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Found 38 with Last Name = 'bolte' and Initial = 'm'
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50283374(CHEMBL4169273)
Affinity DataKi:  1.10E+3nMAssay Description:Non-competitive inhibition of mushroom tyrosinase using L-DOPA as substrate preincubated for 10 mins followed by substrate addition measured up to 5 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187512(CHEMBL3827984)
Affinity DataIC50:  1.23E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187562(CHEMBL3827593)
Affinity DataIC50:  1.34E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50283374(CHEMBL4169273)
Affinity DataIC50:  1.57E+3nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrate preincubated for 10 mins followed by substrate addition measured for 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187561(CHEMBL3827501)
Affinity DataIC50:  1.92E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187558(CHEMBL3828565)
Affinity DataIC50:  2.11E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50283383(CHEMBL4173772)
Affinity DataIC50:  2.32E+3nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrate preincubated for 10 mins followed by substrate addition measured for 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187551(CHEMBL3828756)
Affinity DataIC50:  2.86E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187554(CHEMBL3827183)
Affinity DataIC50:  2.91E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187559(CHEMBL3827899)
Affinity DataIC50:  3.24E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50283382(CHEMBL4176197)
Affinity DataIC50:  3.37E+3nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrate preincubated for 10 mins followed by substrate addition measured for 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187583(CHEMBL3828346)
Affinity DataIC50:  3.64E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187516(CHEMBL3827414)
Affinity DataIC50:  3.79E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187511(CHEMBL3827344)
Affinity DataIC50:  4.45E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187564(CHEMBL3827068)
Affinity DataIC50:  5.38E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187550(CHEMBL3827341)
Affinity DataIC50:  5.58E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187514(CHEMBL3827052)
Affinity DataIC50:  6.32E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50283437(CHEMBL4162005)
Affinity DataIC50:  6.46E+3nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrate preincubated for 10 mins followed by substrate addition measured for 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187581(CHEMBL3828387)
Affinity DataIC50:  6.53E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187552(CHEMBL3828020)
Affinity DataIC50:  7.04E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187582(CHEMBL3828309)
Affinity DataIC50:  7.41E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50283385(CHEMBL4177122)
Affinity DataIC50:  7.75E+3nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrate preincubated for 10 mins followed by substrate addition measured for 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50283438(CHEMBL4172660)
Affinity DataIC50:  7.99E+3nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrate preincubated for 10 mins followed by substrate addition measured for 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187515(CHEMBL3827835)
Affinity DataIC50:  8.59E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187563(CHEMBL3828544)
Affinity DataIC50:  9.72E+3nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50283440(CHEMBL4176054)
Affinity DataIC50:  1.01E+4nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrate preincubated for 10 mins followed by substrate addition measured for 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187560(CHEMBL3827717)
Affinity DataIC50:  1.17E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187510(CHEMBL3827287)
Affinity DataIC50:  1.24E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187553(CHEMBL3828203)
Affinity DataIC50:  1.26E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187557(CHEMBL3828702)
Affinity DataIC50:  1.43E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50031467(5-HYDROXY-2-(HYDROXYMETHYL)-4H-PYRAN-4-ONE | 5-Hyd...)
Affinity DataIC50:  1.61E+4nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrate preincubated for 10 mins followed by substrate addition measured for 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187556(CHEMBL1448267)
Affinity DataIC50:  1.64E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50283439(CHEMBL4165446)
Affinity DataIC50:  1.66E+4nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrate preincubated for 10 mins followed by substrate addition measured for 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187555(CHEMBL3827841)
Affinity DataIC50:  1.75E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50283384(CHEMBL4165846)
Affinity DataIC50:  1.95E+4nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrate preincubated for 10 mins followed by substrate addition measured for 20 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPolyphenol oxidase 2(Agaricus bisporus (Common mushroom))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50283441(CHEMBL4168871)
Affinity DataIC50:  1.97E+4nMAssay Description:Inhibition of mushroom tyrosinase using L-DOPA as substrate preincubated for 10 mins followed by substrate addition measured for 20 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50187513(CHEMBL3827087)
Affinity DataIC50:  2.01E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUrease(Canavalia ensiformis (Jack bean) (Horse bean))
Quaid-I-Azam University

Curated by ChEMBL
LigandPNGBDBM50229993(2-thiourea | CHEMBL260876 | Thiocarbamid | Thiohar...)
Affinity DataIC50:  2.23E+4nMAssay Description:Inhibition of jack bean urease using urea as substrate assessed as reduction in ammonia production after 30 mins by indophenol methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed