Affinity DataKi: 0.560nMAssay Description:Displacement of [3H]-CGS-21680 from human adenosine A2A receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 0.800nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.30nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.60nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 1.80nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 2nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 4.70nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 7.70nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 9.40nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 11.1nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 15.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 16.2nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 21.1nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 22nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 29nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 29.5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 32nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 33nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 33.4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 34nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 44nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 45nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 51.5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 53nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 54nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 56nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 71nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 74nMAssay Description:Displacement of [3H]clonidine from imidazoline receptor I-1 of bovine chromaffin cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 78nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center
Curated by ChEMBL
University Of Minnesota Health Science Center
Curated by ChEMBL
Affinity DataKi: 80.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair