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Found 17 with Last Name = 'bannwarth' and Initial = 'l'
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  100nMAssay Description:Inhibition of dimerization of HIV1 protease 150V mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  200nMAssay Description:Inhibition of dimerization of HIV1 protease ANAM-11 mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191464(CHEMBL212749 | methyl (2S)-2-[(2S)-2-[(2S)-2-(4-{[...)
Affinity DataKi:  200nMAssay Description:Inhibition of wild type HIV1 protease dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  240nMAssay Description:Inhibition of dimerization of HIV1 protease V82A mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  400nMAssay Description:Inhibition of wild type HIV1 protease dimerizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  500nMAssay Description:Inhibition of dimerization of HIV1 protease D30N mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  500nMAssay Description:Inhibition of dimerization of HIV1 protease G48V/L90M mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191463(CHEMBL378467 | methyl (2S)-2-[(2R)-2-[(2S)-2-{4-[(...)
Affinity DataKi:  4.80E+3nMAssay Description:Inhibition of dimerization of HIV1 protease MDR-HM mutantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191465(CHEMBL386205 | methyl (2S)-2-[(2R)-2-[(2S)-2-[4-({...)
Affinity DataKi:  8.40E+3nMAssay Description:Inhibition of wild type HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGag-Pol polyprotein [489-587](Human immunodeficiency virus type 1)
Paris-Sud University

Curated by ChEMBL
LigandPNGBDBM50191466(CHEMBL426149 | methyl (2S)-2-[(2R)-2-[(2S)-2-(4-{[...)
Affinity DataKi:  9.70E+3nMAssay Description:Inhibition of wild type HIV1 proteaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 6(Homo sapiens (Human))
Yale University School of Medicine

LigandPNGBDBM50056922(1,4-Dihydroxy-10-methoxy-5,8-dimethyl-3,7-dioxo-1,...)
Affinity DataIC50:  2.40E+4nMAssay Description:The labeled fragment can be distinguished from full-length MKK by a change in fluorescence polarization. MKK6 was used as a substrate because it cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 6(Homo sapiens (Human))
Yale University School of Medicine

LigandPNGBDBM29673(1,4,10-Trihydroxy-5-hydroxymethyl-8-methyl-3,7-dio...)
Affinity DataIC50:  4.20E+4nMAssay Description:The labeled fragment can be distinguished from full-length MKK by a change in fluorescence polarization. MKK6 was used as a substrate because it cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 6(Homo sapiens (Human))
Yale University School of Medicine

LigandPNGBDBM50056939(4-Formyl-3-hydroxy-8-methoxy-1,9-dimethyl-11-oxo-1...)
Affinity DataIC50:  1.25E+5nMAssay Description:The labeled fragment can be distinguished from full-length MKK by a change in fluorescence polarization. MKK6 was used as a substrate because it cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 6(Homo sapiens (Human))
Yale University School of Medicine

LigandPNGBDBM29678(Reduced parellic acid, 9)
Affinity DataIC50: >2.50E+5nMAssay Description:The labeled fragment can be distinguished from full-length MKK by a change in fluorescence polarization. MKK6 was used as a substrate because it cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 6(Homo sapiens (Human))
Yale University School of Medicine

LigandPNGBDBM29674(Reduced stictic acid, 8)
Affinity DataIC50: >2.50E+5nMAssay Description:The labeled fragment can be distinguished from full-length MKK by a change in fluorescence polarization. MKK6 was used as a substrate because it cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 6(Homo sapiens (Human))
Yale University School of Medicine

LigandPNGBDBM50056904(3,8-Dihydroxy-11-oxo-1-(2-oxo-heptyl)-6-pentyl-11H...)
Affinity DataIC50: >2.50E+5nMAssay Description:The labeled fragment can be distinguished from full-length MKK by a change in fluorescence polarization. MKK6 was used as a substrate because it cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDual specificity mitogen-activated protein kinase kinase 6(Homo sapiens (Human))
Yale University School of Medicine

LigandPNGBDBM92359(Gangleoidin, 4)
Affinity DataIC50: >2.50E+5nMAssay Description:The labeled fragment can be distinguished from full-length MKK by a change in fluorescence polarization. MKK6 was used as a substrate because it cou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed