Compile Data Set for Download or QSAR
maximum 50k data
Found 1201 with Last Name = 'may' and Initial = 'k'
TargetAdenosine receptor A2a(Homo sapiens (Human))
Yamasa

Curated by ChEMBL
LigandPNGBDBM50018688(CHEMBL3291301)
Affinity DataKi:  0.560nMAssay Description:Displacement of [3H]-CGS-21680 from human adenosine A2A receptor expressed in HEK293 cells after 90 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203781((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  0.800nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50386999(CHEMBL2049152)
Affinity DataKi:  0.810nMAssay Description:Inhibition of furinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50387001(CHEMBL2049154)
Affinity DataKi:  1nMAssay Description:Inhibition of furinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203803((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203803((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.10nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM26349((2S)-2-[(2S)-2-[(2S)-2-[(2S)-2-amino-3-(4-hydroxyp...)
Affinity DataKi:  1.30nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50387000(CHEMBL2049153)
Affinity DataKi:  1.60nMAssay Description:Inhibition of furinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203782((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.60nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203794((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203811((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  2nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50387002(CHEMBL2049155)
Affinity DataKi:  3.30nMAssay Description:Inhibition of furinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203802((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  4.70nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203814((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082670(4-(4-Chloro-phenyl)-1-(4,4-diphenyl-butyl)-4-hydro...)
Affinity DataKi:  6nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203813((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  7.70nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082715(4-(4-Chloro-phenyl)-1-(4-cyano-4,4-diphenyl-butyl)...)
Affinity DataKi:  8nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082729(1-{5-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl...)
Affinity DataKi:  9nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203816((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  9.30nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203791((2S)-N-[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1-{[(1S)-1...)
Affinity DataKi:  9.40nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203800((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  11.1nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203779((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  15.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203789((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  16.2nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203810((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  21.1nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082682(5-{3-[4-(4-Bromo-phenyl)-4-hydroxy-piperidin-1-yl]...)
Affinity DataKi:  22nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082694(4-(4-Chloro-phenyl)-1-(4-cyano-4-naphthalen-2-yl-b...)
Affinity DataKi:  22nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082671(5-{3-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl...)
Affinity DataKi:  24nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082737(9-{3-[4-(4-Bromo-phenyl)-4-hydroxy-piperidin-1-yl]...)
Affinity DataKi:  29nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203780((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  29.5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082690(11-{3-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-y...)
Affinity DataKi:  32nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082720(5-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-2...)
Affinity DataKi:  33nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203787((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  33.4nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082706(11-{3-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-y...)
Affinity DataKi:  34nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082705(5-{3-[4-(4-Fluoro-phenyl)-4-hydroxy-piperidin-1-yl...)
Affinity DataKi:  44nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082688(5-{3-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl...)
Affinity DataKi:  45nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082668(5-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-2...)
Affinity DataKi:  51nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203799((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  51.5nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50027216(5-(4-(4-chlorophenyl)-4-hydroxy-piperidin-1-yl)-2,...)
Affinity DataKi:  52nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082716(5-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-2...)
Affinity DataKi:  53nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50386998(CHEMBL2049151)
Affinity DataKi:  53nMAssay Description:Inhibition of furinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082733(5-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-2...)
Affinity DataKi:  54nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082674(5-{3-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl...)
Affinity DataKi:  56nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50386989(CHEMBL2049013)
Affinity DataKi:  63nMAssay Description:Inhibition of furinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082692(5-{3-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl...)
Affinity DataKi:  71nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082692(5-{3-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl...)
Affinity DataKi:  71nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082701(2-(3-Bromo-4-methoxy-phenyl)-5-[4-(4-chloro-phenyl...)
Affinity DataKi:  74nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50070328(CHEBI:8862 | Rilmenidine)
Affinity DataKi:  74nMAssay Description:Displacement of [3H]clonidine from imidazoline receptor I-1 of bovine chromaffin cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-C chemokine receptor type 1(Homo sapiens (Human))
Berlex Biosciences

Curated by ChEMBL
LigandPNGBDBM50082691(6-[4-(4-Chloro-phenyl)-4-hydroxy-piperidin-1-yl]-2...)
Affinity DataKi:  78nMAssay Description:Inhibition of [125I]-MIP-1 alpha binding to recombinant human C-C chemokine receptor type 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Torrey Pines Institute For Molecular Studies

Curated by ChEMBL
LigandPNGBDBM50386987(CHEMBL2049015)
Affinity DataKi:  78nMAssay Description:Inhibition of furinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKiSS-1 receptor(Homo sapiens (Human))
University Of Minnesota Health Science Center

Curated by ChEMBL
LigandPNGBDBM50203797((2S)-2-{[(2S)-1-[(2S)-2-amino-4-methylpentanoyl]py...)
Affinity DataKi:  80.8nMAssay Description:Displacement of [125]metastin from metastin receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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