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Found 14 with Last Name = 'bobrov' and Initial = 'm'
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  90nMAssay Description:Binding affinity of the compound towards Cannabinoid receptor 1 in rat forebrain membranes using [3H]-CP-55,940 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50128915((8Z,11Z,14Z)-1-Hydroxy-tricosa-8,11,14,17-tetraen-...)
Affinity DataKi:  360nMAssay Description:Binding affinity of the compound towards Cannabinoid receptor 1 in rat forebrain membranes using [3H]-CP-55,940 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM20462((5Z,8Z,11Z,14Z)-N-[2-(3,4-dihydroxyphenyl)ethyl]ic...)
Affinity DataKi:  380nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50096883((5Z,8Z,11Z,14Z,17Z)-Icosa-5,8,11,14,17-pentaenoic ...)
Affinity DataKi:  620nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  800nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50096881((10Z,13Z,16Z,19Z)-Docosa-7,10,13,16,19-pentaenoic ...)
Affinity DataKi:  1.37E+3nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50096882((5Z,9Z,12Z)-Octadeca-5,9,12-trienoic acid [2-(3,4-...)
Affinity DataKi:  1.72E+3nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50128912((5Z,8Z,11Z)-2,2-Dimethyl-icosa-5,8,11,14-tetraenoi...)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity of the compound towards Fatty-acid amide hydrolase (FAAH) in rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50128914((12Z,15Z)-1-Hydroxy-henicosa-12,15-dien-4-one | CH...)
Affinity DataKi:  2.10E+3nMAssay Description:Binding affinity of the compound towards Cannabinoid receptor 1 in rat forebrain membranes using [3H]-CP-55,940 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50096885((6Z,9Z,12Z,15Z)-Octadeca-6,9,12,15-tetraenoic acid...)
Affinity DataKi:  2.43E+3nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFatty-acid amide hydrolase 1 [30-579](Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM22988((5Z,8Z,11Z,14Z)-N-(2-hydroxyethyl)icosa-5,8,11,14-...)
Affinity DataKi:  3.00E+3nMAssay Description:Binding affinity of the compound towards Fatty-acid amide hydrolase (FAAH) in rat forebrain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50096884((9Z,12Z,15Z)-Octadeca-9,12,15-trienoic acid [2-(3,...)
Affinity DataKi:  3.13E+3nMAssay Description:Concentration required to displace 0.4 nM [3H]-SR-141,716A from CB1 receptor in rat brain preparations in the presence of 0.1 mM phenylmethyl sulphon...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50128912((5Z,8Z,11Z)-2,2-Dimethyl-icosa-5,8,11,14-tetraenoi...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity of the compound towards Cannabinoid receptor 1 in rat forebrain membranes using [3H]-CP-55,940 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Rattus norvegicus (rat))
Umr Cnrs 5074

Curated by ChEMBL
LigandPNGBDBM50128913((5Z,8Z,11Z)-Icosa-5,8,11,14-tetraenoic acid 2-hydr...)
Affinity DataKi: >1.00E+4nMAssay Description:Binding affinity of the compound towards Cannabinoid receptor 1 in rat forebrain membranes using [3H]-CP-55,940 as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed