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Found 228 with Last Name = 'ko' and Initial = 'hh'
TargetBeta-glucuronidase(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibitory effect of compound on the release of Beta-glucuronidase in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50335242(3-Chloro-3'-((2-cyclopentyl-3-oxo-2,3-dihydrobenzo...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of CYP2C9 in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucuronidase(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50142192(3-(2,4-Dihydroxy-phenyl)-5,7-dihydroxy-chromen-4-o...)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibitory effect of compound on the release of Beta-glucuronidase in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 1A2(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50335242(3-Chloro-3'-((2-cyclopentyl-3-oxo-2,3-dihydrobenzo...)
Affinity DataIC50:  6.20E+3nMAssay Description:Inhibition of CYP1A2 in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucuronidase(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM79181(10-[3-(4-methyl-1-piperazinyl)propyl]-2-(trifluoro...)
Affinity DataIC50:  7.80E+3nMAssay Description:Inhibitory effect of compound on the release of Beta-glucuronidase in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50335253(4-Chloro-3'-((2-cyclopentyl-1-oxoisoindolin-5-ylox...)
Affinity DataIC50:  8.15E+3nMAssay Description:Inhibition of radioligand binding to human histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50335253(4-Chloro-3'-((2-cyclopentyl-1-oxoisoindolin-5-ylox...)
Affinity DataIC50:  8.15E+3nMAssay Description:Inhibition of radioligand binding to human adrenergic alpha1a receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 2C9(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50335253(4-Chloro-3'-((2-cyclopentyl-1-oxoisoindolin-5-ylox...)
Affinity DataIC50:  8.20E+3nMAssay Description:Inhibition of CYP2C9 in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysozyme C-1(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM79181(10-[3-(4-methyl-1-piperazinyl)propyl]-2-(trifluoro...)
Affinity DataIC50:  9.00E+3nMAssay Description:Inhibitory effect of compound on the release of lysozyme in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysozyme C-1(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50142192(3-(2,4-Dihydroxy-phenyl)-5,7-dihydroxy-chromen-4-o...)
Affinity DataIC50:  9.70E+3nMAssay Description:Inhibitory effect of compound on the release of lysozyme in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50017268(CHEMBL3287723 | US10099993, Compound 96)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to human histamine H4 receptor at 10 uM by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H2 receptor(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50017268(CHEMBL3287723 | US10099993, Compound 96)
Affinity DataIC50: >1.00E+4nMAssay Description:Binding affinity to human histamine H2 receptor at 10 uM by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 4(Rattus norvegicus (Rat))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50017264(CHEMBL3287718)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat mGlu4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1D adrenergic receptor(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50335253(4-Chloro-3'-((2-cyclopentyl-1-oxoisoindolin-5-ylox...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of radioligand binding to human adrenergic alpha1d receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H1 receptor(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50335242(3-Chloro-3'-((2-cyclopentyl-3-oxo-2,3-dihydrobenzo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of radioligand binding to human histamine H1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50017264(CHEMBL3287718)
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at rat mGlu1 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(1A) dopamine receptor(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50335242(3-Chloro-3'-((2-cyclopentyl-3-oxo-2,3-dihydrobenzo...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of radioligand binding to human dopamine D1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucuronidase(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50077323(7,4'-Dihydroxyflavone | 7-hydroxy-2-(4-hydroxyphen...)
Affinity DataIC50:  1.37E+4nMAssay Description:Inhibitory effect of compound on the release of Beta-glucuronidase in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysozyme C-1(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM7458(5,7-dihydroxy-2-(4-hydroxyphenyl)-4H-chromen-4-one...)
Affinity DataIC50:  1.77E+4nMAssay Description:Inhibitory effect of compound on the release of lysozyme in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCytochrome P450 3A4(Homo sapiens (Human))
Sanford-Burnham Medical Research Institute

Curated by ChEMBL
LigandPNGBDBM50335242(3-Chloro-3'-((2-cyclopentyl-3-oxo-2,3-dihydrobenzo...)
Affinity DataIC50: >2.50E+4nMAssay Description:Inhibition of CYP3A4 in human liver microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysozyme C-1(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50142193(2'-hydroxydaidzein | 3-(2,4-dihydroxyphenyl)-7-hyd...)
Affinity DataIC50:  2.63E+4nMAssay Description:Inhibitory effect of compound on the release of lysozyme in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysozyme C-1(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50142191(5,7-Dihydroxy-3-(4-hydroxy-2-methoxy-phenyl)-chrom...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory effect of compound on the release of lysozyme in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysozyme C-1(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50077323(7,4'-Dihydroxyflavone | 7-hydroxy-2-(4-hydroxyphen...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory effect of compound on the release of lysozyme in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucuronidase(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50142190(2-((11bR,12R)-9-Hydroxy-5b,11b-dihydro-6H-3,7,12-t...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory effect of compound on the release of Beta-glucuronidase in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucuronidase(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50142191(5,7-Dihydroxy-3-(4-hydroxy-2-methoxy-phenyl)-chrom...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory effect of compound on the release of Beta-glucuronidase in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysozyme C-1(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50142190(2-((11bR,12R)-9-Hydroxy-5b,11b-dihydro-6H-3,7,12-t...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory effect of compound on the release of lysozyme in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucuronidase(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50366927(CHEMBL1159471)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory effect of compound on the release of Beta-glucuronidase in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBeta-glucuronidase(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50142193(2'-hydroxydaidzein | 3-(2,4-dihydroxyphenyl)-7-hyd...)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory effect of compound on the release of Beta-glucuronidase in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysozyme C-1(Rattus norvegicus)
Kaohsiung Medical University

Curated by ChEMBL
LigandPNGBDBM50366927(CHEMBL1159471)
Affinity DataIC50: >3.00E+4nMAssay Description:Inhibitory effect of compound on the release of lysozyme in rat neutrophils stimulated with fMLP/CBMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295965(2,3,4'-Trihydroxy-4-methoxydeoxybenzoin | CHEMBL54...)
Affinity DataIC50:  4.31E+4nMAssay Description:Inhibition of mushroom tyrosinase activity after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295965(2,3,4'-Trihydroxy-4-methoxydeoxybenzoin | CHEMBL54...)
Affinity DataIC50:  4.34E+4nMAssay Description:Inhibition of mushroom tyrosinase activity after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295965(2,3,4'-Trihydroxy-4-methoxydeoxybenzoin | CHEMBL54...)
Affinity DataIC50:  4.61E+4nMAssay Description:Inhibition of mushroom tyrosinase activity after 150 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295964(2,4,6-Trihydroxy-4'-methoxydeoxybenzoin | CHEMBL55...)
Affinity DataIC50:  7.11E+4nMAssay Description:Inhibition of mushroom tyrosinase activity after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295962(1-(2,4-dihydroxyphenyl)-2-(4-methoxyphenyl)ethanon...)
Affinity DataIC50:  7.89E+4nMAssay Description:Inhibition of mushroom tyrosinase activity after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295969(2,4,5-Trihydroxy-4'-methoxydeoxybenzoin | CHEMBL55...)
Affinity DataIC50:  8.44E+4nMAssay Description:Inhibition of mushroom tyrosinase activity after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295961(2,4-Dihydroxy-3',4'-dimethoxydeoxybenzoin | CHEMBL...)
Affinity DataIC50:  1.12E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295966(2,3,4-Trihydroxy-3',4'-dimethoxydeoxybenzoin | CHE...)
Affinity DataIC50:  1.32E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50031467(5-HYDROXY-2-(HYDROXYMETHYL)-4H-PYRAN-4-ONE | 5-Hyd...)
Affinity DataIC50:  1.33E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50166034(1-(2,4-Dihydroxy-phenyl)-2-(4-hydroxy-phenyl)-etha...)
Affinity DataIC50:  1.36E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295966(2,3,4-Trihydroxy-3',4'-dimethoxydeoxybenzoin | CHE...)
Affinity DataIC50:  1.40E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 150 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295969(2,4,5-Trihydroxy-4'-methoxydeoxybenzoin | CHEMBL55...)
Affinity DataIC50:  1.44E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295962(1-(2,4-dihydroxyphenyl)-2-(4-methoxyphenyl)ethanon...)
Affinity DataIC50:  1.60E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295960(3,4-Dihydroxy-4'-methoxydeoxybenzoin | CHEMBL55018...)
Affinity DataIC50:  1.68E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50166034(1-(2,4-Dihydroxy-phenyl)-2-(4-hydroxy-phenyl)-etha...)
Affinity DataIC50:  1.72E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 150 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50031467(5-HYDROXY-2-(HYDROXYMETHYL)-4H-PYRAN-4-ONE | 5-Hyd...)
Affinity DataIC50:  1.76E+5nMAssay Description:Inhibition of mushroom tyrosinase after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295960(3,4-Dihydroxy-4'-methoxydeoxybenzoin | CHEMBL55018...)
Affinity DataIC50:  1.78E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 150 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50166034(1-(2,4-Dihydroxy-phenyl)-2-(4-hydroxy-phenyl)-etha...)
Affinity DataIC50:  1.78E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 30 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295962(1-(2,4-dihydroxyphenyl)-2-(4-methoxyphenyl)ethanon...)
Affinity DataIC50:  1.81E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 150 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295969(2,4,5-Trihydroxy-4'-methoxydeoxybenzoin | CHEMBL55...)
Affinity DataIC50:  1.97E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 150 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
National Taiwan University

Curated by ChEMBL
LigandPNGBDBM50295968(2,3,4-Trihydroxy-4'-methoxydeoxybenzoin | CHEMBL26...)
Affinity DataIC50:  2.03E+5nMAssay Description:Inhibition of mushroom tyrosinase activity after 90 mins by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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