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Found 59 with Last Name = 'aubertin' and Initial = 'am'
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50029662(3-Amino-4-(3,5-dimethyl-phenylsulfanyl)-5-ethyl-6-...)
Affinity DataIC50:  15nMAssay Description:Inhibition of HIV-1 reverse transcriptase(RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Institut Curie

LigandPNGBDBM10908(3-(dimethylamino)-4-[(3,5-dimethylphenyl)methyl]-5...)
Affinity DataIC50:  20nMpH: 8.0 T: 2°CAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50029665(4-(3,5-Dimethyl-phenylsulfanyl)-5-ethyl-6-methyl-3...)
Affinity DataIC50:  30nMAssay Description:Inhibition of HIV-1 reverse transcriptase(RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Institut Curie

LigandPNGBDBM10903(4-[(3,5-dimethylphenyl)sulfanyl]-5-ethyl-6-methyl-...)
Affinity DataIC50:  30nMpH: 8.0 T: 2°CAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Institut Curie

LigandPNGBDBM10905(3-Amino-4-(3,5-dimethylbenzyl)-5-ethyl-6-methylpyr...)
Affinity DataIC50:  100nMpH: 8.0 T: 2°CAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Institut Curie

LigandPNGBDBM10906(3-Amino-4-(3,5-dimethylbenzoyl)-5-ethyl-6-methylpy...)
Affinity DataIC50:  100nMpH: 8.0 T: 2°CAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50029660(3-Amino-4-(3,5-dimethyl-phenylsulfanyl)-5-methyl-1...)
Affinity DataIC50:  100nMAssay Description:Inhibition of HIV-1 reverse transcriptase(RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Institut Curie

LigandPNGBDBM1434(11-cyclopropyl-5,11-dihydro-4-methyl-6H-dipyrido[3...)
Affinity DataIC50:  200nMpH: 8.0 T: 2°CAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Institut Curie

LigandPNGBDBM10907(4-(3,5-Dimethylbenzyl)-5-ethyl-3-formamido-6-methy...)
Affinity DataIC50:  200nMpH: 8.0 T: 2°CAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [588-1027]/[588-1147](Human immunodeficiency virus type 1)
Institut Curie

LigandPNGBDBM10904(1-[(benzyloxy)methyl]-5-methyl-6-(phenylsulfanyl)-...)
Affinity DataIC50:  300nMpH: 8.0 T: 2°CAssay Description:The IC50 of reverse transcriptase is the concentration that inhibits 50% of recombinant HIV-1 RT RNA-directed DNA polymerase activity in vitro.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50029678(4-(3,5-Dimethyl-phenylsulfanyl)-5-ethyl-6-methyl-1...)
Affinity DataIC50:  400nMAssay Description:Inhibition of HIV-1 reverse transcriptase(RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM10904(1-[(benzyloxy)methyl]-5-methyl-6-(phenylsulfanyl)-...)
Affinity DataIC50:  400nMAssay Description:Inhibition of HIV-1 reverse transcriptase(RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50029663(4-(3,5-Dimethyl-phenylsulfanyl)-5-ethyl-6-methyl-2...)
Affinity DataIC50:  600nMAssay Description:Inhibition of HIV-1 reverse transcriptase(RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50029679(3-Amino-5-methyl-4-m-tolylsulfanyl-1H-pyridin-2-on...)
Affinity DataIC50: >4.00E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase(RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50029671(CHEMBL126931 | N-[4-(3,5-Dimethyl-phenylsulfanyl)-...)
Affinity DataIC50: >4.00E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase(RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50029672(CHEMBL341880 | N-[4-(3,5-Dimethyl-phenylsulfanyl)-...)
Affinity DataIC50: >4.00E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase(RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50004152((HEPT) 1-(2-Hydroxy-ethoxymethyl)-5-methyl-6-pheny...)
Affinity DataIC50: >6.00E+3nMAssay Description:Inhibition of HIV-1 reverse transcriptase(RT)More data for this Ligand-Target Pair
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50029675(4-(3,5-Dimethyl-phenylsulfanyl)-5-methyl-3-nitro-1...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase(RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50029666(5-Methyl-3-nitro-4-m-tolylsulfanyl-1H-pyridin-2-on...)
Affinity DataIC50: >1.00E+4nMAssay Description:Inhibition of HIV-1 reverse transcriptase(RT)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408890(CHEMBL57301)
Affinity DataEC50:  2.40E+4nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408891(CHEMBL58891)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408892(CHEMBL418118)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408893(CHEMBL58914)
Affinity DataEC50:  2.80E+3nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408894(CHEMBL292392)
Affinity DataEC50:  4.20E+4nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408895(CHEMBL440482)
Affinity DataEC50:  1.70E+3nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408896(CHEMBL56328)
Affinity DataEC50:  800nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408897(CHEMBL262003)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM10905(3-Amino-4-(3,5-dimethylbenzyl)-5-ethyl-6-methylpyr...)
Affinity DataEC50:  17nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408899(CHEMBL300607)
Affinity DataEC50: >1.00E+5nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408900(CHEMBL417953)
Affinity DataEC50:  7.80E+3nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408901(CHEMBL60873)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50002692((AZT) 1-(4-Azido-5-hydroxymethyl-tetrahydro-furan-...)
Affinity DataEC50:  2nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408902(CHEMBL58653)
Affinity DataEC50:  2.00E+4nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408883(CHEMBL58497)
Affinity DataEC50:  3.20E+3nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408882(CHEMBL59514)
Affinity DataEC50: >1.00E+4nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50145605(4-amino-1-[(2R,5S)-5-(hydroxymethyl)tetrahydrofura...)
Affinity DataEC50:  31nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetReverse transcriptase/RNaseH(Human immunodeficiency virus 1)
Institut Curie

Curated by ChEMBL
LigandPNGBDBM50408881(CHEMBL418119)
Affinity DataEC50:  4.50E+3nMAssay Description:Effective concentration required to achieve 50% inhibition of HIV-1 LAI replication in human T4 lymphoblastoid CEM-SS cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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