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Found 69 with Last Name = 'bittman' and Initial = 'r'
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50064519(3-[(3R,4R)-3,4-Dimethyl-1-((S)-2-phenyl-cyclopropy...)
Affinity DataKi:  1.80nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336606(3-((1S,5R)-2-Cinnamyl-2-azabicyclo[3.3.1]nonan-5-y...)
Affinity DataKi:  2nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336611(3-((1R,5S)-2-(((1'S,2'S)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  3nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336603(3-((1R,5S)-2-(((1'R,2'R)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  4nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336607(3-((1R,5S)-2-Cinnamyl-2-azabicyclo[3.3.1]nonan-5-y...)
Affinity DataKi:  6nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336613(3-((1R,5S)-2-(((1'R,2'S)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  11nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336609(3-((1R,5S)-2-((Z)-3-phenylallyl)-2-azabicyclo[3.3....)
Affinity DataKi:  14nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336602(3-((1S,5R)-2-(((1'S,2'S)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  16nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336608(3-((1S,5R)-2-((Z)-3-phenylallyl)-2-azabicyclo[3.3....)
Affinity DataKi:  26nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336610(3-((1S,5R)-2-(((1'R,2'R)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  47nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336611(3-((1R,5S)-2-(((1'S,2'S)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  72nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336612(3-((1S,5R)-2-(((1'S,2'R)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  76nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336608(3-((1S,5R)-2-((Z)-3-phenylallyl)-2-azabicyclo[3.3....)
Affinity DataKi:  123nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336606(3-((1S,5R)-2-Cinnamyl-2-azabicyclo[3.3.1]nonan-5-y...)
Affinity DataKi:  125nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336606(3-((1S,5R)-2-Cinnamyl-2-azabicyclo[3.3.1]nonan-5-y...)
Affinity DataKi:  138nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336607(3-((1R,5S)-2-Cinnamyl-2-azabicyclo[3.3.1]nonan-5-y...)
Affinity DataKi:  152nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336604(3-((1S,5R)-2-(((1'R,2'S)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  153nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336611(3-((1R,5S)-2-(((1'S,2'S)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  165nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336612(3-((1S,5R)-2-(((1'S,2'R)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  174nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336602(3-((1S,5R)-2-(((1'S,2'S)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  183nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336613(3-((1R,5S)-2-(((1'R,2'S)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  196nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336603(3-((1R,5S)-2-(((1'R,2'R)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  200nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336603(3-((1R,5S)-2-(((1'R,2'R)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  210nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336607(3-((1R,5S)-2-Cinnamyl-2-azabicyclo[3.3.1]nonan-5-y...)
Affinity DataKi:  225nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336604(3-((1S,5R)-2-(((1'R,2'S)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  265nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336613(3-((1R,5S)-2-(((1'R,2'S)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  322nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336602(3-((1S,5R)-2-(((1'S,2'S)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  323nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336609(3-((1R,5S)-2-((Z)-3-phenylallyl)-2-azabicyclo[3.3....)
Affinity DataKi:  359nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336609(3-((1R,5S)-2-((Z)-3-phenylallyl)-2-azabicyclo[3.3....)
Affinity DataKi:  367nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336610(3-((1S,5R)-2-(((1'R,2'R)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  390nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336608(3-((1S,5R)-2-((Z)-3-phenylallyl)-2-azabicyclo[3.3....)
Affinity DataKi:  454nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMu-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336605(3-((1R,5S)-2-(((1'S,2'R)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  459nMAssay Description:Displacement of [125I]IOXY from human recombinant mu opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKappa-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336605(3-((1R,5S)-2-(((1'S,2'R)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  475nMAssay Description:Displacement of [125I]IOXY from human recombinant kappa opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336612(3-((1S,5R)-2-(((1'S,2'R)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  547nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336604(3-((1S,5R)-2-(((1'R,2'S)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  610nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336610(3-((1S,5R)-2-(((1'R,2'R)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  800nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443388(CHEMBL3086782 | US9688668, SLR080811)
Affinity DataKi:  1.00E+3nMAssay Description:Inhibition of sphingosine kinase 1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDelta-type opioid receptor(Homo sapiens (Human))
National Institute On Drug Abuse

Curated by ChEMBL
LigandPNGBDBM50336605(3-((1R,5S)-2-(((1'S,2'R)-2-Phenylcyclopropyl)methy...)
Affinity DataKi:  1.98E+3nMAssay Description:Displacement of [125I]IOXY from human recombinant delta opioid receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443385(SPC-100270 | Safingol | Safingol HCl)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of sphingosine kinase 1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50004888((S)-Fingolimod Vinylphosphonate | CHEMBL1773676)
Affinity DataKi:  1.00E+4nMAssay Description:Competitive inhibition of SK1 (unknown origin) in presence of ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443389(CHEMBL2376441)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of sphingosine kinase 1 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50393642(CHEMBL2158685)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of SK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50393641(CHEMBL2158686)
Affinity DataKi:  1.65E+4nMAssay Description:Inhibition of SK2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50041978(CHEMBL3134157)
Affinity DataIC50:  28nMAssay Description:Inhibition of recombinant SK1 (unknown origin) using sphingosine and [gamma-32P]ATP as substrate after 30 minsMore data for this Ligand-Target Pair
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443384(CHEMBL3086799)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of recombinant sphingosine kinase 1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50473216(CHEMBL1315457)
Affinity DataIC50:  2.60E+3nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50473214(CHEMBL2113330)
Affinity DataIC50:  2.80E+3nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443387(CHEMBL3086811)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of recombinant sphingosine kinase 1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins in presence of...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C alpha type(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50473219(CHEMBL2113338)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of human recombinant PKCalphaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSphingosine kinase 2(Homo sapiens (Human))
The City University Of New York

Curated by ChEMBL
LigandPNGBDBM50443383(CHEMBL3086796)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of sphingosine kinase 2 (unknown origin) using sphingosine as substrate after 30 mins in presence of [gamma32P]-ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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