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Found 369 with Last Name = 'solmajer' and Initial = 't'
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141559(Azaphenylalanine derivative | CHEMBL37318)
Affinity DataKi:  4nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141568(Azaphenylalanine derivative | CHEMBL38626)
Affinity DataKi:  5nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141554(Azaphenylalanine derivative | CHEMBL41947)
Affinity DataKi:  9nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141566(Azaphenylalanine derivative | CHEMBL40043)
Affinity DataKi:  11nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141565(Azaphenylalanine derivative | CHEMBL288862)
Affinity DataKi:  32nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141570(Azaphenylalanine derivative | CHEMBL291101)
Affinity DataKi:  45nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141554(Azaphenylalanine derivative | CHEMBL41947)
Affinity DataKi:  53nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141558(Azaphenylalanine derivative | CHEMBL39760)
Affinity DataKi:  85nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141560(Azaphenylalanine derivative | CHEMBL41220)
Affinity DataKi:  95nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141559(Azaphenylalanine derivative | CHEMBL37318)
Affinity DataKi:  110nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50132526(CHEMBL320542 | N-(2-Amino-4,5,6,7-tetrahydro-benzo...)
Affinity DataKi:  120nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124076((S)-1-((R)-3-Cyclohexyl-1-oxo-2-phenylmethanesulfo...)
Affinity DataKi:  140nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141568(Azaphenylalanine derivative | CHEMBL38626)
Affinity DataKi:  140nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141555(Azaphenylalanine derivative | CHEMBL43017)
Affinity DataKi:  150nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50132525(2-(6-Methyl-2-oxo-3-phenylmethanesulfonylamino-2H-...)
Affinity DataKi:  170nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141564(Azaphenylalanine derivative | CHEMBL39587)
Affinity DataKi:  210nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124071(((R)-1-Cyclohexylmethyl-2-oxo-2-{(S)-2-[(4,5,6,7-t...)
Affinity DataKi:  280nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50132522(CHEMBL100181 | N-(1H-Indazol-5-ylmethyl)-2-(6-meth...)
Affinity DataKi:  301nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124073((S)-1-((R)-2-Amino-1-oxo-3,3-diphenyl-propyl)-pyrr...)
Affinity DataKi:  360nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141569(Azaphenylalanine derivative | CHEMBL39590)
Affinity DataKi:  380nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141571(Azaphenylalanine derivative | CHEMBL37857)
Affinity DataKi:  430nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141561(Azaphenylalanine derivative | CHEMBL38491)
Affinity DataKi:  470nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124083(((R)-1-Benzhydryl-2-oxo-2-{(S)-2-[(4,5,6,7-tetrahy...)
Affinity DataKi:  530nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141562(Azaphenylalanine derivative | CHEMBL39078)
Affinity DataKi:  590nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141563(Azaphenylalanine derivative | CHEMBL289331)
Affinity DataKi:  610nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124075((S)-1-[(R)-2-Amino-3-(3,4-dichloro-phenyl)-1-oxo-p...)
Affinity DataKi:  690nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141567(Azaphenylalanine derivative | CHEMBL39911)
Affinity DataKi:  770nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141573(Azaphenylalanine derivative | CHEMBL38467)
Affinity DataKi:  1.60E+3nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141556(Azaphenylalanine derivative | CHEMBL36960)
Affinity DataKi:  1.90E+3nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50132523(CHEMBL110565 | N-(2-Amino-4,5,6,7-tetrahydro-benzo...)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141554(Azaphenylalanine derivative | CHEMBL41947)
Affinity DataKi:  3.00E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124077(((R)-1-(3,4-Dichloro-benzyl)-2-oxo-2-{(S)-2-[(4,5,...)
Affinity DataKi:  3.33E+3nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141568(Azaphenylalanine derivative | CHEMBL38626)
Affinity DataKi:  3.90E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141572(Azaphenylalanine derivative | CHEMBL41359)
Affinity DataKi:  4.20E+3nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124072(((R)-2-{(S)-2-[(2-Amino-5,6,7,8-tetrahydro-quinazo...)
Affinity DataKi:  4.50E+3nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50132527(2-(6-Methyl-2-oxo-3-phenylmethanesulfonylamino-2H-...)
Affinity DataKi:  4.70E+3nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141559(Azaphenylalanine derivative | CHEMBL37318)
Affinity DataKi:  5.30E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124078((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  5.38E+3nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141557(Azaphenylalanine derivative | CHEMBL43817)
Affinity DataKi:  5.40E+3nMAssay Description:In vitro inhibition of Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50132528(CHEMBL321895 | N-(2-Amino-5,6,7,8-tetrahydro-quina...)
Affinity DataKi:  6.90E+3nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141565(Azaphenylalanine derivative | CHEMBL288862)
Affinity DataKi:  1.00E+4nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50132529(2-(6-Methyl-2-oxo-3-phenylmethanesulfonylamino-2H-...)
Affinity DataKi:  1.18E+4nMAssay Description:Inhibitory activity against thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141557(Azaphenylalanine derivative | CHEMBL43817)
Affinity DataKi:  1.20E+4nMAssay Description:In vitro inhibition of human alpha-thrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124074((S)-1-((R)-3-Cyclohexyl-2-phenylmethanesulfonylami...)
Affinity DataKi:  1.28E+4nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124084((S)-1-((R)-2-Amino-3,3-diphenyl-propionyl)-pyrroli...)
Affinity DataKi:  1.29E+4nMAssay Description:In vitro inhibitory activity against ThrombinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141564(Azaphenylalanine derivative | CHEMBL39587)
Affinity DataKi:  1.30E+4nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141560(Azaphenylalanine derivative | CHEMBL41220)
Affinity DataKi:  1.30E+4nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141563(Azaphenylalanine derivative | CHEMBL289331)
Affinity DataKi:  1.70E+4nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50141570(Azaphenylalanine derivative | CHEMBL291101)
Affinity DataKi:  1.80E+4nMAssay Description:In vitro inhibition of trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine protease 1(Homo sapiens (Human))
University Of Ljubljana

Curated by ChEMBL
LigandPNGBDBM50124071(((R)-1-Cyclohexylmethyl-2-oxo-2-{(S)-2-[(4,5,6,7-t...)
Affinity DataKi:  1.99E+4nMAssay Description:In vitro inhibitory activity against TrypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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