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Found 54 with Last Name = 'barbe' and Initial = 'b'
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50407297(CHEMBL2052008)
Affinity DataKi:  0.700nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50407297(CHEMBL2052008)
Affinity DataKi:  0.700nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50407299(CHEMBL2052007)
Affinity DataKi:  1.60nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50407299(CHEMBL2052007)
Affinity DataKi:  1.60nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50407299(CHEMBL2052007)
Affinity DataKi:  1.90nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50407299(CHEMBL2052007)
Affinity DataKi:  1.90nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50407298(CHEMBL2051772)
Affinity DataKi:  5.30nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50407298(CHEMBL2051772)
Affinity DataKi:  10nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50407297(CHEMBL2052008)
Affinity DataKi:  16nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50407297(CHEMBL2052008)
Affinity DataKi:  80nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041071((2-Mercaptomethyl-3-phenyl-butyrylamino)-acetic ac...)
Affinity DataIC50:  1.30nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041067(2-[3-(4-Fluoro-phenyl)-2-mercaptomethyl-butyrylami...)
Affinity DataIC50:  2nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50407297(CHEMBL2052008)
Affinity DataIC50:  2nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041069(3-(4-Hydroxy-phenyl)-2-(2-mercaptomethyl-3-phenyl-...)
Affinity DataIC50:  2nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041058(2-(3-Benzo[1,3]dioxol-5-yl-2-mercaptomethyl-butyry...)
Affinity DataIC50:  2nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041070(3-(4-Hydroxy-phenyl)-2-(2-mercaptomethyl-3-phenyl-...)
Affinity DataIC50:  2.40nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041062(3-(4-Hydroxy-phenyl)-2-[2-mercaptomethyl-3-(4-meth...)
Affinity DataIC50:  2.5nMAssay Description:In vivo inhibitory potency against Neutral Endopeptidase by measuring the displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041054(3-(4-Hydroxy-phenyl)-2-(2-mercaptomethyl-3-phenyl-...)
Affinity DataIC50:  2.5nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041061(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-hexanoi...)
Affinity DataIC50:  3.10nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041053(2-[3-(3,4-Difluoro-phenyl)-2-mercaptomethyl-butyry...)
Affinity DataIC50:  3.5nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041059(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-4-methy...)
Affinity DataIC50:  3.5nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041062(3-(4-Hydroxy-phenyl)-2-[2-mercaptomethyl-3-(4-meth...)
Affinity DataIC50:  3.60nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041063(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-pentano...)
Affinity DataIC50:  4nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041060(2-[3-(3,4-Dimethoxy-phenyl)-2-mercaptomethyl-butyr...)
Affinity DataIC50:  4nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041063(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-pentano...)
Affinity DataIC50:  4nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041066(3-Benzyloxy-2-(2-mercaptomethyl-3-phenyl-butyrylam...)
Affinity DataIC50:  4nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041054(3-(4-Hydroxy-phenyl)-2-(2-mercaptomethyl-3-phenyl-...)
Affinity DataIC50:  4.30nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041057(2-[3-(3,4-Difluoro-phenyl)-2-mercaptomethyl-butyry...)
Affinity DataIC50:  4.5nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041053(2-[3-(3,4-Difluoro-phenyl)-2-mercaptomethyl-butyry...)
Affinity DataIC50:  5nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041057(2-[3-(3,4-Difluoro-phenyl)-2-mercaptomethyl-butyry...)
Affinity DataIC50:  5.20nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041052(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-butyric...)
Affinity DataIC50:  5.40nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041064(2-[3-(4-Fluoro-phenyl)-2-mercaptomethyl-butyrylami...)
Affinity DataIC50:  5.90nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041052(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-butyric...)
Affinity DataIC50:  6.30nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041064(2-[3-(4-Fluoro-phenyl)-2-mercaptomethyl-butyrylami...)
Affinity DataIC50:  6.90nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041061(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-hexanoi...)
Affinity DataIC50:  7nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041068(3-(4-Hydroxy-phenyl)-2-[3-(4-hydroxy-phenyl)-2-mer...)
Affinity DataIC50:  7.90nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041068(3-(4-Hydroxy-phenyl)-2-[3-(4-hydroxy-phenyl)-2-mer...)
Affinity DataIC50:  9nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041058(2-(3-Benzo[1,3]dioxol-5-yl-2-mercaptomethyl-butyry...)
Affinity DataIC50:  9.5nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041067(2-[3-(4-Fluoro-phenyl)-2-mercaptomethyl-butyrylami...)
Affinity DataIC50:  10nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041050(3-(4-Hydroxy-phenyl)-2-(2-mercaptomethyl-3-o-tolyl...)
Affinity DataIC50:  11nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041055(2-[3-(4-Amino-phenyl)-2-mercaptomethyl-butyrylamin...)
Affinity DataIC50:  12nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041051(2-[3-(4-Hydroxy-3-methoxy-phenyl)-2-mercaptomethyl...)
Affinity DataIC50:  14nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041065(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-3-methy...)
Affinity DataIC50:  15nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041060(2-[3-(3,4-Dimethoxy-phenyl)-2-mercaptomethyl-butyr...)
Affinity DataIC50:  16nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeprilysin(Homo sapiens (Human))
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041055(2-[3-(4-Amino-phenyl)-2-mercaptomethyl-butyrylamin...)
Affinity DataIC50:  16nMAssay Description:In vivo inhibitory potency against neutral endopeptidase by displacement of [3H]-HACBOGly binding in mouse kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041059(2-(2-Mercaptomethyl-3-phenyl-butyrylamino)-4-methy...)
Affinity DataIC50:  19nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50407297(CHEMBL2052008)
Affinity DataIC50:  20nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041069(3-(4-Hydroxy-phenyl)-2-(2-mercaptomethyl-3-phenyl-...)
Affinity DataIC50:  25nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041071((2-Mercaptomethyl-3-phenyl-butyrylamino)-acetic ac...)
Affinity DataIC50:  32nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAngiotensin-converting enzyme(Mus musculus)
University Of Paris

Curated by ChEMBL
LigandPNGBDBM50041066(3-Benzyloxy-2-(2-mercaptomethyl-3-phenyl-butyrylam...)
Affinity DataIC50:  43nMAssay Description:Inhibitory potency against angiotensin converting enzyme by displacement of [3H]-trandolaprilate binding in mouse lungMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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