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Found 574 with Last Name = 'bolton' and Initial = 's'
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225074((1S,3S,5S)-2-[(S)-2-amino-2-(3-hydroxy-adamantan-1...)
Affinity DataKi:  0.600nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225073((S)-2-amino-1-(1S,5R)-2-aza-bicyclo[3.1.0]hex-2-yl...)
Affinity DataKi:  2.90nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225053(2-(S)-amino-1-(1S,5R)-2-aza-bicyclo[3.1.0]hex-2-yl...)
Affinity DataKi:  10nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225049(2-(S)-amino-1-(1S,5R)-2-aza-bicyclo[3.1.0]hex-2-yl...)
Affinity DataKi:  14nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225050((S)-2-amino-2-(3-hydroxy-adamantan-1-yl)-1-thiazol...)
Affinity DataKi:  28nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225045((S)-2-amino-2-(3-hydroxy-adamantan-1-yl)-1-pyrroli...)
Affinity DataKi:  49nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225076((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi:  112nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225055((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi:  152nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225070((S)-2-amino-1-(3-aza-bicyclo[3.1.0]hex-3-yl)-2-(3,...)
Affinity DataKi:  270nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225071((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi:  356nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225077((2S,3S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)...)
Affinity DataKi:  530nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225051((S)-2-amino-2-(3-hydroxy-5,7-dimethyl-adamantan-1-...)
Affinity DataKi:  607nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225044((2S,3R)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)...)
Affinity DataKi:  731nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225060((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi:  877nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225058((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi:  1.01E+3nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225075((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi:  1.07E+3nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225046((S)-2-amino-2-(3-hydroxy-adamantan-1-yl)-1-(1H-iso...)
Affinity DataKi:  1.42E+3nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225059(2-(S)-amino-1-(1R,5R)-2-aza-bicyclo[3.1.0]hex-2-yl...)
Affinity DataKi:  1.94E+3nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225061((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi:  3.01E+3nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225042(1-(1S,5R)-2-aza-bicyclo[3.1.0]hex-2-yl-2-(3-hydrox...)
Affinity DataKi:  3.08E+3nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225065((S)-2-amino-1-(1S,5R)-2-aza-bicyclo[3.1.0]hex-2-yl...)
Affinity DataKi:  3.26E+3nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225057((S)-2-amino-1-(4,5-dihydro-pyrazol-1-yl)-2-(3-hydr...)
Affinity DataKi:  3.31E+3nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225040((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi:  3.65E+3nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225066((S)-2-amino-2-(3-hydroxy-adamantan-1-yl)-1-(2-meth...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225063((S)-4-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-3-a...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225068((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225069((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225048((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225067((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225043((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225041(CHEMBL236097 | N-((S)-6-((1S,5R)-2-aza-bicyclo[3.1...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225072((S)-1-((1R,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225039((S)-2-amino-3,3-dimethyl-1-(pyrazolidin-1-yl)butan...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225062((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225064((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2,5...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225047((2S,3R)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225054((S)-2-amino-1-(2,3-dihydro-indol-1-yl)-2-(3-hydrox...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225056((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetDipeptidyl peptidase 4(Homo sapiens (Human))
Bristol-Myers Squibb Research And Development

Curated by ChEMBL
LigandPNGBDBM50225052((S)-1-((1S,5R)-2-aza-bicyclo[3.1.0]hexan-2-yl)-2-a...)
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human DPP4More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50217812(CHEMBL322526)
Affinity DataIC50:  0.400nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50217626(CHEMBL322538)
Affinity DataIC50:  0.700nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50217627(CHEMBL110061)
Affinity DataIC50:  0.700nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50217622(CHEMBL443539)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50217599(CHEMBL109888)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50144582((R)-1-[4-(6-Naphthalen-2-yl-hexanoyl)-piperazine-1...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase delta(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50217801(CHEMBL111250)
Affinity DataIC50:  1nMAssay Description:In vitro inhibition of human tryptase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50144577((R)-1-[4-(6-Naphthalen-1-yl-hexanoyl)-piperazine-1...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50144555((R)-1-{4-[2-(4-Benzyloxy-phenyl)-acetyl]-piperazin...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50144586((R)-1-[4-(7-Naphthalen-1-yl-heptanoyl)-piperazine-...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity against human tryptaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTryptase beta-2/delta/gamma(Homo sapiens (Human))
The Bristol-Myers Squibb Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50144535((2S,3R)-4-Oxo-1-[4-(6-phenyl-hexanoyl)-piperazine-...)
Affinity DataIC50:  1nMAssay Description:Inhibitory activity of compound against human tryptase was determinedMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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