Affinity DataKi: 0.300nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 0.420nMAssay Description:Inhibitory constant against dopamine D2 receptor using 0.2 nM [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 0.490nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Inhibitory constant was determined against 5-hydroxytryptamine 1A receptor using 1.2 nM [3H]8-OH-DPATMore data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 1.48nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 1.59nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 1.70nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 2.20nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 2.52nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 2.66nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 2.69nMAssay Description:Inhibitory constant against dopamine D2 receptor using 0.2 nM [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 3.02nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 3.38nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 3.38nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 3.61nMAssay Description:Inhibitory constant against Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 3.61nMAssay Description:Inhibitory constant against dopamine D2 receptor using 0.2 nM [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 3.61nMAssay Description:Inhibitory constant against Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 3.61nMAssay Description:Inhibitory constant against Dopamine receptor D2More data for this Ligand-Target Pair
Affinity DataKi: 3.80nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 4.63nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 4.75nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 5.35nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 5.98nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 6.65nMAssay Description:Inhibitory constant against dopamine D2 receptor using 0.2 nM [3H]-spiperoneMore data for this Ligand-Target Pair
Affinity DataKi: 7.90nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 9.40nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 9.80nMAssay Description:Inhibitory activity against Xanthine OxidaseMore data for this Ligand-Target Pair
Affinity DataKi: 9.90nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 11.5nMAssay Description:Inhibitory constant was determined against 5-hydroxytryptamine 1A receptor using 1.2 nM [3H]8-OH-DPATMore data for this Ligand-Target Pair
Affinity DataKi: 11.6nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 11.9nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 12.2nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 14.1nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 15.4nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair
Affinity DataKi: 16nMAssay Description:Inhibitory constant against sigma receptor type 2 using 3 nM [3H]ditolylguanidineMore data for this Ligand-Target Pair
Affinity DataKi: 16.2nMAssay Description:Inhibitory constant against sigma receptor type 1 using 3 nM [3H]pentazocineMore data for this Ligand-Target Pair