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Found 502 with Last Name = 'bostrom' and Initial = 'll'
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM12751(1-(3-carbamimidoylphenyl)-3-methyl-N-[4-(2-sulfamo...)
Affinity DataKi:  0.0130nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50097624(3-(3-Carbamimidoyl-phenyl)-3H-[1,2,3]triazole-4-ca...)
Affinity DataKi:  0.0230nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM12751(1-(3-carbamimidoylphenyl)-3-methyl-N-[4-(2-sulfamo...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity towards Rabbit Coagulation factor X in a rabbit arterio-venous (A-V) shunt modelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Oryctolagus cuniculus)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM12751(1-(3-carbamimidoylphenyl)-3-methyl-N-[4-(2-sulfamo...)
Affinity DataKi:  0.0300nMAssay Description:Binding affinity towards human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50097626(1-(3-Carbamimidoyl-phenyl)-1H-tetrazole-5-carboxyl...)
Affinity DataKi:  0.0370nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50369433(CHEMBL1202108)
Affinity DataKi:  0.0400nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProthrombin(Homo sapiens (Human))
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50369433(CHEMBL1202108)
Affinity DataKi:  0.0450nMAssay Description:The binding affinity towards thrombin obtained from human purified enzymes.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50097625(4-(3-Carbamimidoyl-phenyl)-2-methyl-thiazole-5-car...)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity towards Rabbit Coagulation factor X in a rabbit arterio-venous (A-V) shunt modelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Oryctolagus cuniculus)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50097625(4-(3-Carbamimidoyl-phenyl)-2-methyl-thiazole-5-car...)
Affinity DataKi:  0.0800nMAssay Description:Binding affinity towards human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50087536(3-(3-Carbamimidoyl-phenyl)-isoxazole-4-carboxylic ...)
Affinity DataKi:  0.100nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50087533(3-(3-Carbamimidoyl-phenyl)-isoxazole-4-carboxylic ...)
Affinity DataKi:  0.150nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM12657(1-[3-(Aminomethyl)phenyl]-N-[3-fluoro-2-(methylsul...)
Affinity DataKi:  0.150nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50087533(3-(3-Carbamimidoyl-phenyl)-isoxazole-4-carboxylic ...)
Affinity DataKi:  0.150nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50096095(2-(3-Carbamimidoyl-phenyl)-2H-pyrazole-3-carboxyli...)
Affinity DataKi:  0.160nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50097620(3-(3-Carbamimidoyl-phenyl)-1-methyl-1H-pyrazole-4-...)
Affinity DataKi:  0.200nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM12657(1-[3-(Aminomethyl)phenyl]-N-[3-fluoro-2-(methylsul...)
Affinity DataKi:  0.300nMAssay Description:Tested in vitro for inhibition of rabbit Coagulation factor XMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50097619(1-(3-Carbamimidoyl-phenyl)-4-methyl-1H-imidazole-2...)
Affinity DataKi:  0.300nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50097621(1-(3-Carbamimidoyl-phenyl)-1H-imidazole-2-carboxyl...)
Affinity DataKi:  0.330nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Oryctolagus cuniculus)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087533(3-(3-Carbamimidoyl-phenyl)-isoxazole-4-carboxylic ...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity towards human trypsinMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Oryctolagus cuniculus)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087533(3-(3-Carbamimidoyl-phenyl)-isoxazole-4-carboxylic ...)
Affinity DataKi:  0.400nMAssay Description:Inhibitory activity of the compound was tested against rabbit Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50097632(4-(3-Carbamimidoyl-phenyl)-2-methyl-oxazole-5-carb...)
Affinity DataKi:  0.400nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135953(2-(2-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  0.460nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50087540(3-(3-Carbamimidoyl-phenyl)-5-hydroxymethyl-isoxazo...)
Affinity DataKi:  0.5nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135943(2-(2-Aminomethyl-4-methoxy-phenyl)-5-trifluorometh...)
Affinity DataKi:  0.540nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50087538((4S,5S)-3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl...)
Affinity DataKi:  0.550nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50087532(3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl-isoxazo...)
Affinity DataKi:  0.630nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Oryctolagus cuniculus)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50087538((4S,5S)-3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl...)
Affinity DataKi:  0.640nMAssay Description:Inhibitory activity of the compound was tested against rabbit Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50087535(3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl-isoxazo...)
Affinity DataKi:  0.75nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50096084(1-(3-Carbamimidoyl-phenyl)-1H-pyrrole-2-carboxylic...)
Affinity DataKi:  0.800nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Oryctolagus cuniculus)
Dupont Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50079252(3-(3-Carbamimidoyl-phenyl)-5-methoxymethyl-4,5-dih...)
Affinity DataKi:  0.800nMAssay Description:Inhibitory activity of the compound was tested against rabbit Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50097631(4-(3-Carbamimidoyl-phenyl)-thiazole-5-carboxylic a...)
Affinity DataKi:  0.820nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50079211(CHEMBL327404 | {3-(3-Carbamimidoyl-phenyl)-5-[5-(2...)
Affinity DataKi:  0.830nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50079211(CHEMBL327404 | {3-(3-Carbamimidoyl-phenyl)-5-[5-(2...)
Affinity DataKi:  0.830nMAssay Description:Binding affinity to purified human coagulation factor Xa (FXa)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135960(2-(2-Aminomethyl-4-methoxy-phenyl)-5-trifluorometh...)
Affinity DataKi:  0.880nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135945(1-[2-(aminomethyl)phenyl]-N-(3-fluoro-2'-sulfamoyl...)
Affinity DataKi:  0.910nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50097627(2-(3-Carbamimidoyl-phenyl)-N-(2'-sulfamoyl-bipheny...)
Affinity DataKi:  1nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135966(2-(2-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  1nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50097630(3-(3-Carbamimidoyl-phenyl)-3H-imidazole-4-carboxyl...)
Affinity DataKi:  1.10nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50079236(3-(3-Carbamimidoyl-phenyl)-5-tetrazol-1-ylmethyl-4...)
Affinity DataKi:  1.60nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135961(2-(2-Aminomethyl-4-methoxy-phenyl)-5-trifluorometh...)
Affinity DataKi:  1.70nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135951(2-(2-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  1.80nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50087539((4S,5R)-3-(3-Carbamimidoyl-phenyl)-5-methyl-4,5-di...)
Affinity DataKi:  1.80nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50087537((4S,5S)-3-(3-Carbamimidoyl-phenyl)-5-tetrazol-1-yl...)
Affinity DataKi:  2.30nMAssay Description:Inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50097622(5-(3-Carbamimidoyl-phenyl)-2-oxo-2,3-dihydro-1H-im...)
Affinity DataKi:  2.30nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135954(2-(2-Aminomethyl-4-methoxy-phenyl)-5-trifluorometh...)
Affinity DataKi:  2.40nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50097628(5-(3-Carbamimidoyl-phenyl)-oxazole-4-carboxylic ac...)
Affinity DataKi:  2.5nMAssay Description:Binding affinity towards human Serine protease FXaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135966(2-(2-Aminomethyl-phenyl)-5-trifluoromethyl-2H-pyra...)
Affinity DataKi:  2.60nMAssay Description:Tested in vitro for inhibition of rabbit Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM18965(1-[3-(aminomethyl)phenyl]-3-methyl-N-[4-(2-sulfamo...)
Affinity DataKi:  2.70nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135962(2-(4-Methoxy-phenyl)-5-trifluoromethyl-2H-pyrazole...)
Affinity DataKi:  2.80nMAssay Description:Tested in vitro for inhibition of human Coagulation factor XMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCoagulation factor X(Homo sapiens (Human))
Pharmaceutical Research Institute

Curated by ChEMBL
LigandPNGBDBM50135945(1-[2-(aminomethyl)phenyl]-N-(3-fluoro-2'-sulfamoyl...)
Affinity DataKi:  2.90nMAssay Description:Tested in vitro for inhibition of rabbit Coagulation factor XMore data for this Ligand-Target Pair
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