Affinity DataKi: 10nMAssay Description:Binding affinity at Metabotropic glutamate receptor 1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
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Curated by ChEMBL
Affinity DataKi: 13nMAssay Description:Binding affinity at Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
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Curated by ChEMBL
Affinity DataKi: 110nMAssay Description:Binding affinity at Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
Affinity DataKi: 340nMAssay Description:Binding affinity at Metabotropic glutamate receptor 1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
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Curated by ChEMBL
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Curated by ChEMBL
Affinity DataKi: 470nMAssay Description:Binding affinity at Metabotropic glutamate receptor 4More data for this Ligand-Target Pair
Affinity DataKi: 900nMAssay Description:Binding affinity at Metabotropic glutamate receptor 1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
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Curated by ChEMBL
Affinity DataKi: 1.20E+3nMAssay Description:Binding affinity at Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
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Curated by ChEMBL
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Curated by ChEMBL
Affinity DataKi: 1.60E+3nMAssay Description:Binding affinity at Metabotropic glutamate receptor 4More data for this Ligand-Target Pair
Affinity DataKi: 3.70E+3nMAssay Description:Binding affinity at Metabotropic glutamate receptor 1More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
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Curated by ChEMBL
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Curated by ChEMBL
Affinity DataKi: 1.12E+5nMAssay Description:Binding affinity at Metabotropic glutamate receptor 4More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
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Curated by ChEMBL
Affinity DataKi: 1.13E+5nMAssay Description:Binding affinity at Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
Parc Club Orsay Universit£
Curated by ChEMBL
Affinity DataKi: 1.29E+5nMAssay Description:Binding affinity at Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 4(Homo sapiens (Human))
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Curated by ChEMBL
Parc Club Orsay Universit£
Curated by ChEMBL
Affinity DataKi: 8.38E+5nMAssay Description:Binding affinity at Metabotropic glutamate receptor 4More data for this Ligand-Target Pair
TargetMetabotropic glutamate receptor 2(Homo sapiens (Human))
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Curated by ChEMBL
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Curated by ChEMBL
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity at Metabotropic glutamate receptor 2More data for this Ligand-Target Pair
Affinity DataKi: >1.00E+6nMAssay Description:Binding affinity at Metabotropic glutamate receptor 1More data for this Ligand-Target Pair
Affinity DataEC50: 3.00E+3nMAssay Description:Agonist activity in rat at Metabotropic glutamate receptor 1 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.61E+5nMAssay Description:Agonist activity in rat at mGlu2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 8.00E+3nMAssay Description:Agonist activity in rat at Metabotropic glutamate receptor 8 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.37E+5nMAssay Description:Agonist activity in rat at mGlu2 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 5.30E+4nMAssay Description:Agonist activity in rat at mGlu8a receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 6.90E+4nMAssay Description:Agonist activity in rat at mGlu8a receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.60E+4nMAssay Description:Agonist activity in rat at Metabotropic glutamate receptor 2 expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 3.73E+5nMAssay Description:Agonist activity in rat at mGlu1a receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 1.10E+4nMAssay Description:Agonist activity in rat at mGlu1a receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair