Compile Data Set for Download or QSAR
maximum 50k data
Found 195 with Last Name = 'balagtas' and Initial = 'c'
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179883((4-Isopropylphenyl)-(4-isoquinolin-5-yl-phthalazin...)
Affinity DataIC50:  17nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179883((4-Isopropylphenyl)-(4-isoquinolin-5-yl-phthalazin...)
Affinity DataIC50:  17nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM21(CHEMBL24828 | N-(4-bromo-2-fluorophenyl)-6-methoxy...)
Affinity DataIC50:  45nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179881((4-Chlorophenyl)-(4-isoquinolin-5-yl-phthalazin-1-...)
Affinity DataIC50:  48nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179881((4-Chlorophenyl)-(4-isoquinolin-5-yl-phthalazin-1-...)
Affinity DataIC50:  48nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179890((4-tert-Butylphenyl)-(4-isoquinolin-5-yl-phthalazi...)
Affinity DataIC50:  75nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179890((4-tert-Butylphenyl)-(4-isoquinolin-5-yl-phthalazi...)
Affinity DataIC50:  75nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173019(4-(4-(4-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  78nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173019(4-(4-(4-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  78nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179889(CHEMBL382818 | N-(4-(chlorodifluoromethoxy)phenyl)...)
Affinity DataIC50:  79nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179889(CHEMBL382818 | N-(4-(chlorodifluoromethoxy)phenyl)...)
Affinity DataIC50:  79nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173031(4-(4-(4-bromophenylamino)phthalazin-1-yl)benzamide...)
Affinity DataIC50:  100nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173031(4-(4-(4-bromophenylamino)phthalazin-1-yl)benzamide...)
Affinity DataIC50:  100nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179888((3,4-Dichloro-phenyl)-(4-isoquinolin-5-yl-phthalaz...)
Affinity DataIC50:  110nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179888((3,4-Dichloro-phenyl)-(4-isoquinolin-5-yl-phthalaz...)
Affinity DataIC50:  110nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179891((4-Chloro-3-trifluoromethylphenyl)-(4-isoquinolin-...)
Affinity DataIC50:  120nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179891((4-Chloro-3-trifluoromethylphenyl)-(4-isoquinolin-...)
Affinity DataIC50:  120nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173045(4-(4-(4-tert-butylphenylamino)phthalazin-1-yl)-N-m...)
Affinity DataIC50:  130nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173045(4-(4-(4-tert-butylphenylamino)phthalazin-1-yl)-N-m...)
Affinity DataIC50:  130nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192487((7,8-dimethoxy-10,11-dihydro-5H-2,4,5,11-tetraaza-...)
Affinity DataIC50:  150nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173049(4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthala...)
Affinity DataIC50:  190nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173049(4-(4-(4-(chlorodifluoromethoxy)phenylamino)phthala...)
Affinity DataIC50:  190nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192474(CHEMBL215191 | benzyl-(7,8-dimethoxy-10,11-dihydro...)
Affinity DataIC50:  200nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179893((4-Isoquinolin-5-yl-phthalazin-1-yl)-(2-methyl-1Hi...)
Affinity DataIC50:  230nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179893((4-Isoquinolin-5-yl-phthalazin-1-yl)-(2-methyl-1Hi...)
Affinity DataIC50:  230nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179884((4-Isoquinolin-5-yl-phthalazin-1-yl)-m-tolylamine ...)
Affinity DataIC50:  270nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179884((4-Isoquinolin-5-yl-phthalazin-1-yl)-m-tolylamine ...)
Affinity DataIC50:  270nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192498((3-chloro-4-fluoro-benzyl)-(7,8-dimethoxy-10,11-di...)
Affinity DataIC50:  300nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50180448((3-Bromo-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-ox...)
Affinity DataIC50:  300nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192477((3-chloro-2-fluoro-phenyl)-(7,8-dimethoxy-10,11-di...)
Affinity DataIC50:  300nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173007(4-[4-(4-Chloro-phenylamino)-phthalazin-1-yl]-benzo...)
Affinity DataIC50:  360nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179894((4-Isoquinolin-5-yl-phthalazin-1-yl)-(4-morpholin-...)
Affinity DataIC50:  390nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179894((4-Isoquinolin-5-yl-phthalazin-1-yl)-(4-morpholin-...)
Affinity DataIC50:  390nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173022(3-(4-(4-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  400nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173022(3-(4-(4-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  400nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179882((2-Fluoro-4-methylphenyl)-(4-isoquinolin-5-ylphtha...)
Affinity DataIC50:  430nMAssay Description:Inhibition of VEGFR2 by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50179882((2-Fluoro-4-methylphenyl)-(4-isoquinolin-5-ylphtha...)
Affinity DataIC50:  430nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173034(4-(4-(3-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  470nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173034(4-(4-(3-tert-butylphenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  470nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192471((7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-d...)
Affinity DataIC50:  500nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192487((7,8-dimethoxy-10,11-dihydro-5H-2,4,5,11-tetraaza-...)
Affinity DataIC50:  500nMAssay Description:Inhibition of EGFR autophosphorylation in DiFi cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50180448((3-Bromo-phenyl)-(7,8-dimethoxy-10,11-dihydro-5-ox...)
Affinity DataIC50:  500nMAssay Description:Inhibition of EGFR autophosphorylation in DiFi cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173021(4-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-pht...)
Affinity DataIC50:  630nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173021(4-{4-[4-(Chloro-difluoro-methoxy)-phenylamino]-pht...)
Affinity DataIC50:  630nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50180453((3-Chloro-4-fluoro-phenyl)-(7,8-dimethoxy-10,11-di...)
Affinity DataIC50:  700nMAssay Description:Inhibition of EGFR autophosphorylation in DiFi cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192478(1-(3-bromo-phenoxy)-7,8-dimethoxy-10,11-dihydro-5-...)
Affinity DataIC50:  700nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192497((7,8-dimethoxy-10,11-dihydro-5H-2,4,5,11-tetraaza-...)
Affinity DataIC50:  800nMAssay Description:Inhibition of EGFR measured as pGAT-biotin peptide phosphorylation in presence of 2.0 uM ATP by HTRF assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173051(4-(4-(3,4-dichlorophenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  840nMAssay Description:Inhibition of Vascular endothelial growth factor receptor 2 kinase phosphorylation of pGAT-biotin peptideMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50173051(4-(4-(3,4-dichlorophenylamino)phthalazin-1-yl)benz...)
Affinity DataIC50:  840nMAssay Description:Inhibition of VEGFR2 (unknown origin) by HTRF methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Imclone Systems

Curated by ChEMBL
LigandPNGBDBM50192501((7,8-dimethoxy-10,11-dihydro-5-oxa-2,4,11-triaza-d...)
Affinity DataIC50:  900nMAssay Description:Inhibition of EGFR autophosphorylation in DiFi cells by ELISAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Displayed 1 to 50 (of 195 total ) | Next | Last >>
Jump to: