Affinity DataKi: 3nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 6.20nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
Affinity DataKi: 7nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 9nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 9.30nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
Affinity DataKi: 11nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
TargetUrokinase-type plasminogen activator(Homo sapiens (Human))
University Of Antwerp
Curated by ChEMBL
University Of Antwerp
Curated by ChEMBL
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 16nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Displacement of [3H]-5-CT from human 5-HT7R expressed in human HEK293 cells assessed as inhibitory constant incubated for 1 hr by radioligand binding...More data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Displacement of [3H]-8-OH-DPAT from human 5-HT1A expressed in human HEK293 cells assessed as inhibitory constant incubated for 1 hr by radioligand bi...More data for this Ligand-Target Pair
Affinity DataKi: 23nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 27nMAssay Description:Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...More data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 30nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 41nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 53nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 77nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 81nMAssay Description:Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...More data for this Ligand-Target Pair
Affinity DataKi: 87nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 92nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 99nMAssay Description:Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...More data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 99nMAssay Description:Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...More data for this Ligand-Target Pair
Affinity DataKi: 111nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 118nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 126nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 128nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 129nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 132nMAssay Description:Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...More data for this Ligand-Target Pair
Affinity DataKi: 148nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 159nMAssay Description:Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...More data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 177nMAssay Description:Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...More data for this Ligand-Target Pair
Affinity DataKi: 197nMAssay Description:Displacement of [3H]-Ketanserin from human 5-HT2A expressed in CHO-K1 cells incubated for 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 197nMAssay Description:Displacement of [3H]-Ketanserin from human 5-HT2A expressed in CHO-K1 cells incubated for 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 200nMAssay Description:Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...More data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 201nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
Affinity DataKi: 207nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 227nMAssay Description:Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...More data for this Ligand-Target Pair
Affinity DataKi: 235nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 242nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 329nMAssay Description:Displacement of [3H]-raclopride from human D2L receptor expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 338nMAssay Description:Displacement of [3H]-PK11195 from wild type TSPO (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 90 m...More data for this Ligand-Target Pair
Affinity DataKi: 355nMAssay Description:Displacement of [3H]-LSD from human 5-HT6R expressed in human HEK293 cells incubated for 1 hr by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 376nMAssay Description:Displacement of [3H]-Ketanserin from human 5-HT2A expressed in CHO-K1 cells incubated for 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 406nMAssay Description:Displacement of [3H]-Ketanserin from human 5-HT2A expressed in CHO-K1 cells incubated for 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 407nMAssay Description:Displacement of [3H]-Ketanserin from human 5-HT2A expressed in CHO-K1 cells incubated for 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 430nMAssay Description:Displacement of [3H]-Ketanserin from human 5-HT2A expressed in CHO-K1 cells incubated for 1.5 hrs by radioligand binding assayMore data for this Ligand-Target Pair
TargetTranslocator protein(Homo sapiens (Human))
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Faculty Of Science And The University Of Sydney
Curated by ChEMBL
Affinity DataKi: 460nMAssay Description:Displacement of [3H]-PK11195 from TSPO A147T mutant (unknown origin) expressed in human HEK293T cells assessed as inhibitory constant incubated for 9...More data for this Ligand-Target Pair