Found 148 with Last Name = 'aumelas' and Initial = 'a' 
Affinity DataKi: 0.0230nMAssay Description:Binding affinity of the compound towards human cloned B1 receptor was determined using [3H]-[des-Arg10-Leu9]-kallidin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 0.110nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
Affinity DataKi: 0.120nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.130nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
Affinity DataKi: 0.160nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.180nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
Affinity DataKi: 0.240nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
Affinity DataKi: 0.300nMAssay Description:Binding affinity towards OT receptor in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.460nMAssay Description:Tested for inhibition constant determined from vasopressin induced inositol phosphates accumulation performed on WRK1 cell line of V1a receptor subty...More data for this Ligand-Target Pair
Affinity DataKi: 0.470nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:Binding affinity towards OT receptor in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
Affinity DataKi: 0.650nMAssay Description:Tested for inhibition constant at OT receptor of rat mamary glandsMore data for this Ligand-Target Pair
Affinity DataKi: 1.40nMAssay Description:Tested for inhibition constant at OT receptor of rat mamary glandsMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataKi: 2.30nMAssay Description:Binding affinity towards OT receptor in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataKi: 4.80nMAssay Description:Tested for inhibition constant at OT receptor of rat mamary glandsMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataKi: 9.16nMAssay Description:Binding affinity of the compound towards human cloned B2 receptor was determined using [3H]-BK as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataKi: 17.8nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Binding affinity towards OT receptor in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18nMAssay Description:Tested for inhibition constant at OT receptor of rat mamary glandsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Inhibition constant for V1a receptor of rat liver membraneMore data for this Ligand-Target Pair
Affinity DataKi: 24.1nMAssay Description:Binding affinity of the compound towards human cloned B1 receptor was determined using [3H]-[des-Arg10-Leu9]-kallidin as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Inhibitory activity against endopeptidase 24.15More data for this Ligand-Target Pair
Affinity DataKi: 37.7nMAssay Description:Tested for inhibition constant at OT receptor of rat mamary glandsMore data for this Ligand-Target Pair
Affinity DataKi: 40nMAssay Description:Inhibitory activity against endopeptidase 24.11More data for this Ligand-Target Pair
Affinity DataKi: 52nMAssay Description:Inhibitory activity against Leucine aminopeptidaseMore data for this Ligand-Target Pair
Affinity DataKi: 58nMAssay Description:Inhibitory activity against endopeptidase 24.16More data for this Ligand-Target Pair
Affinity DataKi: 1.32E+3nMAssay Description:Inhibitory activity against endopeptidase 24.16More data for this Ligand-Target Pair
Affinity DataKi: 1.19E+4nMAssay Description:Binding affinity of the compound towards human cloned B2 receptor was determined using [3H]-BK as radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 1.60E+4nMAssay Description:Tested for inhibition constant at V2 receptor of rat kidney membraneMore data for this Ligand-Target Pair
Affinity DataKi: 7.00E+4nMAssay Description:Inhibitory activity against angiotensin converting enzymeMore data for this Ligand-Target Pair
Affinity DataIC50: 0.200nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.290nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.300nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.320nMAssay Description:Ability to inhibit OT-induced inositol phosphate accumulation was determined in CHO cells expressing the human OT receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.5nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 0.5nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 0.600nMAssay Description:Inhibition of [125I]BH-CCK-9 binding to Cholecystokinin receptor of guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(RAT)
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 1.5nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated rat pancreatic aciniMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Inhibition of [125I]-BH-CCK- binding to cholecystokinin type B receptor from jurkat TcellsMore data for this Ligand-Target Pair
TargetCholecystokinin receptor type A/Gastrin/cholecystokinin type B receptor(Homo sapiens (Human))
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Centre De Pharmacologie-Endocrinologie (Montpellier, France)
Curated by ChEMBL
Affinity DataIC50: 2nMAssay Description:Ability of compound to Inhibit the binding of [125I]BH-CCK-8 to Cholecystokinin receptor in isolated guinea pig brain membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Tested in vitro for inhibition of amylase release from rat pancreatic aciniMore data for this Ligand-Target Pair
