TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 970nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 1.30E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 1.70E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 2.30E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 2.30E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 2.40E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 4.30E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 4.30E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 5.25E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 8.70E+3nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 1.37E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 1.42E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 2.12E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 2.15E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 3.92E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 5.84E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 8.83E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 9.90E+4nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 1.01E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 1.04E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 1.12E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
TargetBcl-2-like protein 2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 1.16E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-wMore data for this Ligand-Target Pair
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 1.34E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 1.61E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
TargetBcl2-associated agonist of cell death(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 1.76E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl-XlMore data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 2.26E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 2.43E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: 2.60E+5nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
TargetApoptosis regulator Bcl-2(Homo sapiens (Human))
University Of Minnesota Minneapolis
Curated by ChEMBL
University Of Minnesota Minneapolis
Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Inhibition of Bak peptide binding to human recombinant Bcl2More data for this Ligand-Target Pair
Affinity DataIC50: 250nMAssay Description:Binding affinity to recombinant human full length GST-tagged BAX expressed in Escherichia coli BL21 (DE3) measured after 20 mins by fluorescence pola...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 3.30E+3nMAssay Description:Binding affinity to recombinant human full length GST-tagged BAX expressed in Escherichia coli BL21 (DE3) measured after 20 mins by fluorescence pola...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 4.00E+3nMAssay Description:Inhibition of recombinant human BAX expressed in Escherichia coli BL21 (DE3) assessed as inhibition of liposome permeabilization and measured for 2 h...More data for this Ligand-Target Pair
Ligand Info
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of recombinant human BAX expressed in Escherichia coli BL21 (DE3) assessed as inhibition of liposome permeabilization and measured for 2 h...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKd: 3.70E+4nMAssay Description:Binding affinity to BAX (unknown origin) assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Affinity DataKd: 1.50E+4nMAssay Description:Binding affinity to recombinant human BAX (1 to 92 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant incubated for...More data for this Ligand-Target Pair
Ligand Info
Affinity DataKd: 1.50E+4nMAssay Description:Binding affinity to recombinant human BAX (1 to 92 residues) expressed in Escherichia coli BL21 (DE3) assessed as dissociation constant incubated for...More data for this Ligand-Target Pair
Affinity DataKd: 255nMAssay Description:Binding affinity to recombinant human BAX assessed as dissociation constant by ITC analysisMore data for this Ligand-Target Pair
Ligand Info