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Found 303 with Last Name = 'bell' and Initial = 'mr'
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039635(2,6-Dichloro-3-(4-methyl-piperazine-1-sulfonyl)-be...)
Affinity DataKi:  0.00700nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50036480(2,6-Dichloro-3-(2-morpholin-4-yl-ethoxy)-benzoic a...)
Affinity DataKi:  0.00800nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039646(2,6-Dichloro-3-(2-morpholin-4-yl-ethoxy)-benzoic a...)
Affinity DataKi:  0.00800nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039637(2,6-Dichloro-3-[(2-dimethylamino-ethyl)-methyl-sul...)
Affinity DataKi:  0.0100nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50036478(3-Carboxymethoxy-2,6-dichloro-benzoic acid 4-isopr...)
Affinity DataKi:  0.0110nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50036476(2,6-Dichloro-3-(4-methyl-piperazine-1-sulfonyl)-be...)
Affinity DataKi:  0.0110nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50036481(2,6-Dichloro-3-[(2-dimethylamino-ethyl)-methyl-sul...)
Affinity DataKi:  0.0130nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50036477(2,6-Dichloro-3-(2-morpholin-4-yl-ethoxy)-benzoic a...)
Affinity DataKi:  0.0130nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50036475(2,6-Dichloro-3-(2-pyrrolidin-1-yl-ethoxy)-benzoic ...)
Affinity DataKi:  0.0140nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50029699(2,6-Dichloro-benzoic acid 4-isopropyl-6-methoxy-1,...)
Affinity DataKi:  0.0230nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039631(2,6-Dichloro-benzoic acid 4-isopropyl-1,1,3-trioxo...)
Affinity DataKi:  0.0300nMAssay Description:Ratio of Kreact to that of Kinact was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039631(2,6-Dichloro-benzoic acid 4-isopropyl-1,1,3-trioxo...)
Affinity DataKi:  0.0300nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286326(2,6-Dichloro-benzoic acid 6-fluoro-4-isopropyl-1,1...)
Affinity DataKi:  0.0300nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039631(2,6-Dichloro-benzoic acid 4-isopropyl-1,1,3-trioxo...)
Affinity DataKi:  0.0300nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039631(2,6-Dichloro-benzoic acid 4-isopropyl-1,1,3-trioxo...)
Affinity DataKi:  0.0302nMAssay Description:Observed binding affinity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039641(2,6-Dichloro-benzoic acid 4-sec-butyl-1,1,3-trioxo...)
Affinity DataKi:  0.0600nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039642(2,6-Dichloro-benzoic acid 4-ethyl-1,1,3-trioxo-1,3...)
Affinity DataKi:  0.0708nMAssay Description:Observed binding affinity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039642(2,6-Dichloro-benzoic acid 4-ethyl-1,1,3-trioxo-1,3...)
Affinity DataKi:  0.170nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50036482(2,6-Dichloro-3-(4-methyl-piperazine-1-sulfonyl)-be...)
Affinity DataKi:  0.200nMAssay Description:Potency of inhibition against human leukocyte elastase (HLE) expressed as an apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286333(5,6-Dimethoxy-1,1-dioxo-2-(1-phenyl-1H-tetrazol-5-...)
Affinity DataKi:  0.200nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50029703(4-Isopropyl-6-methoxy-1,1-dioxo-2-(1-phenyl-1H-tet...)
Affinity DataKi:  0.270nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50282874(4-Isopropyl-1,1-dioxo-2-(1-phenyl-1H-tetrazol-5-yl...)
Affinity DataKi:  0.300nMAssay Description:Potency of Inhibition of human leukocyte elastase (HLE) expressed as apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50282874(4-Isopropyl-1,1-dioxo-2-(1-phenyl-1H-tetrazol-5-yl...)
Affinity DataKi:  0.300nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50005147((S)-1-{(S)-2-[4-(4-Bromo-benzenesulfonylaminocarbo...)
Affinity DataKi:  0.400nMAssay Description:Potency of Inhibition of human leukocyte elastase (HLE) expressed as apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50005147((S)-1-{(S)-2-[4-(4-Bromo-benzenesulfonylaminocarbo...)
Affinity DataKi:  0.400nMAssay Description:Ratio of Kreact to that of Kinact was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50005147((S)-1-{(S)-2-[4-(4-Bromo-benzenesulfonylaminocarbo...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity for human leukocyte elastase (HLE); Kreact/KinactMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286327(4,6-Dimethoxy-1,1-dioxo-2-(1-phenyl-1H-tetrazol-5-...)
Affinity DataKi:  0.600nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50282873(4-sec-Butyl-1,1-dioxo-2-(1-phenyl-1H-tetrazol-5-yl...)
Affinity DataKi:  0.600nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50282873(4-sec-Butyl-1,1-dioxo-2-(1-phenyl-1H-tetrazol-5-yl...)
Affinity DataKi:  0.600nMAssay Description:Potency of Inhibition of human leukocyte elastase (HLE) expressed as apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50282868(1,1-Dioxo-2-(1-phenyl-1H-tetrazol-5-ylsulfanylmeth...)
Affinity DataKi:  0.700nMAssay Description:Potency of Inhibition of human leukocyte elastase (HLE) expressed as apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50282868(1,1-Dioxo-2-(1-phenyl-1H-tetrazol-5-ylsulfanylmeth...)
Affinity DataKi:  0.700nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286322(2,6-Dichloro-benzoic acid 4-ethyl-1,1,3-trioxo-1,3...)
Affinity DataKi:  0.700nMAssay Description:Ratio of Kreact to that of Kinact was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286322(2,6-Dichloro-benzoic acid 4-ethyl-1,1,3-trioxo-1,3...)
Affinity DataKi:  0.708nMAssay Description:Observed binding affinity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286305(2-[2-Chloro-4-(morpholine-4-sulfonyl)-phenoxymethy...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity for human leukocyte elastase (HLE); Kreact/KinactMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286324(2,6-Dichloro-benzoic acid 3,3,5-trioxo-3lambda*6*-...)
Affinity DataKi:  0.800nMAssay Description:Ratio of Kreact to that of Kinact was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039634(2,6-Dichloro-benzoic acid 1,1,3-trioxo-4-phenyl-1,...)
Affinity DataKi:  1nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286320(2,6-Dichloro-benzoic acid 4-isopropyl-1,1,3-trioxo...)
Affinity DataKi:  1nMAssay Description:Observed binding affinity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286320(2,6-Dichloro-benzoic acid 4-isopropyl-1,1,3-trioxo...)
Affinity DataKi:  1nMAssay Description:Ratio of Kreact to that of Kinact was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286321(2,6-Dichloro-benzoic acid 4,4-dimethyl-1,1,3-triox...)
Affinity DataKi:  1nMAssay Description:Ratio of Kreact to that of Kinact was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286323(2,6-Dichloro-benzoic acid 4-methyl-1,1,3-trioxo-1,...)
Affinity DataKi:  1nMAssay Description:Ratio of Kreact to that of Kinact was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286323(2,6-Dichloro-benzoic acid 4-methyl-1,1,3-trioxo-1,...)
Affinity DataKi:  1nMAssay Description:Ratio of Kreact to that of Kinact was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286329(2,6-Dichloro-benzoic acid 4-isopropyl-6-(4-methyl-...)
Affinity DataKi:  1.10nMAssay Description:Evaluated for inhibitory activity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286307(2,6-Dichloro-4-(4-isopropyl-1,1,3-trioxo-1,3-dihyd...)
Affinity DataKi:  1.60nMAssay Description:Binding affinity for human leukocyte elastase (HLE); Kreact/KinactMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50282865(2-Chloromethyl-1,1-dioxo-1,2-dihydro-1lambda*6*-be...)
Affinity DataKi:  1.80nMAssay Description:Potency of Inhibition of human leukocyte elastase (HLE) expressed as apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50282866(4-Ethyl-1,1-dioxo-2-(1-phenyl-1H-tetrazol-5-ylsulf...)
Affinity DataKi:  2nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50282866(4-Ethyl-1,1-dioxo-2-(1-phenyl-1H-tetrazol-5-ylsulf...)
Affinity DataKi:  2nMAssay Description:Potency of Inhibition of human leukocyte elastase (HLE) expressed as apparent binding constantMore data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039644(2,6-Dichloro-benzoic acid 4-methyl-1,1,3-trioxo-1,...)
Affinity DataKi:  2nMAssay Description:In vitro inhibition constant of human leukocyte elastase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039636(2,6-Dichloro-benzoic acid 1,1,3-trioxo-1,3-dihydro...)
Affinity DataKi:  2nMAssay Description:Observed binding affinity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50286330(4,5-Dimethoxy-1,1-dioxo-2-(1-phenyl-1H-tetrazol-5-...)
Affinity DataKi:  2nMAssay Description:Ratio of Koff to that of Kon was determined on human leukocyte elastase(HLE)More data for this Ligand-Target Pair
In DepthDetails Article
TargetNeutrophil elastase(Homo sapiens (Human))
Sterling Winthrop Pharmaceutical Research Division

Curated by ChEMBL
LigandPNGBDBM50039644(2,6-Dichloro-benzoic acid 4-methyl-1,1,3-trioxo-1,...)
Affinity DataKi:  2nMAssay Description:Observed binding affinity against Human leukocyte elastase (HLE)More data for this Ligand-Target Pair
In DepthDetails Article
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