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Found 68 with Last Name = 'tanaka' and Initial = 'r'
TargetBeta-secretase 1(Homo sapiens (Human))
National Institute Of Health Sciences

Curated by ChEMBL
LigandPNGBDBM50157300((1-{(S)-2-Allylcarbamoyl-1-[(1S,2S,4R)-4-((S)-1-be...)
Affinity DataKi:  27nMAssay Description:Binding affinity against human brain memapsin 2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
National Institute Of Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50335557(CHEMBL1652605 | N,N-dipropyl-N'-[4-({[(1H-imidazol...)
Affinity DataIC50:  0.610nMAssay Description:Displacement of [125I]SDF-1alpha form CXCR4 expressed in CHO cells by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128787(4-[4-(2-Bromo-phenyl)-3-nitro-1-pyridin-3-ylmethyl...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128787(4-[4-(2-Bromo-phenyl)-3-nitro-1-pyridin-3-ylmethyl...)
Affinity DataIC50:  1.90nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
National Institute Of Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50335557(CHEMBL1652605 | N,N-dipropyl-N'-[4-({[(1H-imidazol...)
Affinity DataIC50:  2.80nMAssay Description:Inhibition of Mab 12G5 binding to wild type CXCR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128790(4-[4-(2-Bromo-phenyl)-3-nitro-1-pyridin-3-ylmethyl...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128790(4-[4-(2-Bromo-phenyl)-3-nitro-1-pyridin-3-ylmethyl...)
Affinity DataIC50:  8.20nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128796(4-[4-(2-Bromo-phenyl)-3-nitro-1-pyridin-3-ylmethyl...)
Affinity DataIC50:  13nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128795(4-(2-Bromo-phenyl)-6-(3,4-dihydroxy-phenyl)-5-nitr...)
Affinity DataIC50:  30nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128800(6-(3-Amino-4-hydroxy-phenyl)-4-(2-bromo-phenyl)-5-...)
Affinity DataIC50:  97nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128789(4-(2-Bromo-phenyl)-6-(4-hydroxy-phenyl)-5-nitro-1-...)
Affinity DataIC50:  140nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetC-X-C chemokine receptor type 4(Homo sapiens (Human))
National Institute Of Infectious Diseases

Curated by ChEMBL
LigandPNGBDBM50035696(1,1''-{1,4-phenylenebis(methylene)}-bis{1,4,8,11-t...)
Affinity DataIC50:  289nMAssay Description:Inhibition of Mab 12G5 binding to wild type CXCR4 expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128790(4-[4-(2-Bromo-phenyl)-3-nitro-1-pyridin-3-ylmethyl...)
Affinity DataIC50: >310nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128787(4-[4-(2-Bromo-phenyl)-3-nitro-1-pyridin-3-ylmethyl...)
Affinity DataIC50: >310nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128793(4-(3-Chloro-phenyl)-6-(4-hydroxy-phenyl)-5-nitro-1...)
Affinity DataIC50:  320nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128794(4-(3-Bromo-phenyl)-6-(4-hydroxy-phenyl)-5-nitro-1-...)
Affinity DataIC50:  350nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128794(4-(3-Bromo-phenyl)-6-(4-hydroxy-phenyl)-5-nitro-1-...)
Affinity DataIC50:  350nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128801(6-(4-Hydroxy-phenyl)-5-nitro-1-pyridin-3-ylmethyl-...)
Affinity DataIC50:  410nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University Of Science

Curated by ChEMBL
LigandPNGBDBM15236(3,5,7-trihydroxy-2-(3,4,5-trihydroxyphenyl)-4H-chr...)
Affinity DataIC50:  560nMAssay Description:Inhibition of recombinant human His-tagged glyoxalase 1 expressed in Escherichia coli BL21 assessed as formation of S-D-lactoylglutathione after 5 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128789(4-(2-Bromo-phenyl)-6-(4-hydroxy-phenyl)-5-nitro-1-...)
Affinity DataIC50:  950nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128789(4-(2-Bromo-phenyl)-6-(4-hydroxy-phenyl)-5-nitro-1-...)
Affinity DataIC50:  950nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128802(6-(4-Hydroxy-phenyl)-5-nitro-4-phenyl-1-pyridin-3-...)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128791(4-(2-Bromo-phenyl)-6-(4-hydroxy-3-hydroxymethyl-ph...)
Affinity DataIC50: >1.20E+3nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128803(4-(2-Bromo-phenyl)-6-(4-methoxy-phenyl)-5-nitro-1-...)
Affinity DataIC50: >1.20E+3nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128795(4-(2-Bromo-phenyl)-6-(3,4-dihydroxy-phenyl)-5-nitr...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128795(4-(2-Bromo-phenyl)-6-(3,4-dihydroxy-phenyl)-5-nitr...)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50483935(CHEMBL1783812)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50483937(CHEMBL1783813)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50474910(CHEMBL189836)
Affinity DataIC50:  1.86E+3nMAssay Description:Inhibitory concentration against human DNA topoisomerase IIMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLactoylglutathione lyase(Homo sapiens (Human))
Tokyo University Of Science

Curated by ChEMBL
LigandPNGBDBM50355547(CHEMBL1910548)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of recombinant human His-tagged glyoxalase 1 expressed in Escherichia coli BL21 assessed as formation of S-D-lactoylglutathione after 5 mi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50483932(Betulin 3,28-Diacetate | Betulin Diacetate)
Affinity DataIC50:  2.65E+3nMAssay Description:Antiviral activity against HIV1 Reverse transcriptase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50483934(24-Methylenecycloartanol Ferulate | 24-Methylenecy...)
Affinity DataIC50:  3.07E+3nMAssay Description:Antiviral activity against HIV1 Reverse transcriptase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50483936(3-O-Ferulylcycloartenol | Cycloartenol Ferulate | ...)
Affinity DataIC50:  3.64E+3nMAssay Description:Antiviral activity against HIV1 Reverse transcriptase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128792(5-Amino-4-(3-bromo-phenyl)-6-(4-hydroxy-phenyl)-1-...)
Affinity DataIC50: >3.70E+3nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128798(4-(3-Bromo-phenyl)-5-hydroxyamino-6-(4-hydroxy-phe...)
Affinity DataIC50: >3.70E+3nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128799(4-(3-Bromo-phenyl)-6-(4-hydroxy-phenyl)-5-nitro-1-...)
Affinity DataIC50: >3.70E+3nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128797(4-(4-Bromo-phenyl)-6-(4-hydroxy-phenyl)-5-nitro-1-...)
Affinity DataIC50: >3.70E+3nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50128788(4-(3-Bromo-phenyl)-6-(4-hydroxy-phenyl)-5-nitro-1-...)
Affinity DataIC50: >3.70E+3nMAssay Description:Inhibition of bovine brain farnesyltransferase (FTase) farnesylation of viral K-RasMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50346601(NSC-114945 | OLEANOLIC_ACID | Oleanolic acid | Ole...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM23208((1R,2R,5S,8R,9R,10R,13R,14R,17S,19R)-17-hydroxy-1,...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50483933(CHEMBL1783816 | Karounidiol 29-Benzoate)
Affinity DataIC50:  4.03E+3nMAssay Description:Antiviral activity against HIV1 Reverse transcriptase activityMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetReverse transcriptase(Human immunodeficiency virus 1)
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50241944(CHEMBL486393 | Lupenone | lupeone)
Affinity DataIC50:  4.94E+3nMAssay Description:Antiviral activity against HIV1 Reverse transcriptase activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataIC50:  6.00E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50148911((3beta)-3-hydroxyurs-12-en-28-oic acid | 3beta-hyd...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtease(Human immunodeficiency virus 1 (HIV-1))
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50346601(NSC-114945 | OLEANOLIC_ACID | Oleanolic acid | Ole...)
Affinity DataIC50:  8.00E+3nMAssay Description:Inhibition of HIV1 protease activityMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Osaka University Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50377927(Clerodol | Fagarasterol | Farganasterol | LUPEOL |...)
Affinity DataIC50:  1.04E+4nMAssay Description:Inhibition of human 1 unit topoisomerase 2alpha catalytic activity assessed as relaxation of 198 ng supercoiled pBR322 DNA by agarose gel electrophor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha(Homo sapiens (Human))
Osaka University Of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50260250(CHEMBL491188 | Olean-12-en-3beta,15alpha-diol)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of human 1 unit topoisomerase 2alpha catalytic activity assessed as relaxation of 198 ng supercoiled pBR322 DNA by agarose gel electrophor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50474907(CHEMBL193251)
Affinity DataIC50:  1.83E+4nMAssay Description:Inhibitory concentration against human DNA topoisomerase IIMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetDNA topoisomerase 2-alpha/2-beta(Homo sapiens (Human))
Osaka University of Pharmaceutical Sciences

Curated by ChEMBL
LigandPNGBDBM50474904(CHEMBL191216)
Affinity DataIC50:  2.27E+4nMAssay Description:Inhibitory concentration against human DNA topoisomerase IIMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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