545 | N-(5-(4-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  104nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50224383(1-(2-chloro-2-(4-chlorophenyl)ethyl)-6-(methylthio...)
Affinity DataKi:  110nMAssay Description:Inhibition of human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50224374(CHEMBL241749 | N-benzyl-1-(2-chloro-2-(4-chlorophe...)
Affinity DataKi:  110nMAssay Description:Inhibition of human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50343430(CHEMBL1775036 | N-(3-Chlorophenyl)-1-(2-chloro-2-p...)
Affinity DataKi:  120nMAssay Description:Inhibition of AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50224369(1-(2-chloro-2-phenylethyl)-6-(ethylthio)-N-pheneth...)
Affinity DataKi:  130nMAssay Description:Inhibition of human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50262665(CHEMBL478181 | N-(5-(4-fluorobenzyl)thiazol-2-yl)t...)
Affinity DataKi:  130nMAssay Description:Inhibition of Abl kinase (unknown origin) by cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50262669(CHEMBL477343 | N-(5-(3-(trifluoromethyl)benzyl)thi...)
Affinity DataKi:  136nMAssay Description:Inhibition of Abl kinase (unknown origin) by cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50343431(1-(2-Chloro-2-phenylethyl)-6-[(2-morpholin-4-yleth...)
Affinity DataKi:  150nMAssay Description:Inhibition of AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50224382(CHEMBL399627 | N-(3-bromophenyl)-1-(2-chloro-2-(4-...)
Affinity DataKi:  150nMAssay Description:Inhibition of human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50224376(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenyl)-6-(p...)
Affinity DataKi:  150nMAssay Description:Inhibition of human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86856(CAS_44454904 | N-(5-(4-nitrobenzylthio)-1,3,4-thia...)
Affinity DataKi:  165nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86867(CAS_4573026 | N-(5-(3-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  167nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86866(CAS_44454722 | N-(5-(3-chlorobenzylthio)-1,3,4-thi...)
Affinity DataKi:  169nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50262671(CHEMBL477344 | N-(5-(2-fluorobenzyl)thiazol-2-yl)t...)
Affinity DataKi:  170nMAssay Description:Inhibition of Abl kinase (unknown origin) by cell free assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86870(CAS_44454776 | N-(5-(4-nitrobenzylthio)-1,3,4-thia...)
Affinity DataKi:  170nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86864(CAS_44454803 | N-(5-(4-methoxybenzylthio)-1,3,4-th...)
Affinity DataKi:  189nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50343430(CHEMBL1775036 | N-(3-Chlorophenyl)-1-(2-chloro-2-p...)
Affinity DataKi:  190nMAssay Description:Inhibition of c-SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86874(CAS_44454498 | N-(5-(3-chlorobenzylthio)-1,3,4-thi...)
Affinity DataKi:  195nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86872(CAS_42805643 | N-(5-(4-methoxybenzylthio)-1,3,4-th...)
Affinity DataKi:  195nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86864(CAS_44454803 | N-(5-(4-methoxybenzylthio)-1,3,4-th...)
Affinity DataKi:  199nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50224380(1-(2-chloro-2-phenylethyl)-N-(3-chlorophenethyl)-6...)
Affinity DataKi:  200nMAssay Description:Inhibition of human recombinant AblMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86860(CAS_3320545 | N-(5-(4-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  200nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM50343431(1-(2-Chloro-2-phenylethyl)-6-[(2-morpholin-4-yleth...)
Affinity DataKi:  210nMAssay Description:Inhibition of c-SrcMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86870(CAS_44454776 | N-(5-(4-nitrobenzylthio)-1,3,4-thia...)
Affinity DataKi:  210nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86859(CAS_1327207 | N-(5-(4-bromobenzylthio)-1,3,4-thiad...)
Affinity DataKi:  217nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase ABL1(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86863(CAS_4390766 | N-(5-(3-fluorobenzylthio)-1,3,4-thia...)
Affinity DataKi:  217nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Universit&Aagrov

Curated by PDSP Ki Database
LigandPNGBDBM86857(CAS_44454939 | N-(5-(4-nitrobenzylthio)-1,3,4-thia...)
Affinity DataKi:  219nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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