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Found 28 with Last Name = 'bartenschlager' and Initial = 'r'
TargetFurin(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552678(CHEMBL4759036)
Affinity DataKi:  0.00500nMAssay Description:Inhibition of recombinant soluble human furin using Phac-Arg-Val-Arg-Arg-AMC fluorogenic substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552679(CHEMBL4762678)
Affinity DataKi:  0.00900nMAssay Description:Inhibition of recombinant soluble human furin using Phac-Arg-Val-Arg-Arg-AMC fluorogenic substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552672(CHEMBL4790628)
Affinity DataKi:  0.0100nMAssay Description:Inhibition of recombinant soluble human furin using Phac-Arg-Val-Arg-Arg-AMC fluorogenic substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552676(CHEMBL4794635)
Affinity DataKi:  0.0130nMAssay Description:Inhibition of recombinant soluble human furin using Phac-Arg-Val-Arg-Arg-AMC fluorogenic substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552673(CHEMBL4750900)
Affinity DataKi:  0.0340nMAssay Description:Inhibition of recombinant soluble human furin using Phac-Arg-Val-Arg-Arg-AMC fluorogenic substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552674(CHEMBL4742184)
Affinity DataKi:  0.0360nMAssay Description:Inhibition of recombinant soluble human furin using Phac-Arg-Val-Arg-Arg-AMC fluorogenic substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552677(CHEMBL4779067)
Affinity DataKi:  0.0770nMAssay Description:Inhibition of recombinant soluble human furin using Phac-Arg-Val-Arg-Arg-AMC fluorogenic substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFurin(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552675(CHEMBL4747919)
Affinity DataKi:  0.114nMAssay Description:Inhibition of recombinant soluble human furin using Phac-Arg-Val-Arg-Arg-AMC fluorogenic substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50587014(CHEMBL5094815)
Affinity DataKi:  79nMAssay Description:Competitive inhibition of C-terminal His-tagged ZIKV NSB2 (52 to 96 amino acids)-NS3 (1 to 184 amino acids) protease expressed in Escherichia coli BL...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50587014(CHEMBL5094815)
Affinity DataKi:  343nMAssay Description:Competitive inhibition of C-terminal His-tagged WNV NSB2 (52 to 96 amino acids)-NS3 (1 to 184 amino acids) protease expressed in Escherichia coli BL2...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552678(CHEMBL4759036)
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition pf human plasmin using Mes-Darg-Phe-Arg-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlasminogen(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552672(CHEMBL4790628)
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition pf human plasmin using Mes-Darg-Phe-Arg-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552678(CHEMBL4759036)
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of human factor Xa using Mes-Darg-Pro-Arg-AMC as flurogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552672(CHEMBL4790628)
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of human factor Xa using Mes-Darg-Pro-Arg-AMC as flurogenic substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552672(CHEMBL4790628)
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Bos taurus (Bovine))
Philipps University

Curated by ChEMBL
LigandPNGBDBM50552678(CHEMBL4759036)
Affinity DataKi: >3.00E+3nMAssay Description:Inhibition of bovine thrombin using Tos-Gly-Pro-Arg-AMC as substrate by fluorescence assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50587014(CHEMBL5094815)
Affinity DataKi:  1.27E+4nMAssay Description:Competitive inhibition of recombinant N-terminal His-tagged DENV NS2B-NS3 protease expressed in Escherichia coli BL21(DE3) using Boc-GRR-AMC as subst...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetNonstructural protein 3(Zika virus)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50587014(CHEMBL5094815)
Affinity DataIC50:  125nMAssay Description:Inhibition of C-terminal His-tagged ZIKV NSB2 (52 to 96 amino acids)-NS3 (1 to 184 amino acids) protease expressed in Escherichia coli BL21(DE3) prei...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50587014(CHEMBL5094815)
Affinity DataIC50:  460nMAssay Description:Inhibition of C-terminal His-tagged WNV NSB2 (52 to 96 amino acids)-NS3 (1 to 184 amino acids) protease expressed in Escherichia coli BL21(DE3) using...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50127623(CHEMBL3628260)
Affinity DataIC50:  1.60E+3nMAssay Description:Inhibition of West Nile virus NS2B-NS3 protease preincubated with protein for 15 mins followed by Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)-Tyr substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50127569(CHEMBL3628271)
Affinity DataIC50:  2.48E+3nMAssay Description:Inhibition of West Nile virus NS2B-NS3 protease preincubated with protein for 15 mins followed by Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)-Tyr substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(West Nile virus)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50127568(CHEMBL3628265)
Affinity DataIC50:  3.85E+3nMAssay Description:Inhibition of West Nile virus NS2B-NS3 protease preincubated with protein for 15 mins followed by Abz-Gly-Leu-Lys-Arg-Gly-Gly-3-(NO2)-Tyr substrate a...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50127570(CHEMBL3628279)
Affinity DataIC50:  4.59E+3nMAssay Description:Inhibition of human thrombin preincubated with protein for 15 mins followed by boc-Val-Pro-Arg-AMC substrate addition measured after 10 mins by conti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50517071(CHEMBL4569882)
Affinity DataIC50:  6.30E+3nMAssay Description:Inhibition of Dengue virus NS2B-NS3 protease using FRET Abz-Nle-Lys-Arg-Arg-Ser-3-(NO2)Tyr as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50127571(CHEMBL3628272)
Affinity DataIC50:  7.10E+3nMAssay Description:Inhibition of trypsin (unknown origin) preincubated with protein for 15 mins followed by boc-Val-Pro-Arg-AMC substrate addition measured by continuou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50587014(CHEMBL5094815)
Affinity DataIC50:  1.71E+4nMAssay Description:Inhibition of recombinant N-terminal His-tagged DENV NS2B-NS3 protease expressed in Escherichia coli BL21(DE3) using Boc-GRR-AMC as substrate measure...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetTrypsin(Homo sapiens (Human))
Heidelberg University

Curated by ChEMBL
LigandPNGBDBM50127569(CHEMBL3628271)
Affinity DataIC50:  1.82E+4nMAssay Description:Inhibition of trypsin (unknown origin) preincubated with protein for 15 mins followed by boc-Val-Pro-Arg-AMC substrate addition measured by continuou...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGenome polyprotein(Dengue virus 2)
Freie Universit£T Berlin

Curated by ChEMBL
LigandPNGBDBM50517070(CHEMBL4518162)
Affinity DataIC50:  2.50E+4nMAssay Description:Inhibition of Dengue virus serotype 2 NS2B-NS3 protease expressed in Escherichia coli BL21 lambda (DE3) cells preincubated with enzyme for 15 mins fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed