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Found 1150 with Last Name = 'england' and Initial = 's'
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataKi:  1nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513361(CHEMBL4567766)
Affinity DataKi:  1nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513360(CHEMBL4573390)
Affinity DataKi:  2nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513345(CHEMBL4438830)
Affinity DataKi:  2nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50151923(CHEMBL3774537)
Affinity DataKi:  2nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513344(CHEMBL4447515)
Affinity DataKi:  3nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50151923(CHEMBL3774537)
Affinity DataKi:  3nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278288(2-(2-(4-(2,3-dihydro-1H-inden-2-ylamino)pyrido[3,4...)
Affinity DataKi:  3nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513361(CHEMBL4567766)
Affinity DataKi:  3nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513348(CHEMBL4585876)
Affinity DataKi:  4nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513344(CHEMBL4447515)
Affinity DataKi:  4nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513348(CHEMBL4585876)
Affinity DataKi:  4nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataKi:  4nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513360(CHEMBL4573390)
Affinity DataKi:  5nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278286(CHEMBL511266 | N4-(2,3-dihydro-1H-inden-2-yl)-N6-(...)
Affinity DataKi:  5nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278407(CHEMBL470396 | N-cycloheptyl-6-(2-morpholinoethoxy...)
Affinity DataKi:  6nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513343(CHEMBL4449500)
Affinity DataKi:  7nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278361(CHEMBL471435 | N4-cyclohexyl-N6-(2-morpholinoethyl...)
Affinity DataKi:  10nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278289(CHEMBL469383 | N4-cyclohexyl-N6-(2-methoxyethyl)py...)
Affinity DataKi:  11nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278112(CHEMBL472490 | N4-(2,3-dihydro-1H-inden-2-yl)-N6-m...)
Affinity DataKi:  14nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5B(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513346(CHEMBL4525269)
Affinity DataKi:  16nMAssay Description:Binding affinity to KDM5B (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278358(1-(2-(4-(cyclohexylamino)pyrido[3,4-d]pyrimidin-6-...)
Affinity DataKi:  20nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278232(2-(4-(2,3-dihydro-1H-inden-2-ylamino)pyrido[3,4-d]...)
Affinity DataKi:  21nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50513346(CHEMBL4525269)
Affinity DataKi:  26nMAssay Description:Binding affinity to KDM4A (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278114(CHEMBL513012 | N-cyclohexylquinazolin-4-amine)
Affinity DataKi:  27nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278231(CHEMBL513018 | N4,N6-bis(2,3-dihydro-1H-inden-2-yl...)
Affinity DataKi:  31nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278357(3-(4-(cyclohexylamino)pyrido[3,4-d]pyrimidin-6-ylo...)
Affinity DataKi:  33nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278153(CHEMBL471242 | N-(2,3-dihydro-1H-inden-2-yl)quinaz...)
Affinity DataKi:  34nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50346870(CHEMBL1797647)
Affinity DataKi:  40nMAssay Description:Inhibition of human recombinant KDM1A expressed in Escherichia coli using H3K4me as substrate by peroxidase coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278362(CHEMBL512523 | N-cyclohexyl-6-(2-morpholinoethoxy)...)
Affinity DataKi:  42nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278111(CHEMBL472489 | N4-(2,3-dihydro-1H-inden-2-yl)-N4,N...)
Affinity DataKi:  54nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM113742(N-[4-(2-Hydrazinylethyl)phenyl]-4-phenylbutanamide...)
Affinity DataKi:  59nMAssay Description:Inhibition of GST-tagged KDM1A (unknown origin) expressed in Escherichia coli BL21-CodonPlus-(DE3)-RIPL cells using dimethyl-Lys-4 H3-21 as substrate...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278291(CHEMBL471666 | N-cyclohexyl-6-(2-methoxyethoxy)pyr...)
Affinity DataKi:  101nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278287(CHEMBL469381 | N4-(2,3-dihydro-1H-inden-2-yl)-N6-(...)
Affinity DataKi:  102nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278113(CHEMBL513761 | N-(2,3-dihydro-1H-inden-2-yl)-6-met...)
Affinity DataKi:  115nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278229(2-(6-(2,3-dihydro-1H-inden-2-ylamino)pyrido[3,4-d]...)
Affinity DataKi:  125nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158884(CHEMBL3785550)
Affinity DataKi:  140nMAssay Description:Inhibition of human recombinant His-tagged KDM1A (171 to 836 residues) using H3K4me2 as substrate by peroxidase coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278228(CHEMBL447113 | N6-(2,3-dihydro-1H-inden-2-yl)-N4-m...)
Affinity DataKi:  160nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278290(2-(4-(cyclohexylamino)pyrido[3,4-d]pyrimidin-6-ylo...)
Affinity DataKi:  177nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278853(CHEMBL496897 | N4-(2,3-dihydro-1H-inden-2-yl)-N6,N...)
Affinity DataKi:  185nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278850(CHEMBL497918 | N4-cyclohexyl-N6,N6-dimethylpyrido[...)
Affinity DataKi:  199nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278360(CHEMBL471434 | N6-(3-aminopropyl)-N4-cyclohexylpyr...)
Affinity DataKi:  200nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158882(CHEMBL3786209)
Affinity DataKi:  210nMAssay Description:Inhibition of human recombinant His-tagged KDM1A (171 to 836 residues) using H3K4me2 as substrate by peroxidase coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158883(CHEMBL3785964)
Affinity DataKi:  240nMAssay Description:Inhibition of human recombinant His-tagged KDM1A (171 to 836 residues) using H3K4me2 as substrate by peroxidase coupled enzyme assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158852(CHEMBL3785340)
Affinity DataKi:  280nMAssay Description:Competitive inhibition of recombinant His6-tagged KDM2A (1 to 517 residues) (unknown origin) expressed in Escherichia coli BL21 cells using methylsta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278110(CHEMBL511838 | N4-(2,3-dihydro-1H-inden-2-yl)-N4,N...)
Affinity DataKi:  300nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50158852(CHEMBL3785340)
Affinity DataKi:  420nMAssay Description:Competitive inhibition of recombinant His6-tagged KDM4A (1 to 359 residues) (unknown origin) expressed in Escherichia coli BL21 cells using methylsta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 2A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50158851(CHEMBL3786265)
Affinity DataKi:  420nMAssay Description:Competitive inhibition of recombinant His6-tagged KDM2A (1 to 517 residues) (unknown origin) expressed in Escherichia coli BL21 cells using methylsta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 4A(Homo sapiens (Human))
Institute of Cancer Research

Curated by ChEMBL
LigandPNGBDBM50158851(CHEMBL3786265)
Affinity DataKi:  520nMAssay Description:Competitive inhibition of recombinant His6-tagged KDM4A (1 to 359 residues) (unknown origin) expressed in Escherichia coli BL21 cells using methylsta...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Medical Research Council Technology

Curated by ChEMBL
LigandPNGBDBM50278116(4-(cyclohexyloxy)quinazoline | CHEMBL471866)
Affinity DataKi:  694nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as inhibition of glutamate-evoked increase in calcium internalization preincubated...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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